ATE179708T1 - Chinazoline-derivate - Google Patents

Chinazoline-derivate

Info

Publication number
ATE179708T1
ATE179708T1 AT95937126T AT95937126T ATE179708T1 AT E179708 T1 ATE179708 T1 AT E179708T1 AT 95937126 T AT95937126 T AT 95937126T AT 95937126 T AT95937126 T AT 95937126T AT E179708 T1 ATE179708 T1 AT E179708T1
Authority
AT
Austria
Prior art keywords
pct
date
halogeno
oxo
sec
Prior art date
Application number
AT95937126T
Other languages
English (en)
Inventor
Andrew John Barker
Park
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Application granted granted Critical
Publication of ATE179708T1 publication Critical patent/ATE179708T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Seal Device For Vehicle (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
AT95937126T 1994-11-30 1995-11-28 Chinazoline-derivate ATE179708T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB9424233A GB9424233D0 (en) 1994-11-30 1994-11-30 Quinazoline derivatives

Publications (1)

Publication Number Publication Date
ATE179708T1 true ATE179708T1 (de) 1999-05-15

Family

ID=10765246

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95937126T ATE179708T1 (de) 1994-11-30 1995-11-28 Chinazoline-derivate

Country Status (8)

Country Link
US (1) US5955464A (de)
EP (1) EP0794953B1 (de)
JP (1) JP4012245B2 (de)
AT (1) ATE179708T1 (de)
AU (1) AU3933095A (de)
DE (1) DE69509553T2 (de)
GB (1) GB9424233D0 (de)
WO (1) WO1996016960A1 (de)

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TWI751517B (zh) 2019-04-17 2022-01-01 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TW202210480A (zh) 2019-04-17 2022-03-16 美商基利科學股份有限公司 類鐸受體調節劑之固體形式
TWI879779B (zh) 2019-06-28 2025-04-11 美商基利科學股份有限公司 類鐸受體調節劑化合物的製備方法

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Also Published As

Publication number Publication date
US5955464A (en) 1999-09-21
EP0794953B1 (de) 1999-05-06
JP4012245B2 (ja) 2007-11-21
DE69509553T2 (de) 1999-09-02
JPH10509972A (ja) 1998-09-29
WO1996016960A1 (en) 1996-06-06
EP0794953A1 (de) 1997-09-17
DE69509553D1 (de) 1999-06-10
GB9424233D0 (en) 1995-01-18
AU3933095A (en) 1996-06-19

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