AR231976A1 - Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(4h)-ona y de(7-1-hidroxi-2-amino-etil)-2-benzolinona,y nuevos compuestos intermedios para uso exclusivo en dicho procedimiento - Google Patents
Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(4h)-ona y de(7-1-hidroxi-2-amino-etil)-2-benzolinona,y nuevos compuestos intermedios para uso exclusivo en dicho procedimientoInfo
- Publication number
- AR231976A1 AR231976A1 AR290473A AR29047382A AR231976A1 AR 231976 A1 AR231976 A1 AR 231976A1 AR 290473 A AR290473 A AR 290473A AR 29047382 A AR29047382 A AR 29047382A AR 231976 A1 AR231976 A1 AR 231976A1
- Authority
- AR
- Argentina
- Prior art keywords
- etil
- hydroxi
- amino
- procedure
- benzolinone
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
- C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Feed For Specific Animals (AREA)
- Fodder In General (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19813134590 DE3134590A1 (de) | 1981-09-01 | 1981-09-01 | Neue benzo-heterocyclen |
Publications (1)
Publication Number | Publication Date |
---|---|
AR231976A1 true AR231976A1 (es) | 1985-04-30 |
Family
ID=6140603
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR290473A AR231976A1 (es) | 1981-09-01 | 1982-08-30 | Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(4h)-ona y de(7-1-hidroxi-2-amino-etil)-2-benzolinona,y nuevos compuestos intermedios para uso exclusivo en dicho procedimiento |
AR294856A AR231977A1 (es) | 1981-09-01 | 1983-11-17 | Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(44)-ona y de 7-(1-hidroxi-2-amino-etil)-2-benzoxazolinona |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR294856A AR231977A1 (es) | 1981-09-01 | 1983-11-17 | Procedimiento para la preparacion de derivados de 8-(1-hidroxi-2-amino-etil)-2h-1,4-benzoxazin-3-(44)-ona y de 7-(1-hidroxi-2-amino-etil)-2-benzoxazolinona |
Country Status (25)
Country | Link |
---|---|
EP (1) | EP0073505B1 (fi) |
JP (1) | JPS5852278A (fi) |
KR (1) | KR890000380B1 (fi) |
AR (2) | AR231976A1 (fi) |
AT (1) | ATE16703T1 (fi) |
AU (1) | AU553589B2 (fi) |
CA (1) | CA1180012A (fi) |
CS (1) | CS236679B2 (fi) |
DD (1) | DD204477A5 (fi) |
DE (2) | DE3134590A1 (fi) |
DK (1) | DK158664C (fi) |
ES (3) | ES8308318A1 (fi) |
FI (1) | FI78475C (fi) |
GB (1) | GB2106105B (fi) |
GR (1) | GR77275B (fi) |
HU (1) | HU186112B (fi) |
IE (1) | IE53615B1 (fi) |
IL (1) | IL66683A0 (fi) |
NO (1) | NO157738C (fi) |
NZ (1) | NZ201777A (fi) |
PL (1) | PL139375B1 (fi) |
PT (1) | PT75478A (fi) |
SU (1) | SU1149876A3 (fi) |
YU (1) | YU42794B (fi) |
ZA (1) | ZA826349B (fi) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4554284A (en) * | 1984-09-12 | 1985-11-19 | Smithkline Beckman Corporation | 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones |
DE3743265A1 (de) * | 1987-12-19 | 1989-06-29 | Boehringer Ingelheim Kg | Neue ammoniumverbindungen, ihre herstellung und verwendung |
TW372967B (en) * | 1994-12-27 | 1999-11-01 | Kanebo Ltd | 1,4 benzoxazine derivative, pharmaceutical composition containing the same and use thereof |
US7056916B2 (en) | 2002-11-15 | 2006-06-06 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Medicaments for the treatment of chronic obstructive pulmonary disease |
DE10253282A1 (de) * | 2002-11-15 | 2004-05-27 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Arzneimittel zur Behandlung von chronisch obstruktiver Lungenerkrankung |
PE20040950A1 (es) | 2003-02-14 | 2005-01-01 | Theravance Inc | DERIVADOS DE BIFENILO COMO AGONISTAS DE LOS RECEPTORES ADRENERGICOS ß2 Y COMO ANTAGONISTAS DE LOS RECEPTORES MUSCARINICOS |
GB0307856D0 (en) * | 2003-04-04 | 2003-05-14 | Novartis Ag | Organic compounds |
BRPI0409198A (pt) | 2003-04-04 | 2006-05-02 | Novartis Ag | derivados quinolin-2-ona para o tratamento de doenças de vias aéreas |
CA2565243A1 (en) * | 2004-05-13 | 2005-11-24 | Boehringer Ingelheim International Gmbh | Hydroxy-substituted benzo-condensed heterocycles for use as beta agonists in the treatment of respiratory diseases |
US7307076B2 (en) | 2004-05-13 | 2007-12-11 | Boehringer Ingelheim International Gmbh | Beta agonists for the treatment of respiratory diseases |
DE102004024453A1 (de) * | 2004-05-14 | 2006-01-05 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue langwirksame Bronchodilatoren zur Behandlung von Atemwegserkrankungen |
US7220742B2 (en) | 2004-05-14 | 2007-05-22 | Boehringer Ingelheim International Gmbh | Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments |
DE102004024452A1 (de) * | 2004-05-14 | 2005-12-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Aerosolformulierung für die Inhalation von Betaagonisten |
DE102004024454A1 (de) * | 2004-05-14 | 2005-12-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Enantiomerenreine Betaagonisten, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel |
US7745621B2 (en) | 2004-05-14 | 2010-06-29 | Boehringer Ingelheim International Gmbh | Long acting bronchodilators for the treatment of respiratory diseases |
DE102004024451A1 (de) | 2004-05-14 | 2005-12-22 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Pulverformulierungen für die Inhalation, die Enantiomerenreine Betaagonisten enthalten |
MX2008001976A (es) * | 2005-08-15 | 2008-03-25 | Boehringer Ingelheim Int | Procedimiento para la preparacion de betamimeticos. |
US20070088030A1 (en) | 2005-10-10 | 2007-04-19 | Barbara Niklaus-Humke | Aerosol formulations for the inhalation of beta-agonists |
GB0602778D0 (en) | 2006-02-10 | 2006-03-22 | Glaxo Group Ltd | Novel compound |
WO2008017638A1 (de) * | 2006-08-07 | 2008-02-14 | Boehringer Ingelheim International Gmbh | Enantiomerenreine betaagonisten, verfahren zu deren herstellung und deren verwendung als arzneimittel |
UY30543A1 (es) * | 2006-08-18 | 2008-03-31 | Boehringer Ingelheim Int | Formulacion de aerosol para la inhalacion de beta- agonistas |
BRPI0807806A2 (pt) * | 2007-01-25 | 2014-06-17 | Boehringer Ingelheim Int | " processo para a fabricação de beta-miméticos ". |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2035749A1 (fi) * | 1969-02-06 | 1970-12-24 | Bellon Labor Sa Roger | |
DE2429253A1 (de) * | 1974-06-19 | 1976-01-15 | Boehringer Sohn Ingelheim | Phenylalkanolamine |
-
1981
- 1981-09-01 DE DE19813134590 patent/DE3134590A1/de not_active Withdrawn
-
1982
- 1982-08-27 SU SU823483451A patent/SU1149876A3/ru active
- 1982-08-28 AT AT82107919T patent/ATE16703T1/de not_active IP Right Cessation
- 1982-08-28 DE DE8282107919T patent/DE3267702D1/de not_active Expired
- 1982-08-28 EP EP82107919A patent/EP0073505B1/de not_active Expired
- 1982-08-30 FI FI822985A patent/FI78475C/fi not_active IP Right Cessation
- 1982-08-30 PT PT75478A patent/PT75478A/pt not_active IP Right Cessation
- 1982-08-30 YU YU1949/82A patent/YU42794B/xx unknown
- 1982-08-30 PL PL1982238077A patent/PL139375B1/pl unknown
- 1982-08-30 AR AR290473A patent/AR231976A1/es active
- 1982-08-30 DD DD82242881A patent/DD204477A5/de unknown
- 1982-08-31 GR GR69166A patent/GR77275B/el unknown
- 1982-08-31 DK DK389082A patent/DK158664C/da not_active IP Right Cessation
- 1982-08-31 GB GB08224810A patent/GB2106105B/en not_active Expired
- 1982-08-31 IE IE2105/82A patent/IE53615B1/en not_active IP Right Cessation
- 1982-08-31 NZ NZ201777A patent/NZ201777A/en unknown
- 1982-08-31 CS CS826329A patent/CS236679B2/cs unknown
- 1982-08-31 HU HU822793A patent/HU186112B/hu not_active IP Right Cessation
- 1982-08-31 NO NO822932A patent/NO157738C/no unknown
- 1982-08-31 AU AU87874/82A patent/AU553589B2/en not_active Ceased
- 1982-08-31 JP JP57151626A patent/JPS5852278A/ja active Granted
- 1982-08-31 ZA ZA826349A patent/ZA826349B/xx unknown
- 1982-08-31 ES ES515380A patent/ES8308318A1/es not_active Expired
- 1982-08-31 IL IL66683A patent/IL66683A0/xx not_active IP Right Cessation
- 1982-08-31 CA CA000410462A patent/CA1180012A/en not_active Expired
- 1982-09-01 KR KR8203945A patent/KR890000380B1/ko active
-
1983
- 1983-04-27 ES ES521870A patent/ES8402279A1/es not_active Expired
- 1983-04-27 ES ES521871A patent/ES521871A0/es active Granted
- 1983-11-17 AR AR294856A patent/AR231977A1/es active
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