AR231638A1 - Procedimiento para obtener compuestos de 1-1-2-(1,4-benzoxatio o 1,4-benzoxatian o 1,4-benzodioxan-2-il)-alquilen-4-piperidil-2-imidazolinona,2-hexahidro-pirimidinona o 2-imino-imidazolidina - Google Patents
Procedimiento para obtener compuestos de 1-1-2-(1,4-benzoxatio o 1,4-benzoxatian o 1,4-benzodioxan-2-il)-alquilen-4-piperidil-2-imidazolinona,2-hexahidro-pirimidinona o 2-imino-imidazolidinaInfo
- Publication number
- AR231638A1 AR231638A1 AR282944A AR28294480A AR231638A1 AR 231638 A1 AR231638 A1 AR 231638A1 AR 282944 A AR282944 A AR 282944A AR 28294480 A AR28294480 A AR 28294480A AR 231638 A1 AR231638 A1 AR 231638A1
- Authority
- AR
- Argentina
- Prior art keywords
- pirimidinone
- benzoxatio
- benzoxatian
- piperidil
- benzodioxan
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Psychiatry (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US88808978A | 1978-03-20 | 1978-03-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR231638A1 true AR231638A1 (es) | 1985-01-31 |
Family
ID=25392505
Family Applications (4)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR275879A AR227272A1 (es) | 1978-03-20 | 1979-03-20 | Procedimiento para la obtencion de compuestos de n-oxaciclil-alquil-piperidil-diaza y sus sales |
AR282944A AR231638A1 (es) | 1978-03-20 | 1980-10-20 | Procedimiento para obtener compuestos de 1-1-2-(1,4-benzoxatio o 1,4-benzoxatian o 1,4-benzodioxan-2-il)-alquilen-4-piperidil-2-imidazolinona,2-hexahidro-pirimidinona o 2-imino-imidazolidina |
AR282945A AR227400A1 (es) | 1978-03-20 | 1980-10-20 | Procedimiento para obtener n-oxaciclil-alquil-piperidinas y sus sales |
AR282946A AR227527A1 (es) | 1978-03-20 | 1980-10-20 | Procedimiento para la elaboracion de nuevos compuestos n-oxaciclilalquil-piperidil-diazoicos |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR275879A AR227272A1 (es) | 1978-03-20 | 1979-03-20 | Procedimiento para la obtencion de compuestos de n-oxaciclil-alquil-piperidil-diaza y sus sales |
Family Applications After (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR282945A AR227400A1 (es) | 1978-03-20 | 1980-10-20 | Procedimiento para obtener n-oxaciclil-alquil-piperidinas y sus sales |
AR282946A AR227527A1 (es) | 1978-03-20 | 1980-10-20 | Procedimiento para la elaboracion de nuevos compuestos n-oxaciclilalquil-piperidil-diazoicos |
Country Status (20)
Country | Link |
---|---|
EP (1) | EP0004358B1 (es) |
JP (1) | JPS54157570A (es) |
AR (4) | AR227272A1 (es) |
AT (1) | AT372088B (es) |
AU (1) | AU529838B2 (es) |
DD (1) | DD142341A5 (es) |
DE (1) | DE2961738D1 (es) |
DK (1) | DK113079A (es) |
ES (4) | ES478662A1 (es) |
FI (1) | FI66373C (es) |
GB (1) | GB2019837B (es) |
GR (1) | GR71865B (es) |
HU (1) | HU182941B (es) |
IL (1) | IL56908A (es) |
MY (1) | MY8700122A (es) |
NO (1) | NO150202C (es) |
NZ (1) | NZ189939A (es) |
PL (1) | PL116514B1 (es) |
PT (1) | PT69369A (es) |
ZA (2) | ZA79417B (es) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4329348A (en) * | 1979-02-26 | 1982-05-11 | Ciba-Geigy Corporation | N-Oxacyclic-alkylpiperidines as psychostimulants |
DE3124366A1 (de) * | 1981-06-20 | 1982-12-30 | Hoechst Ag, 6000 Frankfurt | N-oxacyclyl-alkylpiperidin-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und deren verwendung |
FR2524887A1 (fr) * | 1982-04-08 | 1983-10-14 | Bouchara Emile | Nouvelles cyanoguanidines, leur procede d'obtention et les compositions pharmaceutiques en renfermant |
FR2525600A1 (fr) * | 1982-04-21 | 1983-10-28 | Bouchara Emile | Nouvelles carboxamidoguanidines, leur procede d'obtention et les compositions pharmaceutiques en renfermant |
US4556660A (en) * | 1982-07-12 | 1985-12-03 | Janssen Pharmaceutica N.V. | N-(Bicyclic heterocyclyl)-4-piperidinamines |
JP2807577B2 (ja) * | 1990-06-15 | 1998-10-08 | エーザイ株式会社 | 環状アミド誘導体 |
SI9300097B (en) * | 1992-02-27 | 2001-12-31 | Janssen Pharmaceutica Nv | (benzodioxan, benzofuran or benzopyran) alkylamino) alkyl substituted guanidines |
US5703115A (en) * | 1993-02-19 | 1997-12-30 | Janssen Pharmaceutica, N.V. | (benzodioxan, benzofuran or benzopyran) alkylamino! alkyl substituted guanidines |
US6133277A (en) * | 1997-12-05 | 2000-10-17 | Janssen Pharmaceutica N.V. | (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties |
JP2003501428A (ja) | 1999-06-02 | 2003-01-14 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | ピロリジニル、ピペリジニルもしくはホモピペリジニル置換(ベンゾジオキサン、ベンゾフランもしくはベンゾピラン)誘導体 |
BR0011237A (pt) * | 1999-06-02 | 2002-03-05 | Janssen Pharmaceutica Nv | Derivados de benzodioxano, benzofurano ou benzopirano substituìdos com aminoalquila |
JO2352B1 (en) * | 2000-06-22 | 2006-12-12 | جانسين فارماسيوتيكا ان. في | Compounds for the treatment of non-adaptation of the bottom of the uterus |
BRPI0608353A2 (pt) | 2005-02-17 | 2009-12-01 | Wyeth Corp | derivados de indol, benzotiofeno, benzofurano e indeno cicloalquilfundidos |
CN114920686B (zh) * | 2022-05-20 | 2023-11-24 | 山东农业大学 | 5-(苯磺酰基)-n-哌啶-4-基-2-(三氟甲基)苯磺酰胺盐酸盐的合成方法 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3910930A (en) * | 1973-01-04 | 1975-10-07 | Janssen Pharmaceutica Nv | 1-{55 1-{8 2-(1,4-Benzodioxan-2-yl)-2-hydroxyethyl{9 -4-piperidyl{56 -2-benzimidazolinones |
-
1977
- 1977-08-17 GR GR58624A patent/GR71865B/el unknown
-
1979
- 1979-01-31 ZA ZA79417A patent/ZA79417B/xx unknown
- 1979-03-15 ES ES478662A patent/ES478662A1/es not_active Expired
- 1979-03-15 GB GB7909231A patent/GB2019837B/en not_active Expired
- 1979-03-16 DE DE7979100815T patent/DE2961738D1/de not_active Expired
- 1979-03-16 FI FI790894A patent/FI66373C/fi not_active IP Right Cessation
- 1979-03-16 EP EP79100815A patent/EP0004358B1/de not_active Expired
- 1979-03-17 PL PL1979214206A patent/PL116514B1/pl unknown
- 1979-03-19 HU HU79CI1923A patent/HU182941B/hu unknown
- 1979-03-19 AT AT0204479A patent/AT372088B/de not_active IP Right Cessation
- 1979-03-19 NO NO790917A patent/NO150202C/no unknown
- 1979-03-19 NZ NZ189939A patent/NZ189939A/xx unknown
- 1979-03-19 DD DD79211661A patent/DD142341A5/de unknown
- 1979-03-19 IL IL56908A patent/IL56908A/xx unknown
- 1979-03-19 PT PT69369A patent/PT69369A/pt unknown
- 1979-03-19 AU AU45243/79A patent/AU529838B2/en not_active Ceased
- 1979-03-19 ZA ZA791276A patent/ZA791276B/xx unknown
- 1979-03-19 DK DK113079A patent/DK113079A/da not_active Application Discontinuation
- 1979-03-20 AR AR275879A patent/AR227272A1/es active
- 1979-03-20 JP JP3184279A patent/JPS54157570A/ja active Pending
- 1979-09-28 ES ES484571A patent/ES484571A1/es not_active Expired
- 1979-09-28 ES ES484570A patent/ES484570A1/es not_active Expired
- 1979-09-28 ES ES484572A patent/ES484572A1/es not_active Expired
-
1980
- 1980-10-20 AR AR282944A patent/AR231638A1/es active
- 1980-10-20 AR AR282945A patent/AR227400A1/es active
- 1980-10-20 AR AR282946A patent/AR227527A1/es active
-
1987
- 1987-12-30 MY MY122/87A patent/MY8700122A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
PL214206A1 (es) | 1980-02-25 |
ES478662A1 (es) | 1980-01-16 |
ATA204479A (de) | 1983-01-15 |
IL56908A (en) | 1983-09-30 |
NO790917L (no) | 1979-09-21 |
AR227400A1 (es) | 1982-10-29 |
GR71865B (es) | 1983-07-07 |
AU4524379A (en) | 1979-09-27 |
PT69369A (en) | 1979-04-01 |
AT372088B (de) | 1983-08-25 |
ZA791276B (en) | 1980-03-26 |
AR227272A1 (es) | 1982-10-15 |
EP0004358A1 (de) | 1979-10-03 |
NO150202B (no) | 1984-05-28 |
NO150202C (no) | 1984-09-05 |
MY8700122A (en) | 1987-12-31 |
IL56908A0 (en) | 1979-05-31 |
DE2961738D1 (en) | 1982-02-25 |
GB2019837A (en) | 1979-11-07 |
DK113079A (da) | 1979-09-21 |
ZA79417B (en) | 1980-01-30 |
JPS54157570A (en) | 1979-12-12 |
ES484570A1 (es) | 1980-05-16 |
GB2019837B (en) | 1982-08-25 |
FI66373B (fi) | 1984-06-29 |
AR227527A1 (es) | 1982-11-15 |
HU182941B (en) | 1984-03-28 |
EP0004358B1 (de) | 1982-01-06 |
NZ189939A (en) | 1981-12-15 |
FI790894A (fi) | 1979-09-21 |
DD142341A5 (de) | 1980-06-18 |
PL116514B1 (en) | 1981-06-30 |
FI66373C (fi) | 1984-10-10 |
AU529838B2 (en) | 1983-06-23 |
ES484571A1 (es) | 1980-05-16 |
ES484572A1 (es) | 1980-05-16 |
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