MX6242E - Procedimiento para la preparacion de 1,2,3,5,tetrahidroimidazotienopirimidin-2-onas - Google Patents

Procedimiento para la preparacion de 1,2,3,5,tetrahidroimidazotienopirimidin-2-onas

Info

Publication number
MX6242E
MX6242E MX798313U MX831379U MX6242E MX 6242 E MX6242 E MX 6242E MX 798313 U MX798313 U MX 798313U MX 831379 U MX831379 U MX 831379U MX 6242 E MX6242 E MX 6242E
Authority
MX
Mexico
Prior art keywords
tetrahidroimidazotienopirimidin
onas
procedure
preparation
Prior art date
Application number
MX798313U
Other languages
English (en)
Inventor
Fumiyoshi Ishikawa
Shinichiro Ashida
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Publication of MX6242E publication Critical patent/MX6242E/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14Ortho-condensed systems
MX798313U 1978-08-11 1979-08-10 Procedimiento para la preparacion de 1,2,3,5,tetrahidroimidazotienopirimidin-2-onas MX6242E (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP9783278A JPS5527105A (en) 1978-08-11 1978-08-11 Imidazothienopyrimidinones compound

Publications (1)

Publication Number Publication Date
MX6242E true MX6242E (es) 1985-01-28

Family

ID=14202683

Family Applications (1)

Application Number Title Priority Date Filing Date
MX798313U MX6242E (es) 1978-08-11 1979-08-10 Procedimiento para la preparacion de 1,2,3,5,tetrahidroimidazotienopirimidin-2-onas

Country Status (16)

Country Link
US (1) US4284773A (es)
EP (1) EP0008408B1 (es)
JP (1) JPS5527105A (es)
AU (1) AU529068B2 (es)
CA (1) CA1116597A (es)
CS (1) CS219256B2 (es)
DE (1) DE2961552D1 (es)
DK (1) DK153844C (es)
ES (1) ES483289A1 (es)
GR (1) GR73839B (es)
IL (1) IL57923A (es)
MX (1) MX6242E (es)
PH (1) PH15530A (es)
SU (1) SU880252A3 (es)
YU (1) YU41170B (es)
ZA (1) ZA793909B (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4287340A (en) * 1979-08-27 1981-09-01 Warner-Lambert Company Dihydro-oxo-pyrido[1,2-a]thienopyrimidine compounds
ZW11781A1 (en) * 1980-06-27 1982-01-20 Hoffmann La Roche Pyrimidine derivatives
US7772188B2 (en) 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
US8304420B2 (en) 2006-11-28 2012-11-06 Shire Llc Substituted quinazolines for reducing platelet count
MX354786B (es) 2007-06-04 2018-03-21 Synergy Pharmaceuticals Inc Agonistas de guanilato ciclasa utiles para el tratamiento de trastornos gastrointestinales, inflamacion, cancer y otros trastornos.
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
GB0808950D0 (en) * 2008-05-16 2008-06-25 Shire Llc Substituted quinazolines
AU2009256157B2 (en) 2008-06-04 2014-12-18 Bausch Health Ireland Limited Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
ES2624828T3 (es) 2008-07-16 2017-07-17 Synergy Pharmaceuticals Inc. Agonistas de la guanilato ciclasa útiles para el tratamiento de trastornos gastrointestinales, inflamación, cáncer y otros
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
WO2012118972A2 (en) 2011-03-01 2012-09-07 Synegy Pharmaceuticals Inc. Process of preparing guanylate cyclase c agonists
EP3718557A3 (en) 2013-02-25 2020-10-21 Bausch Health Ireland Limited Guanylate cyclase receptor agonist sp-333 for use in colonic cleansing
AU2014235209B2 (en) 2013-03-15 2018-06-14 Bausch Health Ireland Limited Guanylate cyclase receptor agonists combined with other drugs
CA2905438A1 (en) 2013-03-15 2014-09-25 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase and their uses
CA2913737A1 (en) 2013-06-05 2014-12-11 Synergy Pharmaceuticals, Inc. Ultra-pure agonists of guanylate cyclase c, method of making and using same
CA2920856A1 (en) 2013-08-09 2015-02-12 Ardelyx, Inc. Ph modulating compounds for inhibiting gastrointestinal phosphate uptake
US20200368223A1 (en) 2019-05-21 2020-11-26 Ardelyx, Inc. Methods for inhibiting phosphate transport

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3890321A (en) * 1971-09-20 1975-06-17 Pfizer 6-aryl-5-ethyl-pyrimidin-4-ol compounds useful as intermediates and bronchodilators
US3932407A (en) * 1973-11-19 1976-01-13 Bristol-Myers Company Optionally substituted 1,2,3,5-tetrahydroimidezo(2,1-b)-quinazolin-2-ones and 6(H)-1,2,3,4-tetrahydropyimido(2,1-b)quinazolin-2-ones
DE2411273A1 (de) * 1974-03-06 1975-09-18 Schering Ag Neue thieno eckige klammer auf 2,3-d eckige klammer zu pyrimidinone und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
DK153844C (da) 1989-01-30
PH15530A (en) 1983-02-09
CA1116597A (en) 1982-01-19
DK336779A (da) 1980-02-12
IL57923A0 (en) 1979-11-30
GR73839B (es) 1984-05-04
DK153844B (da) 1988-09-12
SU880252A3 (ru) 1981-11-07
CS219256B2 (en) 1983-03-25
US4284773A (en) 1981-08-18
IL57923A (en) 1982-09-30
EP0008408B1 (en) 1981-12-09
AU4973579A (en) 1980-02-14
YU194779A (en) 1983-10-31
ES483289A1 (es) 1980-09-01
DE2961552D1 (en) 1982-02-04
JPS627914B2 (es) 1987-02-19
ZA793909B (en) 1980-10-29
AU529068B2 (en) 1983-05-26
JPS5527105A (en) 1980-02-27
EP0008408A1 (en) 1980-03-05
YU41170B (en) 1986-12-31

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