AR231638A1 - PROCEDURE FOR OBTAINING COMPOUNDS OF 1-1-2- (1,4-BENZOXATIO OR 1,4-BENZOXATIAN OR 1,4-BENZODIOXAN-2-IL) -ALKYLENE-4-PIPERIDIL-2-IMIDAZOLINONE, 2-HEXAHYDRO-PIRIMIDINONE OR 2-IMINO-IMIDAZOLIDINE - Google Patents
PROCEDURE FOR OBTAINING COMPOUNDS OF 1-1-2- (1,4-BENZOXATIO OR 1,4-BENZOXATIAN OR 1,4-BENZODIOXAN-2-IL) -ALKYLENE-4-PIPERIDIL-2-IMIDAZOLINONE, 2-HEXAHYDRO-PIRIMIDINONE OR 2-IMINO-IMIDAZOLIDINEInfo
- Publication number
- AR231638A1 AR231638A1 AR282944A AR28294480A AR231638A1 AR 231638 A1 AR231638 A1 AR 231638A1 AR 282944 A AR282944 A AR 282944A AR 28294480 A AR28294480 A AR 28294480A AR 231638 A1 AR231638 A1 AR 231638A1
- Authority
- AR
- Argentina
- Prior art keywords
- pirimidinone
- benzoxatio
- benzoxatian
- piperidil
- benzodioxan
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US88808978A | 1978-03-20 | 1978-03-20 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR231638A1 true AR231638A1 (en) | 1985-01-31 |
Family
ID=25392505
Family Applications (4)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR275879A AR227272A1 (en) | 1978-03-20 | 1979-03-20 | PROCEDURE FOR OBTAINING COMPOUNDS OF N-OXACICLIL-ALQUIL-PIPERIDIL-DIAZA AND ITS SALTS |
AR282945A AR227400A1 (en) | 1978-03-20 | 1980-10-20 | PROCEDURE TO OBTAIN N-OXACICLIL-ALKYL-PIPERIDINES AND THEIR SALTS |
AR282944A AR231638A1 (en) | 1978-03-20 | 1980-10-20 | PROCEDURE FOR OBTAINING COMPOUNDS OF 1-1-2- (1,4-BENZOXATIO OR 1,4-BENZOXATIAN OR 1,4-BENZODIOXAN-2-IL) -ALKYLENE-4-PIPERIDIL-2-IMIDAZOLINONE, 2-HEXAHYDRO-PIRIMIDINONE OR 2-IMINO-IMIDAZOLIDINE |
AR282946A AR227527A1 (en) | 1978-03-20 | 1980-10-20 | PROCEDURE FOR THE ELABORATION OF NEW COMPOUNDS N-OXACICLILALQUIL-PIPERIDIL-DIAZOICOS |
Family Applications Before (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR275879A AR227272A1 (en) | 1978-03-20 | 1979-03-20 | PROCEDURE FOR OBTAINING COMPOUNDS OF N-OXACICLIL-ALQUIL-PIPERIDIL-DIAZA AND ITS SALTS |
AR282945A AR227400A1 (en) | 1978-03-20 | 1980-10-20 | PROCEDURE TO OBTAIN N-OXACICLIL-ALKYL-PIPERIDINES AND THEIR SALTS |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR282946A AR227527A1 (en) | 1978-03-20 | 1980-10-20 | PROCEDURE FOR THE ELABORATION OF NEW COMPOUNDS N-OXACICLILALQUIL-PIPERIDIL-DIAZOICOS |
Country Status (20)
Country | Link |
---|---|
EP (1) | EP0004358B1 (en) |
JP (1) | JPS54157570A (en) |
AR (4) | AR227272A1 (en) |
AT (1) | AT372088B (en) |
AU (1) | AU529838B2 (en) |
DD (1) | DD142341A5 (en) |
DE (1) | DE2961738D1 (en) |
DK (1) | DK113079A (en) |
ES (4) | ES478662A1 (en) |
FI (1) | FI66373C (en) |
GB (1) | GB2019837B (en) |
GR (1) | GR71865B (en) |
HU (1) | HU182941B (en) |
IL (1) | IL56908A (en) |
MY (1) | MY8700122A (en) |
NO (1) | NO150202C (en) |
NZ (1) | NZ189939A (en) |
PL (1) | PL116514B1 (en) |
PT (1) | PT69369A (en) |
ZA (2) | ZA79417B (en) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4329348A (en) * | 1979-02-26 | 1982-05-11 | Ciba-Geigy Corporation | N-Oxacyclic-alkylpiperidines as psychostimulants |
DE3124366A1 (en) * | 1981-06-20 | 1982-12-30 | Hoechst Ag, 6000 Frankfurt | N-OXACYCLYL-ALKYLPIPERIDIN DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, PHARMACEUTICAL PREPARATIONS CONTAINING IT AND THE USE THEREOF |
FR2524887A1 (en) * | 1982-04-08 | 1983-10-14 | Bouchara Emile | NOVEL CYANOGUANIDINES, PROCESS FOR OBTAINING THEM AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME |
FR2525600A1 (en) * | 1982-04-21 | 1983-10-28 | Bouchara Emile | NOVEL CARBOXAMIDOGUANIDINES, PROCESS FOR OBTAINING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
US4556660A (en) * | 1982-07-12 | 1985-12-03 | Janssen Pharmaceutica N.V. | N-(Bicyclic heterocyclyl)-4-piperidinamines |
JP2807577B2 (en) * | 1990-06-15 | 1998-10-08 | エーザイ株式会社 | Cyclic amide derivative |
SI9300097B (en) * | 1992-02-27 | 2001-12-31 | Janssen Pharmaceutica Nv | (benzodioxan, benzofuran or benzopyran) alkylamino) alkyl substituted guanidines |
US5703115A (en) * | 1993-02-19 | 1997-12-30 | Janssen Pharmaceutica, N.V. | (benzodioxan, benzofuran or benzopyran) alkylamino! alkyl substituted guanidines |
US6133277A (en) * | 1997-12-05 | 2000-10-17 | Janssen Pharmaceutica N.V. | (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties |
PT1187829E (en) | 1999-06-02 | 2004-04-30 | Janssen Pharmaceutica Nv | (BENZODIOXAN, BENZOFURAN OR BENZOPYRANE) DERIVATIVES SUBSTITUTED WITH AMINOALKYL |
US6900222B1 (en) * | 1999-06-02 | 2005-05-31 | Janssen Pharmaceutica N.V. | Pyrrolidinyl, piperdinyl or homopiperidinyl substituted (benzodioxan, benzofuran or benzopyran) derivatives |
JO2352B1 (en) | 2000-06-22 | 2006-12-12 | جانسين فارماسيوتيكا ان. في | Compounds for treating fundic disaccomodation |
JP2008530229A (en) | 2005-02-17 | 2008-08-07 | ワイス | Cycloalkyl fused indole, benzothiophene, benzofuran and indene derivatives |
CN114920686B (en) * | 2022-05-20 | 2023-11-24 | 山东农业大学 | Synthesis method of 5- (benzenesulfonyl) -N-piperidin-4-yl-2- (trifluoromethyl) benzenesulfonamide hydrochloride |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3910930A (en) * | 1973-01-04 | 1975-10-07 | Janssen Pharmaceutica Nv | 1-{55 1-{8 2-(1,4-Benzodioxan-2-yl)-2-hydroxyethyl{9 -4-piperidyl{56 -2-benzimidazolinones |
-
1977
- 1977-08-17 GR GR58624A patent/GR71865B/el unknown
-
1979
- 1979-01-31 ZA ZA79417A patent/ZA79417B/en unknown
- 1979-03-15 ES ES478662A patent/ES478662A1/en not_active Expired
- 1979-03-15 GB GB7909231A patent/GB2019837B/en not_active Expired
- 1979-03-16 DE DE7979100815T patent/DE2961738D1/en not_active Expired
- 1979-03-16 FI FI790894A patent/FI66373C/en not_active IP Right Cessation
- 1979-03-16 EP EP79100815A patent/EP0004358B1/en not_active Expired
- 1979-03-17 PL PL1979214206A patent/PL116514B1/en unknown
- 1979-03-19 DK DK113079A patent/DK113079A/en not_active Application Discontinuation
- 1979-03-19 ZA ZA791276A patent/ZA791276B/en unknown
- 1979-03-19 NZ NZ189939A patent/NZ189939A/en unknown
- 1979-03-19 IL IL56908A patent/IL56908A/en unknown
- 1979-03-19 DD DD79211661A patent/DD142341A5/en unknown
- 1979-03-19 PT PT69369A patent/PT69369A/en unknown
- 1979-03-19 AT AT0204479A patent/AT372088B/en not_active IP Right Cessation
- 1979-03-19 NO NO790917A patent/NO150202C/en unknown
- 1979-03-19 HU HU79CI1923A patent/HU182941B/en unknown
- 1979-03-19 AU AU45243/79A patent/AU529838B2/en not_active Ceased
- 1979-03-20 JP JP3184279A patent/JPS54157570A/en active Pending
- 1979-03-20 AR AR275879A patent/AR227272A1/en active
- 1979-09-28 ES ES484570A patent/ES484570A1/en not_active Expired
- 1979-09-28 ES ES484571A patent/ES484571A1/en not_active Expired
- 1979-09-28 ES ES484572A patent/ES484572A1/en not_active Expired
-
1980
- 1980-10-20 AR AR282945A patent/AR227400A1/en active
- 1980-10-20 AR AR282944A patent/AR231638A1/en active
- 1980-10-20 AR AR282946A patent/AR227527A1/en active
-
1987
- 1987-12-30 MY MY122/87A patent/MY8700122A/en unknown
Also Published As
Publication number | Publication date |
---|---|
IL56908A0 (en) | 1979-05-31 |
NO790917L (en) | 1979-09-21 |
FI66373B (en) | 1984-06-29 |
ES484570A1 (en) | 1980-05-16 |
DD142341A5 (en) | 1980-06-18 |
DK113079A (en) | 1979-09-21 |
PL116514B1 (en) | 1981-06-30 |
EP0004358B1 (en) | 1982-01-06 |
ZA791276B (en) | 1980-03-26 |
GB2019837B (en) | 1982-08-25 |
AR227400A1 (en) | 1982-10-29 |
MY8700122A (en) | 1987-12-31 |
ES484572A1 (en) | 1980-05-16 |
NZ189939A (en) | 1981-12-15 |
NO150202C (en) | 1984-09-05 |
ES478662A1 (en) | 1980-01-16 |
AT372088B (en) | 1983-08-25 |
EP0004358A1 (en) | 1979-10-03 |
ES484571A1 (en) | 1980-05-16 |
AR227527A1 (en) | 1982-11-15 |
DE2961738D1 (en) | 1982-02-25 |
FI66373C (en) | 1984-10-10 |
IL56908A (en) | 1983-09-30 |
NO150202B (en) | 1984-05-28 |
GB2019837A (en) | 1979-11-07 |
AR227272A1 (en) | 1982-10-15 |
PT69369A (en) | 1979-04-01 |
JPS54157570A (en) | 1979-12-12 |
PL214206A1 (en) | 1980-02-25 |
HU182941B (en) | 1984-03-28 |
FI790894A (en) | 1979-09-21 |
AU529838B2 (en) | 1983-06-23 |
AU4524379A (en) | 1979-09-27 |
GR71865B (en) | 1983-07-07 |
ATA204479A (en) | 1983-01-15 |
ZA79417B (en) | 1980-01-30 |
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