AR108864A1 - Agentes antibacterianos - Google Patents

Agentes antibacterianos

Info

Publication number
AR108864A1
AR108864A1 ARP170101736A ARP170101736A AR108864A1 AR 108864 A1 AR108864 A1 AR 108864A1 AR P170101736 A ARP170101736 A AR P170101736A AR P170101736 A ARP170101736 A AR P170101736A AR 108864 A1 AR108864 A1 AR 108864A1
Authority
AR
Argentina
Prior art keywords
alkyl
cycloalkyl
optionally substituted
heterocycloalkyl
haloalkyl
Prior art date
Application number
ARP170101736A
Other languages
English (en)
Spanish (es)
Inventor
Darin James Hildebrandt
Timothy Robert Kane
Timothy D Machajewski
Taylor Ann Joo Choi
Andrei W Konradi
Frederick Cohen
Original Assignee
Achaogen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Achaogen Inc filed Critical Achaogen Inc
Publication of AR108864A1 publication Critical patent/AR108864A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D331/00Heterocyclic compounds containing rings of less than five members, having one sulfur atom as the only ring hetero atom
    • C07D331/04Four-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ARP170101736A 2016-06-23 2017-06-22 Agentes antibacterianos AR108864A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201662353910P 2016-06-23 2016-06-23

Publications (1)

Publication Number Publication Date
AR108864A1 true AR108864A1 (es) 2018-10-03

Family

ID=59276882

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP170101736A AR108864A1 (es) 2016-06-23 2017-06-22 Agentes antibacterianos

Country Status (3)

Country Link
AR (1) AR108864A1 (zh)
TW (1) TW201803847A (zh)
WO (1) WO2017223349A1 (zh)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10829440B2 (en) 2015-06-12 2020-11-10 Brown University Antibacterial compounds and methods of making and using same
CN108358887B (zh) * 2018-03-20 2020-12-22 富乐马鸿凯(大连)医药有限公司 一种光学纯的含硫四元杂环药物中间体的合成
CN110283745B (zh) * 2019-06-27 2021-05-11 浙江工业大学 医院不动杆菌fk2及其在降解有机污染物中的应用
US11555010B2 (en) 2019-07-25 2023-01-17 Brown University Diamide antimicrobial agents
CN110563611B (zh) * 2019-09-19 2021-02-02 中国医学科学院医药生物技术研究所 一种异羟肟酸类衍生物及其制备方法和应用
CN113604408B (zh) * 2021-09-06 2023-08-22 浙江树人学院(浙江树人大学) 莫德斯托斯不动杆菌hyy-1及其在降解有机污染物中的应用
CN116730870B (zh) * 2023-08-08 2023-10-13 中国医学科学院医药生物技术研究所 异羟肟酸类化合物或其可药用盐、及其用途和制备方法

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1998018754A1 (en) 1996-10-28 1998-05-07 Versicor, Inc. Methods for solid-phase synthesis of hydroxylamine compounds and derivatives, and combinatorial libraries thereof
EP1169031A1 (en) 1999-04-09 2002-01-09 British Biotech Pharmaceuticals Limited Antimicrobial agents
KR101076018B1 (ko) 2003-01-08 2011-10-21 유니버시티 오브 워싱톤 항균제
JP2010502617A (ja) 2006-08-31 2010-01-28 シェーリング コーポレイション 抗菌物質として有用なヒダントイン誘導体
JP5227304B2 (ja) 2007-02-28 2013-07-03 大正製薬株式会社 新規なヒドロキサム酸誘導体
TWI519508B (zh) 2007-06-12 2016-02-01 Achaogen Inc 抗菌劑
WO2009158369A1 (en) 2008-06-25 2009-12-30 Schering Corporation Synthesis and use of heterocyclic antibacterial agents
JP2011529964A (ja) 2008-08-04 2011-12-15 シェーリング コーポレイション 抗菌剤としての尿素誘導体
WO2010024356A1 (ja) 2008-08-27 2010-03-04 大正製薬株式会社 ナフチリジン-n-オキシドを有する新規ヒドロキサム酸誘導体
US8372885B2 (en) 2008-09-17 2013-02-12 Novartis Ag Organic compounds and their uses
US8722686B2 (en) 2008-09-19 2014-05-13 Pfizer Inc. Hydroxamic acid derivatives useful as antibacterial agents
WO2010100475A1 (en) 2009-03-02 2010-09-10 Astrazeneca Ab Hydroxamic acid derivatives as gram-negative antibacterial agents
WO2011005355A1 (en) 2009-05-07 2011-01-13 Achaogen, Inc. Combinations comprising a lpxc inhibitor and an antibiotic for use in the treatment of infections caused by gram-negative bacteria
CA2774250C (en) 2009-10-13 2013-12-17 Pfizer Inc. C-linked hydroxamic acid derivatives useful as antibacterial agents
US8664401B2 (en) 2009-12-16 2014-03-04 Pfizer Inc. N-linked hydroxamic acid derivatives useful as antibacterial agents
SI2562155T1 (sl) 2010-04-20 2019-08-30 Fujifilm Toyama Chemical Co., Ltd. Derivat hidroksamske kisline
KR20140023869A (ko) 2010-11-10 2014-02-27 아카오젠, 인코포레이티드 하이드록삼산 유도체 및 세균 감염 치료에서의 이들의 사용
AR087843A1 (es) 2011-09-12 2014-04-23 Achaogen Inc Formas polimorficas de n-((s)-3-amino-1-(hidroxiamino)-3-metil-1-oxobutan-2-il)-4-(((1r,2r)-2-(hidroximetil)ciclopropil)buta-1,3-dinil)benzamida
WO2013170030A1 (en) 2012-05-09 2013-11-14 Achaogen, Inc. Antibacterial agents
WO2013170165A1 (en) 2012-05-10 2013-11-14 Achaogen, Inc. Antibacterial agents
WO2014165075A1 (en) 2013-03-12 2014-10-09 Achaogen, Inc. Antibacterial agents

Also Published As

Publication number Publication date
WO2017223349A1 (en) 2017-12-28
TW201803847A (zh) 2018-02-01

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