|
US2466420A
(en)
|
1947-11-26 |
1949-04-05 |
Eastman Kodak Co |
Ketene condensation products with aldehydes
|
|
US3226394A
(en)
|
1964-06-16 |
1965-12-28 |
Shulton Inc |
Pyridylethylated anthranilamides and derivatives thereof
|
|
CH504416A
(de)
|
1966-12-05 |
1971-03-15 |
Ciba Geigy Ag |
Verfahren zur Herstellung von aromatischen Sulfamoylverbindungen
|
|
US4551540A
(en)
|
1983-01-17 |
1985-11-05 |
Borg-Warner Chemicals, Inc. |
Substituted 2,5-dimethylpyrroles
|
|
US5190541A
(en)
|
1990-10-17 |
1993-03-02 |
Boston Scientific Corporation |
Surgical instrument and method
|
|
CA2452130A1
(en)
|
1992-03-05 |
1993-09-16 |
Francis J. Burrows |
Methods and compositions for targeting the vasculature of solid tumors
|
|
US5474765A
(en)
|
1992-03-23 |
1995-12-12 |
Ut Sw Medical Ctr At Dallas |
Preparation and use of steroid-polyanionic polymer-based conjugates targeted to vascular endothelial cells
|
|
US5686472A
(en)
|
1992-10-29 |
1997-11-11 |
Merck & Co., Inc. |
Inhibitors of farnesyl-protein transferase
|
|
US5593992A
(en)
|
1993-07-16 |
1997-01-14 |
Smithkline Beecham Corporation |
Compounds
|
|
EP0785937A1
(en)
|
1994-10-14 |
1997-07-30 |
Smithkline Beecham Plc |
2-(imidazol-4-yl)carbapeneme derivatives, intermediates thereof and use as antibacterials
|
|
KR19990007865A
(ko)
|
1995-04-19 |
1999-01-25 |
스피겔알렌제이 |
약물 방출용 피복 스텐트
|
|
US6117432A
(en)
|
1995-04-20 |
2000-09-12 |
Societe D'exploitation De Produits Pour Les Industries Chimiques (S.E.P.P.I.C.) |
Therapeutic composition comprising an antigen or an in vivo generator of a compound comprising an amino acid sequence
|
|
TW349948B
(en)
|
1995-10-31 |
1999-01-11 |
Janssen Pharmaceutica Nv |
Farnesyl transferase inhibiting 2-quinolone derivatives
|
|
GB9523675D0
(en)
|
1995-11-20 |
1996-01-24 |
Celltech Therapeutics Ltd |
Chemical compounds
|
|
WO1997021701A1
(en)
|
1995-12-08 |
1997-06-19 |
Janssen Pharmaceutica N.V. |
Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives
|
|
US5874442A
(en)
|
1995-12-22 |
1999-02-23 |
Schering-Plough Corporation |
Tricyclic amides useful for inhibition of G-protein function and for treatment of proliferative disease
|
|
US6011029A
(en)
|
1996-02-26 |
2000-01-04 |
Bristol-Myers Squibb Company |
Inhibitors of farnesyl protein transferase
|
|
US5702390A
(en)
|
1996-03-12 |
1997-12-30 |
Ethicon Endo-Surgery, Inc. |
Bioplar cutting and coagulation instrument
|
|
AU711936B2
(en)
|
1996-08-09 |
1999-10-28 |
Banyu Pharmaceutical Co., Ltd. |
Stereoselective deoxygenation reaction
|
|
EP0946565B1
(en)
|
1996-12-20 |
2003-10-15 |
Tovarischestvo S Ogranichennoi Otvetstvennostju "Tabifarm" |
Method and device for production of lyophilized hydrochloride-1ss, 10ss-epoxy-13-dimethylamino-guaia-3(4)-en-6,12-olide
|
|
UA59384C2
(uk)
|
1996-12-20 |
2003-09-15 |
Пфайзер, Інк. |
Похідні сульфонамідів та амідів як агоністи простагландину, фармацевтична композиція та способи лікування на їх основі
|
|
TW591030B
(en)
|
1997-03-10 |
2004-06-11 |
Janssen Pharmaceutica Nv |
Farnesyl transferase inhibiting 1,8-annelated quinolinone derivatives substituted with N- or C-linked imidazoles
|
|
HUP0001122A3
(en)
|
1997-04-25 |
2002-03-28 |
Janssen Pharmaceutica Nv |
Farnesyltransferase inhibiting quinazolinones
|
|
TW491872B
(en)
|
1997-05-27 |
2002-06-21 |
Ciba Sc Holding Ag |
Block oligomers containing l-hydrocarbyloxy-2,2,6,6-tetramethyl-4- piperidyl groups as stabilizers for lower polyolefin
|
|
US6100254A
(en)
|
1997-10-10 |
2000-08-08 |
Board Of Regents, The University Of Texas System |
Inhibitors of protein tyrosine kinases
|
|
ES2176012T3
(es)
|
1998-03-05 |
2002-11-16 |
Formula One Administration Ltd |
Sistema de comunicacion de datos.
|
|
US6303654B1
(en)
|
1998-03-12 |
2001-10-16 |
Wisconsin Alumni Research Foundation |
Acyclic monoterpenoid derivatives
|
|
WO2000001691A1
(en)
|
1998-07-01 |
2000-01-13 |
Merck & Co., Inc. |
Process for making farnesyl-protein transferase inhibitors
|
|
CA2336848A1
(en)
|
1998-07-10 |
2000-01-20 |
Merck & Co., Inc. |
Novel angiogenesis inhibitors
|
|
ES2237125T3
(es)
|
1998-08-27 |
2005-07-16 |
Pfizer Products Inc. |
Derivados de quinolin-2-ona utiles como agentes anticancerigenos.
|
|
ATE321037T1
(de)
|
1998-08-27 |
2006-04-15 |
Pfizer Prod Inc |
Als antikrebsmittel verwendbare alkinyl- substituierte chinolin-2-on-derivate
|
|
GB9824579D0
(en)
|
1998-11-10 |
1999-01-06 |
Novartis Ag |
Organic compounds
|
|
TW531533B
(en)
|
1998-12-23 |
2003-05-11 |
Janssen Pharmaceutica Nv |
1,2-annelated quinoline derivatives having farnesyl transferase and geranylgeranyl transferase inhibiting activity
|
|
EP1140938B1
(en)
|
1999-01-11 |
2003-08-27 |
Princeton University |
High affinity inhibitors for target validation and uses thereof
|
|
US7125875B2
(en)
|
1999-04-15 |
2006-10-24 |
Bristol-Myers Squibb Company |
Cyclic protein tyrosine kinase inhibitors
|
|
HUP0202708A3
(en)
|
1999-04-15 |
2004-12-28 |
Bristol Myers Squibb Co |
Cyclic protein tyrosine kinase inhibitors, pharmaceutical compositions containing them and their use
|
|
ATE269357T1
(de)
|
1999-04-28 |
2004-07-15 |
Univ Texas |
Zusammensetzungen und verfahren zur krebsbehandlung durch die selektive hemmung von vegf
|
|
US6346625B1
(en)
|
1999-06-23 |
2002-02-12 |
Astrazeneca Ab |
Protein kinase inhibitors
|
|
DE19962924A1
(de)
|
1999-12-24 |
2001-07-05 |
Bayer Ag |
Substituierte Oxazolidinone und ihre Verwendung
|
|
WO2001047897A1
(en)
|
1999-12-28 |
2001-07-05 |
Pharmacopeia, Inc. |
Cytokine, especially tnf-alpha, inhibitors
|
|
FR2803592A1
(fr)
|
2000-01-06 |
2001-07-13 |
Aventis Cropscience Sa |
Nouveaux derives de l'acide 3-hydroxypicolinique, leur procede de preparation et compositions fongicides les contenant.
|
|
US6558385B1
(en)
|
2000-09-22 |
2003-05-06 |
Tissuelink Medical, Inc. |
Fluid-assisted medical device
|
|
US6692491B1
(en)
|
2000-03-24 |
2004-02-17 |
Scimed Life Systems, Inc. |
Surgical methods and apparatus for positioning a diagnostic or therapeutic element around one or more pulmonary veins or other body structures
|
|
US6776796B2
(en)
|
2000-05-12 |
2004-08-17 |
Cordis Corportation |
Antiinflammatory drug and delivery device
|
|
US6960590B2
(en)
|
2000-10-17 |
2005-11-01 |
Merck & Co. Inc. |
Orally active salts with tyrosine kinase activity
|
|
US6958243B2
(en)
*
|
2000-12-14 |
2005-10-25 |
Biotage Ab |
Organic reactions with CO generating materials
|
|
US7105682B2
(en)
|
2001-01-12 |
2006-09-12 |
Amgen Inc. |
Substituted amine derivatives and methods of use
|
|
AR035885A1
(es)
|
2001-05-14 |
2004-07-21 |
Novartis Ag |
Derivados de 4-amino-5-fenil-7-ciclobutilpirrolo (2,3-d)pirimidina, un proceso para su preparacion, una composicion farmaceutica y el uso de dichos derivados para la preparacion de una composicion farmaceutica
|
|
WO2003024969A1
(en)
|
2001-09-14 |
2003-03-27 |
Merck & Co., Inc. |
Tyrosine kinase inhibitors
|
|
WO2003024931A1
(en)
|
2001-09-14 |
2003-03-27 |
Merck & Co., Inc. |
Tyrosine kinase inhibitors
|
|
TWI259081B
(en)
|
2001-10-26 |
2006-08-01 |
Sugen Inc |
Treatment of acute myeloid leukemia with indolinone compounds
|
|
TWI302836B
(en)
|
2001-10-30 |
2008-11-11 |
Novartis Ag |
Staurosporine derivatives as inhibitors of flt3 receptor tyrosine kinase activity
|
|
MXPA04006271A
(es)
|
2001-12-27 |
2004-10-04 |
Theravance Inc |
Derivados de indolinona utiles como inhibidores de la proteina cinasa.
|
|
EP1513821B1
(en)
|
2002-05-23 |
2007-10-31 |
Cytopia PTY Ltd |
Protein kinase inhibitors
|
|
PE20040522A1
(es)
|
2002-05-29 |
2004-09-28 |
Novartis Ag |
Derivados de diarilurea dependientes de la cinasa de proteina
|
|
MY141867A
(en)
|
2002-06-20 |
2010-07-16 |
Vertex Pharma |
Substituted pyrimidines useful as protein kinase inhibitors
|
|
GB0215676D0
(en)
|
2002-07-05 |
2002-08-14 |
Novartis Ag |
Organic compounds
|
|
EP1546117A2
(en)
|
2002-08-14 |
2005-06-29 |
Vertex Pharmaceuticals Incorporated |
Protein kinase inhibitors and uses thereof
|
|
BR0313743A
(pt)
|
2002-08-23 |
2005-07-05 |
Chiron Corp |
Benzimidazol quinolinonas e usos destas
|
|
AU2003258491A1
(en)
|
2002-09-05 |
2004-03-29 |
Neurosearch A/S |
Amide derivatives and their use as chloride channel blockers
|
|
CA2500727A1
(en)
|
2002-10-03 |
2004-04-15 |
Targegen, Inc. |
Vasculostatic agents and methods of use thereof
|
|
US20080207617A1
(en)
|
2002-10-29 |
2008-08-28 |
Kirin Beer Kabushiki Kaisha |
Quinoline Derivatives and Quinazoline Derivatives Inhibiting Autophosphrylation of Flt3 and Medicinal Compositions Containing the Same
|
|
BR0316229A
(pt)
|
2002-11-13 |
2005-10-04 |
Chiron Corp |
Métodos de tratamento de câncer e métodos relacionados
|
|
AR042052A1
(es)
|
2002-11-15 |
2005-06-08 |
Vertex Pharma |
Diaminotriazoles utiles como inhibidores de proteinquinasas
|
|
EP1581526B1
(en)
|
2002-12-18 |
2009-03-11 |
Vertex Pharmaceuticals Incorporated |
Benzisoxazole derivatives useful as inhibitors of protein kinases
|
|
MXPA05010945A
(es)
|
2003-04-09 |
2005-11-25 |
Japan Tobacco Inc |
Compuesto pentaciclico heteroaromatico y uso medicinal del mismo.
|
|
US7790724B2
(en)
|
2003-04-25 |
2010-09-07 |
Janssen Pharmaceutica N.V. |
c-fms kinase inhibitors
|
|
MXPA05011503A
(es)
|
2003-04-25 |
2006-05-31 |
Johnson & Johnson |
Inhibidores de la c-fms cinasa.
|
|
US20050113566A1
(en)
|
2003-04-25 |
2005-05-26 |
Player Mark R. |
Inhibitors of C-FMS kinase
|
|
US7427683B2
(en)
*
|
2003-04-25 |
2008-09-23 |
Ortho-Mcneil Pharmaceutical, Inc. |
c-fms kinase inhibitors
|
|
JP5013593B2
(ja)
|
2003-07-28 |
2012-08-29 |
スミスクライン ビーチャム コーポレーション |
化合物
|
|
BRPI0415467A
(pt)
|
2003-10-23 |
2006-12-19 |
Ab Science |
compostos de 2-aminoariloxazol para o tratamento de doenças
|
|
GB0326601D0
(en)
|
2003-11-14 |
2003-12-17 |
Novartis Ag |
Organic compounds
|
|
KR20060129413A
(ko)
|
2004-01-30 |
2006-12-15 |
에이비 사이언스 |
티로신 키나제 억제제로서의2-(3-치환된-아릴)아미노-4-아릴-티아졸
|
|
US7645755B2
(en)
|
2004-10-22 |
2010-01-12 |
Janssen Pharmaceutical N.V. |
Inhibitors of c-fms kinase
|
|
JP5046950B2
(ja)
|
2004-10-22 |
2012-10-10 |
ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ |
C−fmsキナーゼのインヒビター
|
|
WO2006047504A1
(en)
|
2004-10-22 |
2006-05-04 |
Janssen Pharmaceutica, N.V. |
Aromatic amides as inhibitors of c-fms kinase
|
|
NZ555289A
(en)
|
2004-10-22 |
2010-10-29 |
Janssen Pharmaceutica Nv |
Inhibitors of c-fms kinase
|
|
US20060281769A1
(en)
|
2005-06-10 |
2006-12-14 |
Baumann Christian A |
Synergistic modulation of flt3 kinase using thienopyrimidine and thienopyridine kinase modulators
|
|
US20060281700A1
(en)
|
2005-06-10 |
2006-12-14 |
Baumann Christian A |
Synergistic modulation of flt3 kinase using aminopyrimidines kinase modulators
|
|
US20060281755A1
(en)
|
2005-06-10 |
2006-12-14 |
Baumann Christian A |
Synergistic modulation of flt3 kinase using aminopyrimidines kinase modulators
|
|
US20060281788A1
(en)
|
2005-06-10 |
2006-12-14 |
Baumann Christian A |
Synergistic modulation of flt3 kinase using a flt3 inhibitor and a farnesyl transferase inhibitor
|
|
US20060281771A1
(en)
|
2005-06-10 |
2006-12-14 |
Baumann Christian A |
Synergistic modulation of flt3 kinase using aminoquinoline and aminoquinazoline kinase modulators
|
|
JP2009511628A
(ja)
|
2005-10-18 |
2009-03-19 |
ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ |
Flt3キナーゼの阻害方法
|
|
US8697716B2
(en)
|
2006-04-20 |
2014-04-15 |
Janssen Pharmaceutica Nv |
Method of inhibiting C-KIT kinase
|
|
ES2565238T3
(es)
|
2006-04-20 |
2016-04-01 |
Janssen Pharmaceutica N.V. |
Inhibidores de la c-fms quinasa
|
|
EP2021335B1
(en)
|
2006-04-20 |
2011-05-25 |
Janssen Pharmaceutica N.V. |
Heterocyclic compounds as inhibitors of c-fms kinase
|
|
JP5480619B2
(ja)
|
2006-04-20 |
2014-04-23 |
ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ |
c−fmsキナーゼの阻害剤
|
|
CA2672960A1
(en)
*
|
2006-12-20 |
2008-07-10 |
Schering Corporation |
Novel jnk inhibitors
|
|
WO2008138184A1
(fr)
*
|
2007-05-14 |
2008-11-20 |
Shanghai Hengrui Pharmaceutical Co.Ltd. |
Dérivés de pyrrolo-azacycles, leur procédé de fabrication et leur utilisation en tant qu'inhibiteurs de protéine kinases
|
|
JO3240B1
(ar)
|
2007-10-17 |
2018-03-08 |
Janssen Pharmaceutica Nv |
c-fms مثبطات كيناز
|
|
CA2704231A1
(en)
|
2007-10-31 |
2009-05-07 |
Janssen Pharmaceutica N.V. |
Biomarker for assessing response to fms treatment
|
|
WO2010078408A1
(en)
*
|
2008-12-30 |
2010-07-08 |
Biogen Idec Ma Inc. |
Heteroaryl compounds useful as raf kinase inhibitors
|
|
JP2011026305A
(ja)
*
|
2009-06-24 |
2011-02-10 |
Daiichi Sankyo Co Ltd |
イミダゾールカルボニル化合物を含有する医薬組成物
|
|
AR078187A1
(es)
*
|
2009-09-28 |
2011-10-19 |
Hoffmann La Roche |
Derivados heterociclicos de benzoxazepina, composiciones farmaceuticas que los contienen y uso de los mismos en el tratamiento del cancer.
|
|
WO2011090935A1
(en)
*
|
2010-01-19 |
2011-07-28 |
Merck Sharp & Dohme Corp. |
PYRAZOLO[1,5-a]PYRIMIDINE COMPOUNDS AS mTOR INHIBITORS
|
|
US9303046B2
(en)
*
|
2012-08-07 |
2016-04-05 |
Janssen Pharmaceutica Nv |
Process for the preparation of heterocyclic ester derivatives
|