AR004368A1 - Compuestos de piperidina -1,-4 sustituida, procedimientos para prepararlos y un procedimiento para preparar 1-bencil-4-((5,6-dimetoxi-1-indanon)-2-il)metilpiperidina mediante dichos compuestos. - Google Patents
Compuestos de piperidina -1,-4 sustituida, procedimientos para prepararlos y un procedimiento para preparar 1-bencil-4-((5,6-dimetoxi-1-indanon)-2-il)metilpiperidina mediante dichos compuestos.Info
- Publication number
- AR004368A1 AR004368A1 ARP960105577A ARP960105577A AR004368A1 AR 004368 A1 AR004368 A1 AR 004368A1 AR P960105577 A ARP960105577 A AR P960105577A AR P960105577 A ARP960105577 A AR P960105577A AR 004368 A1 AR004368 A1 AR 004368A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparing
- compounds
- indanon
- methylpiperidine
- dimetoxi
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/30—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
- C07D211/32—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US875395P | 1995-12-15 | 1995-12-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR004368A1 true AR004368A1 (es) | 1998-11-04 |
Family
ID=21733469
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP960105577A AR004368A1 (es) | 1995-12-15 | 1996-12-10 | Compuestos de piperidina -1,-4 sustituida, procedimientos para prepararlos y un procedimiento para preparar 1-bencil-4-((5,6-dimetoxi-1-indanon)-2-il)metilpiperidina mediante dichos compuestos. |
Country Status (33)
| Country | Link |
|---|---|
| EP (1) | EP0883607A1 (pl) |
| JP (1) | JP3066083B2 (pl) |
| KR (1) | KR20000064387A (pl) |
| AP (1) | AP708A (pl) |
| AR (1) | AR004368A1 (pl) |
| AU (1) | AU716462B2 (pl) |
| BG (1) | BG102525A (pl) |
| BR (1) | BR9612018A (pl) |
| CA (1) | CA2237647A1 (pl) |
| CO (1) | CO4750831A1 (pl) |
| CZ (1) | CZ180898A3 (pl) |
| DZ (1) | DZ2141A1 (pl) |
| GT (1) | GT199600092A (pl) |
| HN (1) | HN1996000065A (pl) |
| HR (1) | HRP960592A2 (pl) |
| HU (1) | HUP9904275A3 (pl) |
| IL (3) | IL136420A0 (pl) |
| IS (1) | IS4752A (pl) |
| MA (1) | MA24032A1 (pl) |
| NO (1) | NO982712L (pl) |
| NZ (1) | NZ318843A (pl) |
| OA (1) | OA10694A (pl) |
| PE (1) | PE25698A1 (pl) |
| PL (1) | PL197306B1 (pl) |
| RO (1) | RO121382B1 (pl) |
| RU (1) | RU2160731C2 (pl) |
| SK (1) | SK75498A3 (pl) |
| TN (1) | TNSN96153A1 (pl) |
| TW (1) | TW414787B (pl) |
| UY (1) | UY24401A1 (pl) |
| WO (1) | WO1997022584A1 (pl) |
| YU (1) | YU49486B (pl) |
| ZA (1) | ZA9610533B (pl) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6252081B1 (en) | 1998-01-16 | 2001-06-26 | Eisai Co., Ltd. | Process for production of donepezil derivative |
| IL125809A (en) * | 1998-08-17 | 2005-08-31 | Finetech Lab Ltd | Process and intermediates for production of donepezil and related compounds |
| US7148354B2 (en) * | 2002-07-24 | 2006-12-12 | Dr. Reddy's Laboratories Limited | Process for preparation of donepezil |
| IL150982A (en) | 2002-07-30 | 2007-02-11 | Ori Lerman | Process for making Donafzil |
| IL151253A0 (en) * | 2002-08-14 | 2003-04-10 | Finetech Lab Ltd | Process for production of highly pure donepezil hydrochloride |
| US6649765B1 (en) | 2003-02-12 | 2003-11-18 | Usv Limited, Bsd Marg. | Process for the preparation of 1-benzyl-4(5,6-dimethoxy-1-indanon)-2-yl) methyl piperidine hydrochloride (Donepezil HCL) |
| US6953856B2 (en) | 2003-02-12 | 2005-10-11 | Usv, Limited | Process for the preparation of 1-benzyl-4-(5,6-dimethoxy-1-indanon)-2-yl) methyl piperidine hydrochloride (Donepezil HCI) |
| US20070129549A1 (en) * | 2003-03-21 | 2007-06-07 | Yatendra Kumar | Stable lamotrigine pharmaceutical compositions and processes for their preparation |
| WO2004099142A1 (en) * | 2003-05-05 | 2004-11-18 | Ranbaxy Laboratories Limited | Hydrobromide salt of benzyl-piperidylmethyl-indanone and its polymorphs |
| WO2005003092A1 (en) | 2003-07-01 | 2005-01-13 | Hetero Drugs Limited | Preparation of intermediates for acetyl cholinesterase inhibitors |
| CN1280273C (zh) * | 2003-11-05 | 2006-10-18 | 天津和美生物技术有限公司 | 合成多奈哌齐及其衍生物的方法 |
| KR20070083679A (ko) | 2004-09-29 | 2007-08-24 | 케마지스 리미티드 | 약학적으로 순수한 비정질 도네페닐 염산염의 제조를 위한정제된 도네페질 말레산염의 용도 |
| CN100436416C (zh) * | 2005-07-29 | 2008-11-26 | 西南合成制药股份有限公司 | 盐酸多奈哌齐合成工艺 |
| GB0515803D0 (en) * | 2005-07-30 | 2005-09-07 | Pliva Hrvatska D O O | Intermediate compounds |
| AR057910A1 (es) | 2005-11-18 | 2007-12-26 | Synthon Bv | Proceso para preparar donepezilo |
| KR20080085195A (ko) * | 2006-01-04 | 2008-09-23 | 씨아이피엘에이 엘티디. | 도네페질의 제조방법 및 중간체 |
| US8247563B2 (en) | 2006-12-11 | 2012-08-21 | Reviva Pharmaceuticals, Inc. | Compositions, synthesis, and methods of using indanone based cholinesterase inhibitors |
| WO2013078608A1 (en) | 2011-11-29 | 2013-06-06 | Ziqiang Gu | Donepezil pamoate and methods of making and using the same |
| ES2888074T3 (es) | 2013-08-16 | 2021-12-30 | Univ Maastricht | Tratamiento del deterioro cognitivo con inhibidor de PDE4 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI95572C (fi) * | 1987-06-22 | 1996-02-26 | Eisai Co Ltd | Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi |
| FR2642069B1 (fr) * | 1989-01-20 | 1991-04-12 | Rhone Poulenc Sante | Nouveaux derives du benzopyranne, leur preparation et les compositions pharmaceutiques qui les contiennent |
| DE4439822A1 (de) * | 1994-11-08 | 1996-08-29 | Bayer Ag | Verfahren zur Herstellung von Benzyl-piperidylmethyl-indanonen |
-
1996
- 1996-10-11 SK SK754-98A patent/SK75498A3/sk unknown
- 1996-10-11 WO PCT/IB1996/001076 patent/WO1997022584A1/en not_active Application Discontinuation
- 1996-10-11 IL IL13642096A patent/IL136420A0/xx unknown
- 1996-10-11 CA CA002237647A patent/CA2237647A1/en not_active Abandoned
- 1996-10-11 PL PL327512A patent/PL197306B1/pl not_active IP Right Cessation
- 1996-10-11 HU HU9904275A patent/HUP9904275A3/hu unknown
- 1996-10-11 IL IL13642196A patent/IL136421A0/xx unknown
- 1996-10-11 NZ NZ318843A patent/NZ318843A/xx unknown
- 1996-10-11 KR KR1019980704423A patent/KR20000064387A/ko not_active Application Discontinuation
- 1996-10-11 JP JP9522607A patent/JP3066083B2/ja not_active Expired - Lifetime
- 1996-10-11 BR BR9612018A patent/BR9612018A/pt not_active Application Discontinuation
- 1996-10-11 RO RO98-01070A patent/RO121382B1/ro unknown
- 1996-10-11 CZ CZ981808A patent/CZ180898A3/cs unknown
- 1996-10-11 AU AU70925/96A patent/AU716462B2/en not_active Ceased
- 1996-10-11 IL IL12445296A patent/IL124452A0/xx unknown
- 1996-10-11 EP EP96931937A patent/EP0883607A1/en not_active Withdrawn
- 1996-10-11 RU RU98111204/04A patent/RU2160731C2/ru not_active IP Right Cessation
- 1996-10-14 TW TW085112515A patent/TW414787B/zh not_active IP Right Cessation
- 1996-10-15 HN HN1996000065A patent/HN1996000065A/es unknown
- 1996-11-18 GT GT199600092A patent/GT199600092A/es unknown
- 1996-12-09 PE PE1996000883A patent/PE25698A1/es not_active Application Discontinuation
- 1996-12-10 AR ARP960105577A patent/AR004368A1/es unknown
- 1996-12-11 TN TNTNSN96153A patent/TNSN96153A1/fr unknown
- 1996-12-11 DZ DZ960186A patent/DZ2141A1/fr active
- 1996-12-11 YU YU66096A patent/YU49486B/sh unknown
- 1996-12-11 MA MA24424A patent/MA24032A1/fr unknown
- 1996-12-12 AP APAP/P/1996/000892A patent/AP708A/en active
- 1996-12-12 UY UY24401A patent/UY24401A1/es not_active IP Right Cessation
- 1996-12-12 CO CO96065334A patent/CO4750831A1/es unknown
- 1996-12-13 HR HR60/008,753A patent/HRP960592A2/xx not_active Application Discontinuation
- 1996-12-13 ZA ZA9610533A patent/ZA9610533B/xx unknown
-
1998
- 1998-05-22 IS IS4752A patent/IS4752A/is unknown
- 1998-06-05 OA OA9800076A patent/OA10694A/en unknown
- 1998-06-09 BG BG102525A patent/BG102525A/xx unknown
- 1998-06-12 NO NO982712A patent/NO982712L/no not_active Application Discontinuation
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR004368A1 (es) | Compuestos de piperidina -1,-4 sustituida, procedimientos para prepararlos y un procedimiento para preparar 1-bencil-4-((5,6-dimetoxi-1-indanon)-2-il)metilpiperidina mediante dichos compuestos. | |
| ATE224715T1 (de) | Formulierung von d-threo methylphenidat mit verzögerter freisetzung | |
| DK0855999T3 (da) | 1-(1,2-disubstituerede piperidinyl)-4-substituerede piperidinderivater som tachykininreceptorantagonister | |
| DE3784669D1 (de) | Vorrichtung zum befestigen einer ersatzbahn, die eine programmierte bewegung durchfuehrt, ohne eine solche bewegung zu unterbrechen. | |
| DK0862566T3 (da) | 1-(1,2-Disubstitueret piperidinyl)-4-substituerede piperazindeivater | |
| DK204388A (da) | Substituerede piperidiner til anvendelse som opioidantagonister og fremgangsmaade til fremstilling af saadenne forbindelser | |
| DK0843679T3 (da) | 1-(1,2-disubstitueret piperidinyl)-4-(kondenseret midazol)-piperidinderivater | |
| FR2628312B1 (fr) | Agrafe chirurgicale, et outil impacteur servant a son implantation | |
| FR2653989B1 (fr) | Implant dentaire, outillage et procede de mise en place. | |
| NO982406D0 (no) | N-acyl-2-substituert-4-(benzimidazolyl-eller imidazopyridinyl-substituerte residuer)-piperidiner som tachykinin antagonister | |
| DE69007213D1 (de) | Leistungsapparat, Leistungsübertrager/Verteilereinheit, sowie ein Auslöseverfahren hierfür. | |
| IT1277329B1 (it) | Procedimento per la metilazione del 2,2,6,6-tetrametil-4-piperidone (triacetonammina) | |
| ECSP961971A (es) | Procedimientos e intermedios para preparar 1 - bencil-4-(5,6-dimetoxi -1-indanon)- 2--il)metilpiperidina | |
| DK215388D0 (da) | Fremgangsmaade og indretning til renovering af en fra en vaeg udragende, armeret betonplade | |
| KR970006301A (ko) | -피페리딘 또는 테트라하이드로피리딘 아자비사이클로카복스아미드 | |
| ES556011A0 (es) | Procedimiento para la obtencion de la 6-(2-(4-(bis(4-fluorofenil)metileno)piperidino)etil)-7-metil-5h-tiazolo(3,2-a)-pirimidin-5-ona | |
| ES556012A0 (es) | Procedimiento para la obtencion de la 6-(2-(4-(bis(4-fluorofenil)metileno)piperidino)etil)-7-metil-5h-tiazolo(3,2-a)-pirimidin-5-ona | |
| SI0765311T1 (en) | 4-aryl-1-(indanmethyl, dihydrobenzofuranmethyl or dihydrobenzothiophenemethyl)piperidines, tetrahydropyridines or piperazines | |
| DK89588A (da) | Fremgangsmaade og maskine til boejning af bygningsstaalsnet til boejlekurve |