AP2014007469A0 - Substituted 3-(BIPHENYL-3-YL)-4-hydroxy-8-METHOXY-1-azaspiro[4.5]DEC-3-EN-2-one - Google Patents

Substituted 3-(BIPHENYL-3-YL)-4-hydroxy-8-METHOXY-1-azaspiro[4.5]DEC-3-EN-2-one

Info

Publication number
AP2014007469A0
AP2014007469A0 AP2014007469A AP2014007469A AP2014007469A0 AP 2014007469 A0 AP2014007469 A0 AP 2014007469A0 AP 2014007469 A AP2014007469 A AP 2014007469A AP 2014007469 A AP2014007469 A AP 2014007469A AP 2014007469 A0 AP2014007469 A0 AP 2014007469A0
Authority
AP
ARIPO
Prior art keywords
azaspiro
biphenyl
methoxy
dec
hydroxy
Prior art date
Application number
AP2014007469A
Other languages
English (en)
Inventor
Reiner Fischer
Christoph-Stephan Hilger
Ningshu Liu
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Publication of AP2014007469A0 publication Critical patent/AP2014007469A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/54—Spiro-condensed
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)
AP2014007469A 2011-08-04 2012-07-31 Substituted 3-(BIPHENYL-3-YL)-4-hydroxy-8-METHOXY-1-azaspiro[4.5]DEC-3-EN-2-one AP2014007469A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102011080406A DE102011080406A1 (de) 2011-08-04 2011-08-04 Substituierte 3-(Biphenyl-3-yl)-4-hydroxy-8-methoxy-1-azaspiro8[4.5]dec-3-en-2-one
PCT/EP2012/064974 WO2013017600A1 (de) 2011-08-04 2012-07-31 Substituierte 3-(biphenyl-3-yl)-4-hydroxy-8-methoxy-1-azaspiro[4.5]dec-3-en-2-one

Publications (1)

Publication Number Publication Date
AP2014007469A0 true AP2014007469A0 (en) 2014-02-28

Family

ID=46584054

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2014007469A AP2014007469A0 (en) 2011-08-04 2012-07-31 Substituted 3-(BIPHENYL-3-YL)-4-hydroxy-8-METHOXY-1-azaspiro[4.5]DEC-3-EN-2-one

Country Status (21)

Country Link
US (1) US9278925B2 (xx)
EP (1) EP2739607A1 (xx)
JP (1) JP2014524413A (xx)
KR (1) KR20140051378A (xx)
CN (1) CN103842337A (xx)
AP (1) AP2014007469A0 (xx)
AU (1) AU2012292069A1 (xx)
BR (1) BR112014002674A2 (xx)
CA (1) CA2843809A1 (xx)
CO (1) CO6870039A2 (xx)
CR (1) CR20140063A (xx)
CU (1) CU20140012A7 (xx)
DE (1) DE102011080406A1 (xx)
DO (1) DOP2014000022A (xx)
EC (1) ECSP14013192A (xx)
HK (1) HK1198167A1 (xx)
IL (1) IL230609A0 (xx)
MX (1) MX2014001393A (xx)
SG (1) SG2014005235A (xx)
TN (1) TN2014000046A1 (xx)
WO (1) WO2013017600A1 (xx)

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EP3043800A1 (en) 2013-09-12 2016-07-20 Pfizer Inc. Use of acetyl-coa carboxylase inhibitors for treating acne vulgaris
EP3059225A4 (en) 2013-10-17 2017-09-06 Shionogi & Co., Ltd. Novel alkylene derivative
EP3225618B1 (en) 2014-11-26 2020-05-06 Takeda Pharmaceutical Company Limited Bicyclic compound
WO2016159049A1 (ja) 2015-03-31 2016-10-06 武田薬品工業株式会社 単環式化合物
TWI767148B (zh) 2018-10-10 2022-06-11 美商弗瑪治療公司 抑制脂肪酸合成酶(fasn)
RU2733369C1 (ru) * 2020-01-15 2020-10-01 Федеральное государственное бюджетное учреждение науки Федеральный исследовательский центр "КОМИ научный центр Уральского отделения Российской академии наук" Хиральные трифторметилированные монотерпеновые тиоацетаты и тиолы пинанового ряда
RU2743302C1 (ru) * 2020-07-21 2021-02-16 Федеральное государственное бюджетное учреждение науки Федеральный исследовательский центр "КОМИ научный центр Уральского отделения Российской академии наук" Хиральные трифторметилированные монотерпеновые тиоацетаты и тиолы на основе миртеналя

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Also Published As

Publication number Publication date
DE102011080406A1 (de) 2013-02-07
WO2013017600A1 (de) 2013-02-07
CA2843809A1 (en) 2013-02-07
TN2014000046A1 (en) 2015-07-01
MX2014001393A (es) 2014-05-27
BR112014002674A2 (pt) 2017-04-11
US20140275199A1 (en) 2014-09-18
CR20140063A (es) 2014-03-19
DOP2014000022A (es) 2014-03-31
KR20140051378A (ko) 2014-04-30
IL230609A0 (en) 2014-03-31
CU20140012A7 (es) 2014-05-27
EP2739607A1 (de) 2014-06-11
HK1198167A1 (xx) 2015-03-13
US9278925B2 (en) 2016-03-08
AU2012292069A1 (en) 2014-02-13
ECSP14013192A (es) 2014-03-31
CN103842337A (zh) 2014-06-04
SG2014005235A (en) 2014-06-27
CO6870039A2 (es) 2014-02-20
JP2014524413A (ja) 2014-09-22

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