AP2005003283A0 - Indole derivatives useful for the treatment os diseases - Google Patents

Indole derivatives useful for the treatment os diseases

Info

Publication number
AP2005003283A0
AP2005003283A0 AP2005003283A AP2005003283A AP2005003283A0 AP 2005003283 A0 AP2005003283 A0 AP 2005003283A0 AP 2005003283 A AP2005003283 A AP 2005003283A AP 2005003283 A AP2005003283 A AP 2005003283A AP 2005003283 A0 AP2005003283 A0 AP 2005003283A0
Authority
AP
ARIPO
Prior art keywords
diseases
treatment
indole derivatives
derivatives useful
useful
Prior art date
Application number
AP2005003283A
Other languages
English (en)
Inventor
Alan Daniel Brown
Mark Edward Et Al Bunnage
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP20020292513 external-priority patent/EP1407769A1/en
Priority claimed from EP03290069A external-priority patent/EP1440966A1/en
Application filed by Pfizer filed Critical Pfizer
Publication of AP2005003283A0 publication Critical patent/AP2005003283A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
AP2005003283A 2002-10-11 2003-10-06 Indole derivatives useful for the treatment os diseases AP2005003283A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP20020292513 EP1407769A1 (en) 2002-10-11 2002-10-11 Indole derivatives as beta-2 agonists
EP03290069A EP1440966A1 (en) 2003-01-10 2003-01-10 Indole derivatives useful for the treatment of diseases
PCT/IB2003/004441 WO2004032921A1 (en) 2002-10-11 2003-10-06 Indole derivatives as beta-2 agonists

Publications (1)

Publication Number Publication Date
AP2005003283A0 true AP2005003283A0 (en) 2005-06-30

Family

ID=32095049

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2005003283A AP2005003283A0 (en) 2002-10-11 2003-10-06 Indole derivatives useful for the treatment os diseases

Country Status (25)

Country Link
EP (1) EP1556034B1 (enExample)
JP (1) JP4490911B2 (enExample)
KR (1) KR20050047552A (enExample)
AP (1) AP2005003283A0 (enExample)
AR (1) AR041566A1 (enExample)
AT (1) ATE392206T1 (enExample)
AU (1) AU2003269316A1 (enExample)
BR (1) BR0315234A (enExample)
CA (1) CA2499314C (enExample)
CO (1) CO5550421A2 (enExample)
DE (1) DE60320439T2 (enExample)
EA (1) EA200500618A1 (enExample)
EC (1) ECSP055780A (enExample)
ES (1) ES2302938T3 (enExample)
IS (1) IS7751A (enExample)
MA (1) MA27452A1 (enExample)
MX (1) MXPA05003866A (enExample)
NO (1) NO20051406L (enExample)
OA (1) OA12938A (enExample)
PA (1) PA8586001A1 (enExample)
PE (1) PE20040775A1 (enExample)
PL (1) PL376396A1 (enExample)
TW (1) TW200424171A (enExample)
UY (1) UY28013A1 (enExample)
WO (1) WO2004032921A1 (enExample)

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JP5584138B2 (ja) 2008-01-11 2014-09-03 ノバルティス アーゲー キナーゼ阻害剤としてのピリミジン類
JP4837800B2 (ja) 2008-05-13 2011-12-14 アストラゼネカ・アクチエボラーグ ムスカリンｍ３受容体アンタゴニストとしてのキヌクリジン誘導体
CA2721065C (en) 2008-05-27 2016-09-27 Astrazeneca Ab Phenoxypyridinylamide derivatives and their use as pde4 inhibitors
EP2300010B1 (en) 2008-06-10 2015-03-04 Novartis AG Pyrazine derivatives as epithelial sodium channel blockers
US8236786B2 (en) 2008-08-07 2012-08-07 Pulmagen Therapeutics (Inflammation) Limited Respiratory disease treatment
WO2010067102A1 (en) 2008-12-09 2010-06-17 Astrazeneca Ab Diazaspiro [5.5] undecane derivatives and related compounds as muscarinic-receptor antagonists and beta-adrenoreceptor agonists for the treatment of pulmonary disorders
WO2010076553A1 (en) 2008-12-30 2010-07-08 Dr. Reddy's Laboratories Ltd Sulfonamide compounds for the treatment of respiratory disorders
WO2010150014A1 (en) 2009-06-24 2010-12-29 Pulmagen Therapeutics (Inflammation) Limited 5r- 5 -deuterated glitazones for respiratory disease treatment
JP5801997B2 (ja) 2009-07-07 2015-10-28 ファイザー・リミテッドＰｆｉｚｅｒ Ｌｉｍｉｔｅｄ 薬品の組合せを吸入するための投薬ユニット、投薬ユニットのパック、および吸入器
MX2012004792A (es) 2009-10-22 2013-02-01 Vertex Pharma Composiciones para el tratamiento de fibrosis quistica y otras enfermedades cronicas.
GB0918924D0 (en) 2009-10-28 2009-12-16 Vantia Ltd Azaindole derivatives
GB0918922D0 (en) 2009-10-28 2009-12-16 Vantia Ltd Aminopyridine derivatives
GB0918923D0 (en) 2009-10-28 2009-12-16 Vantia Ltd Aminothiazole derivatives
WO2011061527A1 (en) 2009-11-17 2011-05-26 Astrazeneca Ab Combinations comprising a glucocorticoid receptor modulator for the treatment of respiratory diseases
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US8247436B2 (en) 2010-03-19 2012-08-21 Novartis Ag Pyridine and pyrazine derivative for the treatment of CF
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UY33597A (es) 2010-09-09 2012-04-30 Irm Llc Compuestos y composiciones como inhibidores de la trk
US8372845B2 (en) 2010-09-17 2013-02-12 Novartis Ag Pyrazine derivatives as enac blockers
GB201016912D0 (en) 2010-10-07 2010-11-24 Astrazeneca Ab Novel combination
JP5959541B2 (ja) 2011-02-25 2016-08-02 ノバルティス アーゲー Ｔｒｋ阻害剤としてのピラゾロ［１，５−ａ］ピリジン
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Also Published As

Publication number Publication date
CA2499314A1 (en) 2004-04-22
ES2302938T3 (es) 2008-08-01
PL376396A1 (en) 2005-12-27
UY28013A1 (es) 2004-04-30
DE60320439D1 (de) 2008-05-29
KR20050047552A (ko) 2005-05-20
BR0315234A (pt) 2005-08-23
EA200500618A1 (ru) 2005-12-29
TW200424171A (en) 2004-11-16
JP4490911B2 (ja) 2010-06-30
AU2003269316A1 (en) 2004-05-04
EP1556034B1 (en) 2008-04-16
IS7751A (is) 2005-03-17
ATE392206T1 (de) 2008-05-15
AR041566A1 (es) 2005-05-18
NO20051406L (no) 2005-04-22
MXPA05003866A (es) 2005-06-22
PE20040775A1 (es) 2004-12-10
ECSP055780A (es) 2005-08-11
EP1556034A1 (en) 2005-07-27
WO2004032921A1 (en) 2004-04-22
DE60320439T2 (de) 2009-05-20
OA12938A (en) 2006-10-13
PA8586001A1 (es) 2005-02-04
JP2006511596A (ja) 2006-04-06
CO5550421A2 (es) 2005-08-31
MA27452A1 (fr) 2005-07-01
CA2499314C (en) 2010-08-24

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