ZA977103B - Benzopiperidine derivatives - Google Patents
Benzopiperidine derivativesInfo
- Publication number
- ZA977103B ZA977103B ZA977103A ZA977103A ZA977103B ZA 977103 B ZA977103 B ZA 977103B ZA 977103 A ZA977103 A ZA 977103A ZA 977103 A ZA977103 A ZA 977103A ZA 977103 B ZA977103 B ZA 977103B
- Authority
- ZA
- South Africa
- Prior art keywords
- benzopiperidine
- derivatives
- benzopiperidine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP21034496 | 1996-08-09 |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA977103B true ZA977103B (en) | 1999-02-08 |
Family
ID=16587858
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA977103A ZA977103B (en) | 1996-08-09 | 1997-08-08 | Benzopiperidine derivatives |
Country Status (7)
Country | Link |
---|---|
US (2) | US6518423B1 (ja) |
EP (1) | EP0934941A1 (ja) |
JP (1) | JP4028894B2 (ja) |
AU (1) | AU3784997A (ja) |
CA (1) | CA2262569A1 (ja) |
WO (1) | WO1998006720A1 (ja) |
ZA (1) | ZA977103B (ja) |
Families Citing this family (37)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU5240099A (en) * | 1998-07-31 | 2000-02-21 | Eli Lilly And Company | Heterocyclic sulphonamide derivatives |
TW526202B (en) * | 1998-11-27 | 2003-04-01 | Shionogi & Amp Co | Broad spectrum cephem having benzo[4,5-b]pyridium methyl group of antibiotic activity |
AU1857600A (en) * | 1998-12-22 | 2000-07-12 | Neurosearch A/S | Ion channel modulating agents |
TWI288745B (en) | 2000-04-05 | 2007-10-21 | Daiichi Seiyaku Co | Ethylenediamine derivatives |
AR034160A1 (es) * | 2000-09-30 | 2004-02-04 | Gruenenthal Gmbh | Sulfonilguanidinas, medicamentos que contienen estos compuestos y el uso de sulfonilguanidinas |
US20030087963A1 (en) | 2001-09-13 | 2003-05-08 | Senanayake Chris H. | Methods of preparing and using 2-hydroxy derivatives of sibutramine and its metabolites |
US7189724B2 (en) * | 2003-04-15 | 2007-03-13 | Valeant Research And Development | Quinoxaline derivatives having antiviral activity |
BRPI0412003A (pt) | 2003-07-02 | 2006-08-15 | Sugen Inc | arilmetil triazol e imidazopirazinas como inibidores de c-met |
JP5213089B2 (ja) * | 2004-04-19 | 2013-06-19 | 広栄化学工業株式会社 | アルキルアミノピリジン類の製造方法。 |
US7241776B2 (en) * | 2004-08-02 | 2007-07-10 | Abbott Laboratories | Cyanoamidine P2X7 antagonists for the treatment of pain |
AU2005295821A1 (en) * | 2004-10-12 | 2006-04-27 | Decode Genetics Ehf | Carboxylic acid peri - substituted bicyclics for occlusive artery disease |
WO2006066197A1 (en) * | 2004-12-17 | 2006-06-22 | Janssen Pharmaceutica, N.V. | Tetrahydroisoquinoline compounds for treatment of cns disorders |
BRPI0516407A (pt) * | 2004-12-24 | 2008-09-02 | Prosidion Ltd | agonistas de receptor acoplado à proteìna g (gpr116) e uso destes para o tratamento de obesidade e diabetes |
US20080261999A1 (en) * | 2005-03-04 | 2008-10-23 | Fionna Mitchell Martin | Azabicycloalkane Derivatives Useful as Nicotinic Acetylcholine Receptor Agonists |
CA2613235A1 (en) | 2005-06-30 | 2007-01-11 | Prosidion Limited | Gpcr agonists |
AR064735A1 (es) | 2007-01-04 | 2009-04-22 | Prosidion Ltd | Agonistas de gpcr y composicion farmaceutica en base al compuesto |
PT2114933E (pt) | 2007-01-04 | 2011-12-20 | Prosidion Ltd | Agonistas do gpcr de piperidina |
AR064736A1 (es) | 2007-01-04 | 2009-04-22 | Prosidion Ltd | Agonistas de gpcr |
WO2008117229A1 (en) * | 2007-03-23 | 2008-10-02 | Ranbaxy Laboratories Limited | Muscarinic receptor antagonists |
JP2010539152A (ja) | 2007-09-10 | 2010-12-16 | プロシディオン・リミテッド | 代謝障害の治療のための化合物 |
GB0812649D0 (en) * | 2008-07-10 | 2008-08-20 | Prosidion Ltd | Compounds |
WO2010004344A1 (en) * | 2008-07-10 | 2010-01-14 | Prosidion Limited | Piperidine gpcr agonists |
GB0812648D0 (en) * | 2008-07-10 | 2008-08-20 | Prosidion Ltd | Compounds |
FR2941696B1 (fr) | 2009-02-05 | 2011-04-15 | Sanofi Aventis | Derives d'azaspiranyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique |
US8580807B2 (en) | 2009-04-03 | 2013-11-12 | Merck Sharp & Dohme Corp. | Bicyclic piperidine and piperazine derivatives as GPCR modulators for the treatment of obesity, diabetes and other metabolic disorders |
FR2945531A1 (fr) * | 2009-05-12 | 2010-11-19 | Sanofi Aventis | Derives de 7-aza-spiro°3,5!nonane-7-carboxylates, leur preparation et leur application en therapeutique |
KR20110049217A (ko) * | 2009-11-04 | 2011-05-12 | 다우어드밴스드디스플레이머티리얼 유한회사 | 신규한 유기 발광 화합물 및 이를 채용하고 있는 유기 전계 발광 소자 |
CN102875467B (zh) * | 2011-07-12 | 2015-06-03 | 无锡药明康德生物技术有限公司 | 1,3-二取代-3-氮杂双环[3,3,1]壬烷衍生物及制备方法 |
FR2985511B1 (fr) * | 2012-01-05 | 2014-01-03 | Servier Lab | Forme cristalline delta du sel d'arginine du perindopril, son procede de preparation, et les compositions pharmaceutiques qui la contiennent |
CA2912057C (en) | 2013-05-10 | 2022-01-11 | University Of Pittsburgh - Of The Commonwealth System Of Higher Education | Treatment of pulmonary and other conditions |
US10457681B2 (en) * | 2017-08-16 | 2019-10-29 | Bristol_Myers Squibb Company | Toll-like receptor 7 (TLR7) agonists having a tricyclic moiety, conjugates thereof, and methods and uses therefor |
AU2019258078B2 (en) * | 2018-04-27 | 2023-12-21 | Chengdu Henghao Investment Co. Limited | 10H-phenothiazine ferroptosis inhibitor and preparation method therefor and application thereof |
CN113453760B (zh) | 2018-12-17 | 2024-05-24 | 弗特克斯药品有限公司 | Apol1抑制剂及其使用方法 |
IL300298A (en) | 2020-08-26 | 2023-04-01 | Vertex Pharma | Apol1 inhibitors and methods of using the same |
WO2023154310A1 (en) * | 2022-02-08 | 2023-08-17 | Vertex Pharmaceuticals Incorporated | 2-methyl-4-phenylpiperidin-4-ol derivatives as inhibitors of apol1 and methods of using same |
WO2023164940A1 (zh) * | 2022-03-04 | 2023-09-07 | 中国福利会国际和平妇幼保健院 | 氮杂吩噻嗪类化合物及其在制备治疗子宫内膜癌的药物中的应用 |
CN115353481B (zh) * | 2022-08-31 | 2024-03-29 | 宁夏格瑞精细化工有限公司 | 一种顺式-1,2,3,6-四氢邻苯二甲酰亚胺的催化合成方法 |
Family Cites Families (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR138F (ja) | 1964-11-30 | |||
FR1488269A (fr) | 1966-03-18 | 1967-07-13 | Chimetron Sarl | Phénothiazines et phénoxazines portant un substituant bicyclique |
FR1516746A (fr) | 1966-04-20 | 1968-02-05 | Rhone Poulenc Sa | Nouveaux dérivés de la phénoxazine et leur préparation |
GB1168094A (en) | 1967-02-14 | 1969-10-22 | Shell Int Research | Substituted Phenazines and their use as Herbicides |
US3808208A (en) * | 1970-02-02 | 1974-04-30 | Dow Chemical Co | P-benzodithino(dioxino)(2,3,-b)pyrazines |
US3663543A (en) * | 1970-02-02 | 1972-05-16 | Dow Chemical Co | 2,3-dichloro-5,10-dihydropyrazino(2,3-b) quinoxaline |
US3746707A (en) | 1970-02-02 | 1973-07-17 | Dow Chemical Co | Tricyclic pyrazino compounds and method for preparing the same |
US3821213A (en) * | 1972-10-24 | 1974-06-28 | Dow Chemical Co | Oxides of 10-h-pyrazino(2,3-b)(1,4)benzothiazine |
US3845044A (en) | 1972-10-24 | 1974-10-29 | Dow Chemical Co | Aminoalkyl derivatives of 10h-pyrazino(2,3-b)(1,4)benzothiazine |
DE2702714A1 (de) | 1977-01-24 | 1978-07-27 | Lek Tovarna Farmacevtskih | Verfahren zur herstellung von phenothiazin-derivaten |
US4370328A (en) | 1977-11-03 | 1983-01-25 | Pfizer Inc. | Cardiac stimulant 1-(3- or 4-substituted piperidino)phthalazines |
GB2007654B (en) | 1977-11-03 | 1982-06-16 | Pfizer Ltd | Therapeutic agents |
CA1086735A (en) * | 1977-11-03 | 1980-09-30 | John C. Danilewicz | Piperidino-quinazolines |
IL59619A0 (en) * | 1979-03-28 | 1980-06-30 | Pfizer | Phthalazine derivatives,their preparation and pharmaceutical compositions containing them |
US4264601A (en) * | 1979-06-12 | 1981-04-28 | The Board Of Regents Of The University Of Oklahoma | Antihypertensive agents and their use in treatment of hypertension |
US4223136A (en) * | 1979-08-03 | 1980-09-16 | G. D. Searle & Co. | 2,3-Dihydro-3-oxo-5H-pyrido[3,4-b][1,4]-benzothiazine-4-carbonitriles |
ES537162A0 (es) | 1983-10-31 | 1985-12-01 | Merck Frosst Canada Inc | Una composicion farmaceutica |
GB8516371D0 (en) | 1985-06-28 | 1985-07-31 | Beecham Group Plc | Compounds |
DE3627310A1 (de) | 1986-08-12 | 1988-02-18 | Biotechnolog Forschung Gmbh | Pyocyanin-derivate und herstellungsverfahren |
JP2969359B2 (ja) | 1989-01-13 | 1999-11-02 | 武田薬品工業株式会社 | 環状アミン化合物 |
JPH02225413A (ja) | 1989-02-28 | 1990-09-07 | Mitsubishi Kasei Corp | 抗潰瘍剤 |
PL167568B1 (pl) * | 1990-07-23 | 1995-09-30 | Pfizer | Sposób wytwarzania nowych pochodnych chinuklidyny PL PL |
CA2118798A1 (en) | 1991-09-12 | 1993-03-18 | Francis D. King | Azabicyclic compounds as 5-ht4 receptor antagonists |
ES2135414T3 (es) * | 1991-09-12 | 1999-11-01 | Smithkline Beecham Plc | Antagonistas del receptor 5-ht4. |
AU680004B2 (en) | 1993-05-26 | 1997-07-17 | Syntex (U.S.A.) Inc. | Novel 1-phenylalkanone 5-HT4 receptor ligands |
KR960704852A (ko) | 1993-09-30 | 1996-10-09 | 오노다 마사요시 | 아졸 유도체 및 이의 약제학적 조성물 (Azole derivative and pharmaceutical composition thereof) |
US5707994A (en) | 1993-10-19 | 1998-01-13 | Sumitomo Pharmaceuticals Company, Limited | 2,3-diaminopropionic acid derivative |
GB9404806D0 (en) | 1994-03-11 | 1994-04-27 | Minnesota Mining & Mfg | Monoaminophenzaine leuco dyes and photothermographic materials |
-
1997
- 1997-08-08 AU AU37849/97A patent/AU3784997A/en not_active Abandoned
- 1997-08-08 WO PCT/JP1997/002787 patent/WO1998006720A1/ja not_active Application Discontinuation
- 1997-08-08 CA CA002262569A patent/CA2262569A1/en not_active Abandoned
- 1997-08-08 JP JP50958998A patent/JP4028894B2/ja not_active Expired - Fee Related
- 1997-08-08 EP EP97934750A patent/EP0934941A1/en not_active Withdrawn
- 1997-08-08 US US09/230,852 patent/US6518423B1/en not_active Expired - Fee Related
- 1997-08-08 ZA ZA977103A patent/ZA977103B/xx unknown
-
2002
- 2002-09-20 US US10/247,310 patent/US20040092737A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
EP0934941A1 (en) | 1999-08-11 |
US20040092737A1 (en) | 2004-05-13 |
WO1998006720A1 (fr) | 1998-02-19 |
US6518423B1 (en) | 2003-02-11 |
JP4028894B2 (ja) | 2007-12-26 |
AU3784997A (en) | 1998-03-06 |
CA2262569A1 (en) | 1998-02-19 |
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