ZA938089B - Novel antimicrobial 5-(N-heterosubstituted amino) quinolones - Google Patents
Novel antimicrobial 5-(N-heterosubstituted amino) quinolonesInfo
- Publication number
- ZA938089B ZA938089B ZA938089A ZA938089A ZA938089B ZA 938089 B ZA938089 B ZA 938089B ZA 938089 A ZA938089 A ZA 938089A ZA 938089 A ZA938089 A ZA 938089A ZA 938089 B ZA938089 B ZA 938089B
- Authority
- ZA
- South Africa
- Prior art keywords
- quinolones
- novel antimicrobial
- heterosubstituted amino
- heterosubstituted
- amino
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US96896092A | 1992-10-30 | 1992-10-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA938089B true ZA938089B (en) | 1994-06-07 |
Family
ID=25514997
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA938089A ZA938089B (en) | 1992-10-30 | 1993-10-29 | Novel antimicrobial 5-(N-heterosubstituted amino) quinolones |
Country Status (21)
| Country | Link |
|---|---|
| EP (1) | EP0666853A1 (ko) |
| JP (1) | JPH08502750A (ko) |
| KR (1) | KR950704301A (ko) |
| CN (1) | CN1064357C (ko) |
| AU (1) | AU687018B2 (ko) |
| BR (1) | BR9307347A (ko) |
| CA (1) | CA2148003A1 (ko) |
| CZ (1) | CZ282581B6 (ko) |
| EG (1) | EG20543A (ko) |
| FI (1) | FI952049A0 (ko) |
| HU (1) | HUT72072A (ko) |
| IL (1) | IL107323A (ko) |
| MX (1) | MX9306814A (ko) |
| NO (1) | NO951640L (ko) |
| NZ (1) | NZ257470A (ko) |
| PL (1) | PL178094B1 (ko) |
| RU (1) | RU2126000C1 (ko) |
| SG (1) | SG59979A1 (ko) |
| SK (1) | SK54795A3 (ko) |
| WO (1) | WO1994010163A1 (ko) |
| ZA (1) | ZA938089B (ko) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5646163A (en) * | 1992-10-30 | 1997-07-08 | The Procter & Gamble Company | Quinolone 5-(N-heterosubstituted amino) antimicrobials |
| WO1996004247A1 (en) * | 1994-08-02 | 1996-02-15 | The Procter & Gamble Company | Process for making antimicrobial compounds |
| JPH10503521A (ja) * | 1994-08-02 | 1998-03-31 | ザ、プロクター、エンド、ギャンブル、カンパニー | キノロニルラクタム抗微生物剤の製造方法及び新規中間化合物 |
| WO1997029102A1 (fr) * | 1996-02-09 | 1997-08-14 | Toyama Chemical Co., Ltd. | Derives de l'acide quinolonecarboxylique et leurs sels |
| US8524734B2 (en) | 2005-05-18 | 2013-09-03 | Mpex Pharmaceuticals, Inc. | Aerosolized fluoroquinolones and uses thereof |
| AU2006247053B2 (en) * | 2005-05-18 | 2013-05-23 | Horizon Therapeutics U.S. Holding Llc | Aerosolized fluoroquinolones and uses thereof |
| CA2528849C (en) | 2005-06-08 | 2014-01-14 | Janssen Pharmaceutica N.V. | Quinoline derivatives as antibacterial agents |
| EA010601B1 (ru) * | 2005-06-09 | 2008-10-30 | Янссен Фармацевтика Н.В. | Производные хинолина в качестве антибактериальных агентов |
| CN101020647B (zh) * | 2007-02-14 | 2011-03-30 | 杭州师范学院 | 一种β-环丙胺基丙烯酸(酯)的合成方法 |
| EP2150544B1 (en) * | 2007-03-19 | 2016-01-13 | Takeda Pharmaceutical Company Limited | Mapk/erk kinase inhibitors |
| EP2214491B1 (en) * | 2007-10-05 | 2016-07-13 | Senhwa Biosciences, Inc. | Quinolone analogs and methods related thereto |
| EP2297107B1 (en) * | 2008-06-03 | 2013-11-13 | Actelion Pharmaceuticals Ltd. | [4-(1-amino-ethyl) -cyclohexyl]-methyl-amine and [6-(1-amino-ethyl) -tetrahydro- pyran-3-yl]-methyl-amine derivatives as antibacterials |
| DK2346509T3 (da) | 2008-10-07 | 2020-08-03 | Horizon Orphan Llc | Inhalation af levofloxacin til at reducere lungeinflammation |
| BRPI0920026B1 (pt) | 2008-10-07 | 2023-11-07 | Horizon Orphan Llc | Composição farmacêutica e respectivos usos |
| AR076222A1 (es) * | 2009-04-09 | 2011-05-26 | Actelion Pharmaceuticals Ltd | Derivados 2-hidroxietil-1h-quinolin-ona y sus analogos azaisotericos con actividad antibacteriana y composiciones farmaceuticas que los contienen |
| IN2012DN02477A (ko) | 2009-09-04 | 2015-08-21 | Mpex Pharmaceuticals Inc |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4668680A (en) * | 1985-12-12 | 1987-05-26 | Warner-Lambert Company | 5-amino-6,8-difluoroquinolones as antibacterial agents |
| JPH0228178A (ja) * | 1988-04-23 | 1990-01-30 | Toyama Chem Co Ltd | 新規なピリドンカルボン酸誘導体およびその塩並びにそれらの製造法 |
| DE3906365A1 (de) * | 1988-07-15 | 1990-01-18 | Bayer Ag | 7-(1-pyrrolidinyl)-3-chinolon- und -naphthyridoncarbonsaeure-derivate, verfahren sowie substituierte (oxa)diazabicyclooctane und -nonane als zwischenprodukte zu ihrer herstellung, und sie enthaltende antibakterielle mittel und futterzusatzstoffe |
| WO1991002526A1 (en) * | 1989-08-16 | 1991-03-07 | Pfizer Inc. | Azabicyclo quinolone carboxylic acids |
| EP0525057B1 (en) * | 1990-04-18 | 2000-06-14 | Procter & Gamble Pharmaceuticals, Inc. | Antimicrobial quinolonyl lactams |
| ES2137942T3 (es) * | 1990-11-30 | 2000-01-01 | Warner Lambert Co | Estereoisomeros individuales de 7-(3-(aminoalquil)-1-pirrolidinil)-quinolonas y de naftiridonas utilizados como agentes antibacterianos. |
-
1993
- 1993-01-30 EG EG68693A patent/EG20543A/xx active
- 1993-10-19 IL IL10732393A patent/IL107323A/xx not_active IP Right Cessation
- 1993-10-22 KR KR1019950701690A patent/KR950704301A/ko active IP Right Grant
- 1993-10-22 NZ NZ257470A patent/NZ257470A/xx unknown
- 1993-10-22 BR BR9307347A patent/BR9307347A/pt not_active Application Discontinuation
- 1993-10-22 CZ CZ951097A patent/CZ282581B6/cs not_active IP Right Cessation
- 1993-10-22 PL PL93308671A patent/PL178094B1/pl unknown
- 1993-10-22 RU RU95110762A patent/RU2126000C1/ru active
- 1993-10-22 EP EP93924393A patent/EP0666853A1/en not_active Withdrawn
- 1993-10-22 SG SG1996007851A patent/SG59979A1/en unknown
- 1993-10-22 JP JP6511167A patent/JPH08502750A/ja active Pending
- 1993-10-22 CA CA002148003A patent/CA2148003A1/en not_active Abandoned
- 1993-10-22 SK SK547-95A patent/SK54795A3/sk unknown
- 1993-10-22 WO PCT/US1993/010091 patent/WO1994010163A1/en not_active Application Discontinuation
- 1993-10-22 AU AU54097/94A patent/AU687018B2/en not_active Ceased
- 1993-10-22 HU HU9501237A patent/HUT72072A/hu unknown
- 1993-10-29 ZA ZA938089A patent/ZA938089B/xx unknown
- 1993-10-29 MX MX9306814A patent/MX9306814A/es not_active IP Right Cessation
- 1993-10-30 CN CN93120224A patent/CN1064357C/zh not_active Expired - Fee Related
-
1995
- 1995-04-28 NO NO951640A patent/NO951640L/no unknown
- 1995-04-28 FI FI952049A patent/FI952049A0/fi unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CZ109795A3 (en) | 1995-12-13 |
| IL107323A (en) | 2000-06-01 |
| RU2126000C1 (ru) | 1999-02-10 |
| FI952049A (fi) | 1995-04-28 |
| CZ282581B6 (cs) | 1997-08-13 |
| BR9307347A (pt) | 1999-05-25 |
| SG59979A1 (en) | 1999-02-22 |
| KR950704301A (ko) | 1995-11-17 |
| SK54795A3 (en) | 1995-12-06 |
| PL178094B1 (pl) | 2000-02-29 |
| JPH08502750A (ja) | 1996-03-26 |
| CN1064357C (zh) | 2001-04-11 |
| FI952049A0 (fi) | 1995-04-28 |
| RU95110762A (ru) | 1997-01-10 |
| CN1092773A (zh) | 1994-09-28 |
| IL107323A0 (en) | 1994-01-25 |
| EP0666853A1 (en) | 1995-08-16 |
| HU9501237D0 (en) | 1995-06-28 |
| WO1994010163A1 (en) | 1994-05-11 |
| MX9306814A (es) | 1994-07-29 |
| NO951640D0 (no) | 1995-04-28 |
| EG20543A (en) | 1999-07-31 |
| HUT72072A (en) | 1996-03-28 |
| AU5409794A (en) | 1994-05-24 |
| AU687018B2 (en) | 1998-02-19 |
| NZ257470A (en) | 1997-08-22 |
| CA2148003A1 (en) | 1994-05-11 |
| NO951640L (no) | 1995-06-30 |
| PL308671A1 (en) | 1995-08-21 |
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