ZA793453B - New 3,20-dioxo-4,9-diene-21-hydroxyl steroid derivatives,a process for preparing them,their use as medicaments and the pharmaceutical compositions containing them - Google Patents
New 3,20-dioxo-4,9-diene-21-hydroxyl steroid derivatives,a process for preparing them,their use as medicaments and the pharmaceutical compositions containing themInfo
- Publication number
- ZA793453B ZA793453B ZA793453A ZA793453A ZA793453B ZA 793453 B ZA793453 B ZA 793453B ZA 793453 A ZA793453 A ZA 793453A ZA 793453 A ZA793453 A ZA 793453A ZA 793453 B ZA793453 B ZA 793453B
- Authority
- ZA
- South Africa
- Prior art keywords
- dioxo
- medicaments
- diene
- preparing
- new
- Prior art date
Links
- 239000003814 drug Substances 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 125000004432 carbon atom Chemical group C* 0.000 abstract 3
- YZCKVEUIGOORGS-NJFSPNSNSA-N Tritium Chemical group [3H] YZCKVEUIGOORGS-NJFSPNSNSA-N 0.000 abstract 1
- 230000001833 anti-estrogenic effect Effects 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000000962 progestomimetic effect Effects 0.000 abstract 1
- 229910052722 tritium Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Investigating Or Analysing Biological Materials (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7820973A FR2430953A1 (fr) | 1978-07-13 | 1978-07-13 | Nouveaux derives 3,20-dioxo 4,9-diene 21-hydroxyle, leur procede de preparation et leur application comme medicaments |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA793453B true ZA793453B (en) | 1980-06-25 |
Family
ID=9210732
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA793453A ZA793453B (en) | 1978-07-13 | 1979-07-10 | New 3,20-dioxo-4,9-diene-21-hydroxyl steroid derivatives,a process for preparing them,their use as medicaments and the pharmaceutical compositions containing them |
Country Status (15)
Country | Link |
---|---|
US (1) | US4273771A (de) |
EP (2) | EP0007823B1 (de) |
JP (2) | JPS5515475A (de) |
AT (1) | ATE8899T1 (de) |
AU (1) | AU527592B2 (de) |
CA (1) | CA1131215A (de) |
DE (1) | DE2965904D1 (de) |
DK (2) | DK163361C (de) |
ES (1) | ES482112A1 (de) |
FR (1) | FR2430953A1 (de) |
HU (1) | HU178088B (de) |
IE (1) | IE49457B1 (de) |
IL (1) | IL57691A (de) |
PT (1) | PT69903A (de) |
ZA (1) | ZA793453B (de) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5830145A (ja) * | 1981-08-17 | 1983-02-22 | Sony Corp | 半導体装置の製造方法 |
FR2549067B1 (fr) * | 1983-06-14 | 1985-12-27 | Roussel Uclaf | Derives estradieniques radioactifs marques au tritium, leur procede de preparation et leur application pour l'etude et le dosage radio-immunologique de steroides dans les fluides biologiques |
US4804541A (en) * | 1987-08-11 | 1989-02-14 | Moleculon, Inc. | Transdermal administration using benzyl alcohol |
US5516790A (en) * | 1989-01-23 | 1996-05-14 | Texas A&M University System Technology Licensing Office | Synthesis and application of alkyl-substituted dibenzofurans as antitumorigenic agents |
FR2692267B1 (fr) * | 1992-06-11 | 1995-05-19 | Roussel Uclaf | Nouveau procédé de préparation de composés stéroïdes 20-céto 21alpha-hydroxy et intermédiaires. |
FR2694007B1 (fr) * | 1992-07-23 | 1994-09-30 | Roussel Uclaf | Nouveau procédé de préparation de composés stéroïdes 20-céto 21 (S) hydroxy et des intermédiaires. |
FR2749012B1 (fr) * | 1996-05-22 | 1998-08-07 | Hoechst Marion Roussel Inc | Nouveaux steroides 1 ou 6-hydroxyles, leur procede de preparation, leur application a titre de medicament et les compositions pharmaceutiques les renfermant |
FR2749514B1 (fr) * | 1996-06-11 | 1998-08-07 | Hoechst Marion Roussel | Systemes transdermiques renfermant 2 principes actifs dans des compartiments separes, leur procede de preparation et leur application comme medicament |
FR2749586B1 (fr) * | 1996-06-11 | 1998-08-07 | Hoechst Marion Roussel Inc | Nouveaux dispositifs destines a l'administration transdermique de la trimegestone, leur procede de preparation et leur application a titre de medicaments |
US5858405A (en) * | 1996-07-26 | 1999-01-12 | American Home Products Corporation | Oral contraceptive |
US5888543A (en) * | 1996-07-26 | 1999-03-30 | American Home Products Corporation | Oral contraceptives |
US6451778B1 (en) | 1996-07-26 | 2002-09-17 | Wyeth | Oral contraceptive |
US6479475B1 (en) | 1996-07-26 | 2002-11-12 | Wyeth | Oral contraceptive |
JP2004522754A (ja) * | 2001-02-02 | 2004-07-29 | ファルマシア・コーポレーション | 月経困難症の治療および予防のための組み合わせ治療としてシクロオキシゲナーゼ‐2阻害剤および性ステロイドを使用する方法 |
TW200306846A (en) * | 2002-04-03 | 2003-12-01 | Wyeth Corp | Hormone replacement therapy |
ITMI20042001A1 (it) * | 2004-10-21 | 2005-01-21 | Ind Chimica Srl | Processo per la preparazione di 21-idrossi steroidi con controllo della distribuzione epimerica nella posizione c-21 |
DE102005034498A1 (de) * | 2005-07-20 | 2007-01-25 | Grünenthal GmbH | Orale Kontrazeption mit Trimegeston |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB902373A (en) * | 1960-01-22 | 1962-08-01 | Pfizer & Co C | Steroids and preparation thereof |
US3810885A (en) * | 1967-12-12 | 1974-05-14 | Roussel Uclaf | Novel steroids and processes |
FR2077877B1 (de) * | 1970-02-20 | 1974-02-01 | Roussel Uclaf | |
FR2149302A1 (en) * | 1971-08-19 | 1973-03-30 | Roussel Uclaf | 21-methyl pregnadienes prepn - used as progestomimetics |
US3923414A (en) * | 1973-07-16 | 1975-12-02 | Valeron Corp | Vibration damping support |
FR2385737A1 (fr) * | 1977-04-01 | 1978-10-27 | Roussel Uclaf | Nouveaux steroides, leur procede de preparation et leur application dans la synthese de steroides marques au tritium |
FR2374335A1 (fr) * | 1976-12-14 | 1978-07-13 | Roussel Uclaf | Nouveaux steroides, leur procede de preparation et leur application dans la synthese de steroides marques au tritium |
JPS5894940U (ja) * | 1981-12-21 | 1983-06-28 | 日野自動車株式会社 | ビスカスダンパ |
-
1978
- 1978-07-13 FR FR7820973A patent/FR2430953A1/fr active Granted
-
1979
- 1979-06-21 HU HU79RO1026A patent/HU178088B/hu unknown
- 1979-06-27 AT AT81201106T patent/ATE8899T1/de active
- 1979-06-27 DE DE7979400426T patent/DE2965904D1/de not_active Expired
- 1979-06-27 EP EP79400426A patent/EP0007823B1/de not_active Expired
- 1979-06-27 EP EP81201106A patent/EP0046001B1/de not_active Expired
- 1979-06-29 IL IL57691A patent/IL57691A/xx unknown
- 1979-07-02 ES ES482112A patent/ES482112A1/es not_active Expired
- 1979-07-05 US US06/055,019 patent/US4273771A/en not_active Expired - Lifetime
- 1979-07-10 ZA ZA793453A patent/ZA793453B/xx unknown
- 1979-07-10 PT PT69903A patent/PT69903A/pt active IP Right Revival
- 1979-07-12 DK DK292579A patent/DK163361C/da not_active IP Right Cessation
- 1979-07-12 CA CA331,655A patent/CA1131215A/fr not_active Expired
- 1979-07-12 AU AU48895/79A patent/AU527592B2/en not_active Expired
- 1979-07-13 JP JP8839679A patent/JPS5515475A/ja active Granted
- 1979-08-08 IE IE1339/79A patent/IE49457B1/en not_active IP Right Cessation
-
1987
- 1987-06-29 JP JP62159945A patent/JPS6333395A/ja active Granted
-
1991
- 1991-07-16 DK DK136391A patent/DK165637C/da not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
DK136391A (da) | 1991-07-16 |
JPS6333395A (ja) | 1988-02-13 |
HU178088B (en) | 1982-03-28 |
EP0007823A2 (de) | 1980-02-06 |
JPS5515475A (en) | 1980-02-02 |
IL57691A (en) | 1983-10-31 |
DK163361B (da) | 1992-02-24 |
PT69903A (fr) | 1979-08-01 |
DK165637B (da) | 1992-12-28 |
EP0007823A3 (en) | 1980-05-14 |
JPS6254119B2 (de) | 1987-11-13 |
EP0007823B1 (de) | 1983-07-20 |
IE49457B1 (en) | 1985-10-16 |
EP0046001B1 (de) | 1984-08-08 |
ATE8899T1 (de) | 1984-08-15 |
AU527592B2 (en) | 1983-03-10 |
EP0046001A1 (de) | 1982-02-17 |
DK136391D0 (da) | 1991-07-16 |
US4273771A (en) | 1981-06-16 |
IL57691A0 (en) | 1979-10-31 |
JPH027600B2 (de) | 1990-02-19 |
DK165637C (da) | 1993-06-01 |
IE791339L (en) | 1980-01-13 |
DE2965904D1 (en) | 1983-08-25 |
CA1131215A (fr) | 1982-09-07 |
FR2430953B1 (de) | 1981-09-11 |
FR2430953A1 (fr) | 1980-02-08 |
ES482112A1 (es) | 1980-07-01 |
DK163361C (da) | 1992-07-13 |
DK292579A (da) | 1980-01-14 |
AU4889579A (en) | 1980-01-17 |
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