DK165637C - Mellemprodukter til brug ved fremstilling af 3,20-dioxo-4,9-dien-21-hydroxylsteroider - Google Patents

Mellemprodukter til brug ved fremstilling af 3,20-dioxo-4,9-dien-21-hydroxylsteroider

Info

Publication number
DK165637C
DK165637C DK136391A DK136391A DK165637C DK 165637 C DK165637 C DK 165637C DK 136391 A DK136391 A DK 136391A DK 136391 A DK136391 A DK 136391A DK 165637 C DK165637 C DK 165637C
Authority
DK
Denmark
Prior art keywords
preparation
intermediates
dioxo
diene
alkyl
Prior art date
Application number
DK136391A
Other languages
English (en)
Other versions
DK136391A (da
DK165637B (da
DK136391D0 (da
Inventor
Daniel Coussediere
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of DK136391A publication Critical patent/DK136391A/da
Publication of DK136391D0 publication Critical patent/DK136391D0/da
Publication of DK165637B publication Critical patent/DK165637B/da
Application granted granted Critical
Publication of DK165637C publication Critical patent/DK165637C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
DK136391A 1978-07-13 1991-07-16 Mellemprodukter til brug ved fremstilling af 3,20-dioxo-4,9-dien-21-hydroxylsteroider DK165637C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7820973A FR2430953A1 (fr) 1978-07-13 1978-07-13 Nouveaux derives 3,20-dioxo 4,9-diene 21-hydroxyle, leur procede de preparation et leur application comme medicaments
FR7820973 1978-07-13

Publications (4)

Publication Number Publication Date
DK136391A DK136391A (da) 1991-07-16
DK136391D0 DK136391D0 (da) 1991-07-16
DK165637B DK165637B (da) 1992-12-28
DK165637C true DK165637C (da) 1993-06-01

Family

ID=9210732

Family Applications (2)

Application Number Title Priority Date Filing Date
DK292579A DK163361C (da) 1978-07-13 1979-07-12 Analogifremgangsmaade til fremstilling af 3,20-dioxo-4,9-dien-21-hydroxylsteroider
DK136391A DK165637C (da) 1978-07-13 1991-07-16 Mellemprodukter til brug ved fremstilling af 3,20-dioxo-4,9-dien-21-hydroxylsteroider

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK292579A DK163361C (da) 1978-07-13 1979-07-12 Analogifremgangsmaade til fremstilling af 3,20-dioxo-4,9-dien-21-hydroxylsteroider

Country Status (15)

Country Link
US (1) US4273771A (da)
EP (2) EP0046001B1 (da)
JP (2) JPS5515475A (da)
AT (1) ATE8899T1 (da)
AU (1) AU527592B2 (da)
CA (1) CA1131215A (da)
DE (1) DE2965904D1 (da)
DK (2) DK163361C (da)
ES (1) ES482112A1 (da)
FR (1) FR2430953A1 (da)
HU (1) HU178088B (da)
IE (1) IE49457B1 (da)
IL (1) IL57691A (da)
PT (1) PT69903A (da)
ZA (1) ZA793453B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5830145A (ja) * 1981-08-17 1983-02-22 Sony Corp 半導体装置の製造方法
FR2549067B1 (fr) * 1983-06-14 1985-12-27 Roussel Uclaf Derives estradieniques radioactifs marques au tritium, leur procede de preparation et leur application pour l'etude et le dosage radio-immunologique de steroides dans les fluides biologiques
US4804541A (en) * 1987-08-11 1989-02-14 Moleculon, Inc. Transdermal administration using benzyl alcohol
US5516790A (en) * 1989-01-23 1996-05-14 Texas A&M University System Technology Licensing Office Synthesis and application of alkyl-substituted dibenzofurans as antitumorigenic agents
FR2692267B1 (fr) * 1992-06-11 1995-05-19 Roussel Uclaf Nouveau procédé de préparation de composés stéroïdes 20-céto 21alpha-hydroxy et intermédiaires.
FR2694007B1 (fr) * 1992-07-23 1994-09-30 Roussel Uclaf Nouveau procédé de préparation de composés stéroïdes 20-céto 21 (S) hydroxy et des intermédiaires.
FR2749012B1 (fr) * 1996-05-22 1998-08-07 Hoechst Marion Roussel Inc Nouveaux steroides 1 ou 6-hydroxyles, leur procede de preparation, leur application a titre de medicament et les compositions pharmaceutiques les renfermant
FR2749514B1 (fr) * 1996-06-11 1998-08-07 Hoechst Marion Roussel Systemes transdermiques renfermant 2 principes actifs dans des compartiments separes, leur procede de preparation et leur application comme medicament
FR2749586B1 (fr) * 1996-06-11 1998-08-07 Hoechst Marion Roussel Inc Nouveaux dispositifs destines a l'administration transdermique de la trimegestone, leur procede de preparation et leur application a titre de medicaments
US6451778B1 (en) 1996-07-26 2002-09-17 Wyeth Oral contraceptive
US5888543A (en) * 1996-07-26 1999-03-30 American Home Products Corporation Oral contraceptives
US5858405A (en) * 1996-07-26 1999-01-12 American Home Products Corporation Oral contraceptive
US6479475B1 (en) 1996-07-26 2002-11-12 Wyeth Oral contraceptive
US20030008870A1 (en) * 2001-02-02 2003-01-09 Joel Krasnow Method of using a cyclooxygenase-2 inhibitor and sex steroids as a combination therapy for the treatment and prevention of dysmenorrhea
TW200306846A (en) * 2002-04-03 2003-12-01 Wyeth Corp Hormone replacement therapy
ITMI20042001A1 (it) * 2004-10-21 2005-01-21 Ind Chimica Srl Processo per la preparazione di 21-idrossi steroidi con controllo della distribuzione epimerica nella posizione c-21
DE102005034498A1 (de) * 2005-07-20 2007-01-25 Grünenthal GmbH Orale Kontrazeption mit Trimegeston

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB902373A (en) * 1960-01-22 1962-08-01 Pfizer & Co C Steroids and preparation thereof
US3810885A (en) * 1967-12-12 1974-05-14 Roussel Uclaf Novel steroids and processes
FR2077877B1 (da) * 1970-02-20 1974-02-01 Roussel Uclaf
FR2149302A1 (en) * 1971-08-19 1973-03-30 Roussel Uclaf 21-methyl pregnadienes prepn - used as progestomimetics
US3923414A (en) * 1973-07-16 1975-12-02 Valeron Corp Vibration damping support
FR2385737A1 (fr) * 1977-04-01 1978-10-27 Roussel Uclaf Nouveaux steroides, leur procede de preparation et leur application dans la synthese de steroides marques au tritium
FR2374335A1 (fr) * 1976-12-14 1978-07-13 Roussel Uclaf Nouveaux steroides, leur procede de preparation et leur application dans la synthese de steroides marques au tritium
JPS5894940U (ja) * 1981-12-21 1983-06-28 日野自動車株式会社 ビスカスダンパ

Also Published As

Publication number Publication date
CA1131215A (fr) 1982-09-07
EP0046001A1 (fr) 1982-02-17
HU178088B (en) 1982-03-28
PT69903A (fr) 1979-08-01
JPS6254119B2 (da) 1987-11-13
JPH027600B2 (da) 1990-02-19
DK292579A (da) 1980-01-14
FR2430953B1 (da) 1981-09-11
DE2965904D1 (en) 1983-08-25
IL57691A0 (en) 1979-10-31
AU527592B2 (en) 1983-03-10
JPS5515475A (en) 1980-02-02
IL57691A (en) 1983-10-31
ZA793453B (en) 1980-06-25
DK163361B (da) 1992-02-24
FR2430953A1 (fr) 1980-02-08
DK136391A (da) 1991-07-16
DK163361C (da) 1992-07-13
EP0007823A3 (en) 1980-05-14
DK165637B (da) 1992-12-28
EP0007823B1 (fr) 1983-07-20
IE49457B1 (en) 1985-10-16
EP0007823A2 (fr) 1980-02-06
DK136391D0 (da) 1991-07-16
ATE8899T1 (de) 1984-08-15
JPS6333395A (ja) 1988-02-13
AU4889579A (en) 1980-01-17
US4273771A (en) 1981-06-16
EP0046001B1 (fr) 1984-08-08
ES482112A1 (es) 1980-07-01
IE791339L (en) 1980-01-13

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