ZA753968B - Novel benzimidazolinone derivatives - Google Patents

Novel benzimidazolinone derivatives

Info

Publication number
ZA753968B
ZA753968B ZA3968A ZA753968A ZA753968B ZA 753968 B ZA753968 B ZA 753968B ZA 3968 A ZA3968 A ZA 3968A ZA 753968 A ZA753968 A ZA 753968A ZA 753968 B ZA753968 B ZA 753968B
Authority
ZA
South Africa
Prior art keywords
novel
benzimidazolinone derivatives
benzimidazolinone
derivatives
novel benzimidazolinone
Prior art date
Application number
ZA3968A
Other languages
English (en)
Inventor
P Janssen
A Van Heertum
J Vandenberk
Aa M Van Der
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of ZA753968B publication Critical patent/ZA753968B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/78Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56Nitrogen atoms
    • C07D211/58Nitrogen atoms attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N21/00Investigating or analysing materials by the use of optical means, i.e. using sub-millimetre waves, infrared, visible or ultraviolet light
    • G01N21/75Systems in which material is subjected to a chemical reaction, the progress or the result of the reaction being investigated
    • G01N21/76Chemiluminescence; Bioluminescence
    • G01N21/766Chemiluminescence; Bioluminescence of gases
    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N31/00Investigating or analysing non-biological materials by the use of the chemical methods specified in the subgroup; Apparatus specially adapted for such methods
    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N31/00Investigating or analysing non-biological materials by the use of the chemical methods specified in the subgroup; Apparatus specially adapted for such methods
    • G01N31/10Investigating or analysing non-biological materials by the use of the chemical methods specified in the subgroup; Apparatus specially adapted for such methods using catalysis
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10TTECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T436/00Chemistry: analytical and immunological testing
    • Y10T436/17Nitrogen containing
    • Y10T436/173845Amine and quaternary ammonium
    • Y10T436/175383Ammonia
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10TTECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T436/00Chemistry: analytical and immunological testing
    • Y10T436/17Nitrogen containing
    • Y10T436/177692Oxides of nitrogen
    • Y10T436/178459Only nitrogen dioxide
ZA3968A 1974-06-21 1975-06-20 Novel benzimidazolinone derivatives ZA753968B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/481,594 US3989707A (en) 1974-06-21 1974-06-21 Benzimidazolinone derivatives

Publications (1)

Publication Number Publication Date
ZA753968B true ZA753968B (en) 1977-01-26

Family

ID=23912586

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA3968A ZA753968B (en) 1974-06-21 1975-06-20 Novel benzimidazolinone derivatives

Country Status (25)

Country Link
US (1) US3989707A (xx)
JP (1) JPS5840553B2 (xx)
AT (1) AT345833B (xx)
AU (1) AU500910B2 (xx)
BE (1) BE830403A (xx)
CA (1) CA1053235A (xx)
CH (1) CH615173A5 (xx)
CS (1) CS190480B2 (xx)
DE (1) DE2527261C2 (xx)
DK (1) DK141751B (xx)
ES (1) ES438714A1 (xx)
FI (1) FI59589C (xx)
FR (1) FR2275210A1 (xx)
GB (1) GB1505173A (xx)
HU (1) HU170435B (xx)
IE (1) IE41383B1 (xx)
IL (1) IL47529A (xx)
NL (1) NL180587C (xx)
NO (1) NO142400C (xx)
PH (1) PH13604A (xx)
PL (1) PL98220B1 (xx)
SE (2) SE416298B (xx)
SU (1) SU585811A3 (xx)
YU (1) YU159475A (xx)
ZA (1) ZA753968B (xx)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4066772A (en) * 1975-07-21 1978-01-03 Janssen Pharmaceutica N.V. 1,3-Dihydro-1-[3-(1-piperidinyl)propyl]-2H-benzimidazol-2-ones and related compounds
NZ181256A (en) * 1975-07-21 1978-04-28 Janssen Pharmaceutica Nv 1-(w-benzazol-11-ylalkyl)-piperidine derivatives and pharmaceutical compositions containing certain of these derivatives
US4076821A (en) * 1976-02-27 1978-02-28 Yoshitomi Pharmaceutical Industries, Ltd. 4,4-Diphenylcycloalkylpiperidines and psychotropic compositions thereof
US4219559A (en) * 1979-01-10 1980-08-26 Janssen Pharmaceutica N.V. N-Heterocyclyl-4-piperidinamines
MA19091A1 (fr) * 1980-03-10 1981-10-01 Janssen Pharmaceutica Nv Nouveaux derives de i-(4-aryl-cyclohexyl)piperidine .
US4777265A (en) * 1986-03-11 1988-10-11 Basf Aktiengesellschaft Preparation of acrylates and methacrylates
DE4107857A1 (de) * 1991-03-12 1992-09-17 Thomae Gmbh Dr K Cyclische harnstoffderivate, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung
ATE341542T1 (de) 1996-04-19 2006-10-15 Neurosearch As 1-(4-piperidyl)-benzimidazole mit neurotropher aktivität
ES2226129T3 (es) * 1997-05-30 2005-03-16 Banyu Pharmaceutical Co., Ltd. Derivados de 2-0x0imidazol.
AU1185300A (en) * 1998-11-20 2000-06-13 Banyu Pharmaceutical Co., Ltd. 2-oxoimidazole derivatives
KR20020020788A (ko) * 1999-07-21 2002-03-15 후지야마 아키라 벤즈이미다졸론 유도체 및 포스포디에스테라제억제제로서의 이의 용도
CA2465328C (en) * 2001-11-01 2011-06-14 Michael Francis Gross Piperidines
US8288412B2 (en) * 2005-09-30 2012-10-16 Glaxo Group Limited Compounds which have activity at M1 receptor and their uses in medicine
US8288413B2 (en) * 2005-09-30 2012-10-16 Glaxo Group Limited Benzimidazolones which have activity at M1 receptor
MY148504A (en) * 2005-09-30 2013-04-30 Glaxo Group Ltd Compounds which have activity at m? receptor and their uses in medicine
GB0605784D0 (en) * 2006-03-22 2006-05-03 Glaxo Group Ltd Compounds
EP1997381A1 (en) * 2007-06-01 2008-12-03 Commissariat à l'Energie Atomique Use of a compound having a monogalactosyldiacylglycerol synthase inhibitory activity as herbicide or algaecide, herbicide and algaecide compositions
GB0718415D0 (en) * 2007-09-20 2007-10-31 Glaxo Group Ltd Compounds
JP2013501804A (ja) * 2009-08-12 2013-01-17 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ カテプシンs阻害剤の調製プロセス
AU2022287810A1 (en) * 2021-06-07 2024-01-18 Fuso Pharmaceutical Industries, Ltd. T-type calcium channel blocker

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE633495A (xx) * 1962-06-13
US3161645A (en) * 1962-12-18 1964-12-15 Res Lab Dr C Janssen N V 1-(1-aroylpropyl-4-piperidyl)-2-benzimidazolinones and related compounds
BE659364A (xx) * 1964-02-05
US3799932A (en) * 1970-03-20 1974-03-26 Sumitomo Chemical Co Gamma-piperidinobutyrophenones
JPS5511671B2 (xx) * 1971-08-26 1980-03-26

Also Published As

Publication number Publication date
CS190480B2 (en) 1979-05-31
DK141751C (xx) 1980-11-03
US3989707A (en) 1976-11-02
PL98220B1 (pl) 1978-04-29
SE7507026L (sv) 1975-12-22
IE41383B1 (en) 1979-12-19
NO142400B (no) 1980-05-05
YU159475A (en) 1982-02-28
IE41383L (en) 1975-12-21
ES438714A1 (es) 1977-07-01
FI59589C (fi) 1981-09-10
CA1053235A (en) 1979-04-24
DE2527261A1 (de) 1976-01-08
FI751462A (xx) 1975-12-22
GB1505173A (en) 1978-03-30
SU585811A3 (ru) 1977-12-25
JPS5840553B2 (ja) 1983-09-06
AT345833B (de) 1978-10-10
CH615173A5 (xx) 1980-01-15
FR2275210A1 (fr) 1976-01-16
BE830403A (nl) 1975-12-19
SE7601636L (sv) 1976-02-13
NL180587C (nl) 1987-03-16
AU8113875A (en) 1976-11-18
DE2527261C2 (de) 1986-09-04
FR2275210B1 (xx) 1978-12-22
JPS5113780A (xx) 1976-02-03
PH13604A (en) 1980-08-05
IL47529A (en) 1978-10-31
NL180587B (nl) 1986-10-16
NO142400C (no) 1980-08-13
FI59589B (fi) 1981-05-29
ATA476175A (de) 1978-02-15
AU500910B2 (en) 1979-06-07
NO751735L (xx) 1975-12-23
NL7507368A (nl) 1975-12-23
SE416298B (sv) 1980-12-15
IL47529A0 (en) 1975-08-31
HU170435B (xx) 1977-06-28
DK281975A (xx) 1975-12-22
SE415298B (sv) 1980-09-22
DK141751B (da) 1980-06-09

Similar Documents

Publication Publication Date Title
PH11652A (en) Arloxphenylpropylamines derivatives
IL48592A0 (en) Novel 1-substituted-4-benzylpiperidine derivatives
IL48593A0 (en) Novel 1-substituted-4-benzylidenepiperidine derivatives
ZA753968B (en) Novel benzimidazolinone derivatives
IL46341A (en) -aryl-4-substituted piperidino-alkanol derivatives
GB1519811A (en) Thienothaiazine derivatives
PH12312A (en) Thienothiazine derivatives
ZA757828B (en) 2-methoxy-benzamide derivatives
AU1038176A (en) 4-arylpiperidine derivatives
PH13481A (en) Rifanycin derivative
ZA753496B (en) Novel n-cycloalkylmethyl decahydroisoquinolines
GB1484049A (en) 3-alkoxy-pyrazine-2-carboxamide derivatives
AU7921975A (en) Hexahydro-alpha-carboline derivatives
GB1521320A (en) Quinolisidine derivatives
ZA753315B (en) Oxacyclohexane derivatives
ZA754602B (en) Antiboiotic a2041 derivative
ZA751899B (en) Benzo-bicyclononene derivatives
US3992538A (en) Substituted o-acyl-acrylaldoximes
ZA755543B (en) Thiomethylcephem derivatives
ZA756893B (en) Phenyl-pyridylamine derivatives
ZA753299B (en) Amidino-hydrazone derivatives
AU8332175A (en) New hydroxyphenyl-butazone derivatives
GB1486646A (en) Thieno-pyridine derivatives
JPS51115457A (en) 166methyll9 alphaa halosteroid derivatives
ZA756964B (en) Novel benzylpyrimidines