ZA201407406B - Dosage regimen for a pi-3 kinase inhibitor - Google Patents

Dosage regimen for a pi-3 kinase inhibitor

Info

Publication number
ZA201407406B
ZA201407406B ZA2014/07406A ZA201407406A ZA201407406B ZA 201407406 B ZA201407406 B ZA 201407406B ZA 2014/07406 A ZA2014/07406 A ZA 2014/07406A ZA 201407406 A ZA201407406 A ZA 201407406A ZA 201407406 B ZA201407406 B ZA 201407406B
Authority
ZA
South Africa
Prior art keywords
kinase inhibitor
dosage regimen
regimen
dosage
kinase
Prior art date
Application number
ZA2014/07406A
Other languages
English (en)
Inventor
Cristian Massacesi
Samit Hiwart
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48626588&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA201407406(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of ZA201407406B publication Critical patent/ZA201407406B/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ZA2014/07406A 2012-05-16 2014-10-13 Dosage regimen for a pi-3 kinase inhibitor ZA201407406B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261647654P 2012-05-16 2012-05-16
PCT/US2013/040877 WO2013173283A1 (en) 2012-05-16 2013-05-14 Dosage regimen for a pi-3 kinase inhibitor

Publications (1)

Publication Number Publication Date
ZA201407406B true ZA201407406B (en) 2015-11-25

Family

ID=48626588

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA2014/07406A ZA201407406B (en) 2012-05-16 2014-10-13 Dosage regimen for a pi-3 kinase inhibitor

Country Status (19)

Country Link
US (2) US10213432B2 (cg-RX-API-DMAC10.html)
EP (1) EP2849756A1 (cg-RX-API-DMAC10.html)
JP (2) JP6381523B2 (cg-RX-API-DMAC10.html)
KR (1) KR20150009540A (cg-RX-API-DMAC10.html)
CN (1) CN104349779A (cg-RX-API-DMAC10.html)
AU (1) AU2013263043B2 (cg-RX-API-DMAC10.html)
BR (1) BR112014028420A2 (cg-RX-API-DMAC10.html)
CA (1) CA2872526A1 (cg-RX-API-DMAC10.html)
CL (1) CL2014003101A1 (cg-RX-API-DMAC10.html)
HK (1) HK1202435A1 (cg-RX-API-DMAC10.html)
IL (1) IL235567B (cg-RX-API-DMAC10.html)
MX (1) MX360892B (cg-RX-API-DMAC10.html)
NZ (1) NZ700924A (cg-RX-API-DMAC10.html)
PH (1) PH12014502547A1 (cg-RX-API-DMAC10.html)
RU (1) RU2630975C2 (cg-RX-API-DMAC10.html)
SG (2) SG11201406550QA (cg-RX-API-DMAC10.html)
TN (1) TN2014000433A1 (cg-RX-API-DMAC10.html)
WO (1) WO2013173283A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA201407406B (cg-RX-API-DMAC10.html)

Families Citing this family (9)

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MX342326B (es) 2011-09-27 2016-09-26 Novartis Ag 3-pirimidin-4-il-oxazolidin-2-onas como inhibidoras de idh mutante.
UY34632A (es) 2012-02-24 2013-05-31 Novartis Ag Compuestos de oxazolidin- 2- ona y usos de los mismos
US9296733B2 (en) 2012-11-12 2016-03-29 Novartis Ag Oxazolidin-2-one-pyrimidine derivative and use thereof for the treatment of conditions, diseases and disorders dependent upon PI3 kinases
CA2903979A1 (en) 2013-03-14 2014-09-18 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant idh
DK3076969T3 (da) * 2013-12-06 2021-11-22 Novartis Ag Doseringsregime for en alfa-isoform-selektiv phosphatidylinositol-3-kinase-hæmmer
WO2016109426A1 (en) * 2014-12-29 2016-07-07 Verastem, Inc. Oral dosing regimen of a dual mtor and pi3 inhibitor
WO2017009751A1 (en) 2015-07-15 2017-01-19 Pfizer Inc. Pyrimidine derivatives
CN108472289A (zh) * 2015-11-02 2018-08-31 诺华股份有限公司 磷脂酰肌醇3-激酶抑制剂的给药方案
WO2018009895A1 (en) * 2016-07-08 2018-01-11 Autotelic Llc Methods for trabedersen dosing by auc

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Also Published As

Publication number Publication date
RU2014150860A (ru) 2016-07-10
CN104349779A (zh) 2015-02-11
JP2018108998A (ja) 2018-07-12
NZ700924A (en) 2016-02-26
JP6381523B2 (ja) 2018-08-29
CL2014003101A1 (es) 2015-02-27
SG10201608469RA (en) 2016-11-29
IL235567A0 (en) 2015-01-29
MX2014013904A (es) 2015-01-16
KR20150009540A (ko) 2015-01-26
PH12014502547A1 (en) 2015-01-21
RU2630975C2 (ru) 2017-09-15
SG11201406550QA (en) 2014-11-27
TN2014000433A1 (en) 2016-03-30
BR112014028420A2 (pt) 2017-09-19
JP2015517523A (ja) 2015-06-22
HK1202435A1 (en) 2015-10-02
IL235567B (en) 2019-08-29
MX360892B (es) 2018-11-20
AU2013263043B2 (en) 2016-06-16
WO2013173283A1 (en) 2013-11-21
US20150141426A1 (en) 2015-05-21
CA2872526A1 (en) 2013-11-21
US20190134052A1 (en) 2019-05-09
US10213432B2 (en) 2019-02-26
AU2013263043A1 (en) 2014-10-30
EP2849756A1 (en) 2015-03-25

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