ZA201200819B - N1-acyl-5-fluoropyrimidinone derivatives - Google Patents

N1-acyl-5-fluoropyrimidinone derivatives

Info

Publication number
ZA201200819B
ZA201200819B ZA2012/00819A ZA201200819A ZA201200819B ZA 201200819 B ZA201200819 B ZA 201200819B ZA 2012/00819 A ZA2012/00819 A ZA 2012/00819A ZA 201200819 A ZA201200819 A ZA 201200819A ZA 201200819 B ZA201200819 B ZA 201200819B
Authority
ZA
South Africa
Prior art keywords
acyl
fluoropyrimidinone
derivatives
fluoropyrimidinone derivatives
Prior art date
Application number
ZA2012/00819A
Other languages
English (en)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA201200819(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of ZA201200819B publication Critical patent/ZA201200819B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA2012/00819A 2009-08-07 2012-02-02 N1-acyl-5-fluoropyrimidinone derivatives ZA201200819B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
ZA201200819B true ZA201200819B (en) 2013-05-29

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA2012/00819A ZA201200819B (en) 2009-08-07 2012-02-02 N1-acyl-5-fluoropyrimidinone derivatives

Country Status (33)

Country Link
US (1) US8470839B2 (https=)
EP (1) EP2519512B1 (https=)
JP (1) JP5748754B2 (https=)
KR (1) KR101792285B1 (https=)
CN (1) CN102548981B (https=)
AU (1) AU2010279402B2 (https=)
BR (1) BR112012002810B1 (https=)
CA (1) CA2768510C (https=)
CL (1) CL2012000316A1 (https=)
CO (1) CO6491117A2 (https=)
CR (1) CR20120030A (https=)
CY (1) CY1122115T1 (https=)
DK (1) DK2519512T3 (https=)
EA (1) EA023411B1 (https=)
EC (1) ECSP12011653A (https=)
ES (1) ES2728966T3 (https=)
HN (1) HN2012000269A (https=)
HR (1) HRP20190919T1 (https=)
HU (1) HUE045290T2 (https=)
IL (1) IL217952A (https=)
IN (1) IN2012DN00539A (https=)
LT (1) LT2519512T (https=)
MX (1) MX2012001620A (https=)
NI (1) NI201200022A (https=)
NZ (1) NZ597570A (https=)
PE (1) PE20120688A1 (https=)
PL (1) PL2519512T3 (https=)
PT (1) PT2519512T (https=)
SI (1) SI2519512T1 (https=)
TR (1) TR201908180T4 (https=)
UA (1) UA106889C2 (https=)
WO (1) WO2011017538A1 (https=)
ZA (1) ZA201200819B (https=)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2471371T3 (es) * 2009-08-07 2014-06-26 Dow Agrosciences Llc Derivados de N1-sulfonil-5-fluoropirimidinona
WO2013025795A1 (en) * 2011-08-17 2013-02-21 Dow Agrosciences Llc 5-fluoro-4-imino-3-(substituted)-3,4-dihydropyrimidin-2-(1h)-one derivatives
RU2638556C2 (ru) 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата
CA2894510A1 (en) 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2h)-carboxamide derivatives
MX2015008443A (es) * 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de 1-(benzoilo-sustituido) -5-fluoro-4-imino-3-metil-3, 4-dihidropirimidin-2 (1h)-ona.
AU2013370494B2 (en) * 2012-12-31 2017-08-17 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
NZ722419A (en) 2013-12-31 2018-01-26 Adama Makhteshim Ltd Synergistic fungicidal mixtures and compositions for fungal control
CA2935594C (en) 2013-12-31 2022-05-03 Nakyen Choy 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
CN107001397B (zh) 2014-09-26 2020-10-13 科慕埃弗西有限公司 异氰酸酯衍生的有机硅烷
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
EP3876717A1 (en) 2018-11-05 2021-09-15 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
PY2057637A (es) 2019-09-23 2021-10-05 Adama Makhteshim Ltd Proceso para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto

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Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (https=) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
EP0332579B1 (de) 1988-03-09 1994-08-10 Ciba-Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
BR9609613A (pt) * 1995-07-05 1999-05-25 Du Pont Composto composição fungicida e método de controle de doenças de plantas
ATE216999T1 (de) 1996-03-11 2002-05-15 Syngenta Participations Ag Pyrimidin-4-on derivate als pestizidesmittel
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
US20080269238A1 (en) * 2004-04-01 2008-10-30 Takeda Pharmaceutical Company Limited Thiazolopyrimidine Derivative
WO2008005303A2 (en) * 2006-06-30 2008-01-10 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
PT2562166E (pt) * 2008-01-22 2015-10-28 Dow Agrosciences Llc Derivados de 5-fluoro-pirimidina como fungicidas
CN102215691B (zh) 2008-08-01 2015-02-04 陶氏益农公司 5-氟胞嘧啶作为杀真菌剂的用途
WO2010085377A2 (en) 2009-01-23 2010-07-29 Crystal Biopharmaceutical Llc Hydroxamic acid derivatives
ES2471371T3 (es) * 2009-08-07 2014-06-26 Dow Agrosciences Llc Derivados de N1-sulfonil-5-fluoropirimidinona

Also Published As

Publication number Publication date
JP2013501723A (ja) 2013-01-17
US20110034490A1 (en) 2011-02-10
EA201270253A1 (ru) 2012-07-30
US8470839B2 (en) 2013-06-25
NZ597570A (en) 2014-04-30
PE20120688A1 (es) 2012-06-06
EP2519512A4 (en) 2013-01-16
TR201908180T4 (tr) 2019-06-21
CA2768510A1 (en) 2011-02-10
LT2519512T (lt) 2019-07-25
HN2012000269A (es) 2015-04-27
KR101792285B1 (ko) 2017-10-31
BR112012002810A2 (pt) 2015-09-15
DK2519512T3 (da) 2019-05-27
CR20120030A (es) 2012-03-28
HK1172894A1 (en) 2013-05-03
WO2011017538A1 (en) 2011-02-10
EA023411B1 (ru) 2016-06-30
MX2012001620A (es) 2012-04-11
NI201200022A (es) 2012-05-22
CN102548981B (zh) 2015-05-13
PL2519512T3 (pl) 2019-09-30
BR112012002810B1 (pt) 2018-12-11
IL217952A0 (en) 2012-03-29
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
CY1122115T1 (el) 2020-11-25
CN102548981A (zh) 2012-07-04
IN2012DN00539A (https=) 2015-06-12
CL2012000316A1 (es) 2014-06-27
CA2768510C (en) 2018-05-15
EP2519512B1 (en) 2019-03-20
EP2519512A1 (en) 2012-11-07
KR20120041786A (ko) 2012-05-02
UA106889C2 (uk) 2014-10-27
AU2010279402B2 (en) 2015-04-16
CO6491117A2 (es) 2012-07-31
HRP20190919T1 (hr) 2019-09-20
AU2010279402A1 (en) 2012-02-02
PT2519512T (pt) 2019-06-04
SI2519512T1 (sl) 2019-09-30
ES2728966T3 (es) 2019-10-29
JP5748754B2 (ja) 2015-07-15
IL217952A (en) 2017-11-30

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