ZA201103978B - Novel antimicrobials - Google Patents
Novel antimicrobialsInfo
- Publication number
- ZA201103978B ZA201103978B ZA2011/03978A ZA201103978A ZA201103978B ZA 201103978 B ZA201103978 B ZA 201103978B ZA 2011/03978 A ZA2011/03978 A ZA 2011/03978A ZA 201103978 A ZA201103978 A ZA 201103978A ZA 201103978 B ZA201103978 B ZA 201103978B
- Authority
- ZA
- South Africa
- Prior art keywords
- novel antimicrobials
- antimicrobials
- novel
- Prior art date
Links
- 239000004599 antimicrobial Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A61P31/06—Antibacterial agents for tuberculosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Virology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Communicable Diseases (AREA)
- Pulmonology (AREA)
- Molecular Biology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN2623DE2008 | 2008-11-20 | ||
| PCT/IN2009/000658 WO2010058423A2 (en) | 2008-11-20 | 2009-11-18 | Novel antimicrobials |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA201103978B true ZA201103978B (en) | 2012-09-26 |
Family
ID=42198604
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA2011/03978A ZA201103978B (en) | 2008-11-20 | 2011-05-30 | Novel antimicrobials |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US8841306B2 (OSRAM) |
| EP (1) | EP2367820B1 (OSRAM) |
| JP (1) | JP5662940B2 (OSRAM) |
| KR (1) | KR20110092309A (OSRAM) |
| CN (1) | CN102224151A (OSRAM) |
| AR (1) | AR074387A1 (OSRAM) |
| AU (1) | AU2009318783A1 (OSRAM) |
| CA (1) | CA2743971A1 (OSRAM) |
| MX (1) | MX2011005365A (OSRAM) |
| RU (1) | RU2522582C2 (OSRAM) |
| WO (1) | WO2010058423A2 (OSRAM) |
| ZA (1) | ZA201103978B (OSRAM) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5855668B2 (ja) * | 2010-10-13 | 2016-02-09 | グラクソ グループ リミテッドＧｌａｘｏ Ｇｒｏｕｐ Ｌｉｍｉｔｅｄ | 結核に対して有用な３−アミノ−ピラゾール誘導体 |
| PT106651A (pt) * | 2012-11-20 | 2014-05-20 | Tecnimede Sociedade Tecnico Medicinal S A | Quinolil hidrazonas para o tratamento de tuberculose e doenças relacionadas |
| CN103450173B (zh) * | 2013-09-07 | 2015-06-03 | 吉首大学 | 吡咯酮-苯基-噁唑烷酮型化合物及其制法和用途 |
| WO2017156519A1 (en) * | 2016-03-11 | 2017-09-14 | The Board Of Trustees Of The University Of Illinois | Small-molecules active against gram-negative bacteria |
| WO2018237140A1 (en) | 2017-06-23 | 2018-12-27 | The Board Of Trustees Of The University Of Illinois | Topoisomerase inhibitors with antibacterial and antcancer activity |
| AU2021217225A1 (en) * | 2020-02-07 | 2022-10-06 | University Of South Florida | Inhibition of beta-arrestin oligomerization in tauopathy |
Family Cites Families (53)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100257418B1 (ko) | 1991-11-01 | 2000-05-15 | 로렌스 티. 마이젠헬더 | 치환된 아릴-및 헤테로아릴-페닐옥사졸리디논 |
| SK283420B6 (sk) | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
| EP0718293B1 (en) | 1993-09-06 | 2002-03-13 | Fujisawa Pharmaceutical Co., Ltd. | Cyclodepsipeptide compound |
| CA2218088A1 (en) | 1995-05-11 | 1996-11-14 | Pharmacia & Upjohn Company | Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones |
| CA2228647A1 (en) | 1995-09-01 | 1997-03-13 | Pharmacia & Upjohn Company | Phenyloxazolidinones having a c-c bond to 4-8 membered heterocyclic rings |
| GB9702213D0 (en) * | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
| IL140084A0 (en) * | 1998-06-05 | 2002-02-10 | Astra Ab | Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them |
| JP2000204084A (ja) * | 1998-11-11 | 2000-07-25 | Hokuriku Seiyaku Co Ltd | チオカルバミド酸誘導体 |
| AU1379900A (en) | 1998-11-17 | 2000-06-05 | Bayer Aktiengesellschaft | Novel substituted phenyloxazolidone derivatives |
| HK1046680B (zh) | 1999-05-27 | 2004-12-31 | 法玛西雅厄普约翰美国公司 | 作为抗菌剂的新的双环恶唑烷酮 |
| US6608081B2 (en) | 1999-08-12 | 2003-08-19 | Ortho-Mcneil Pharmaceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| BR0111280A (pt) | 2000-06-05 | 2003-06-10 | Dong A Pharm Co Ltd | Novos derivados de oxazolidinona e um processo para a preparação dos mesmos |
| ATE301474T1 (de) | 2000-06-30 | 2005-08-15 | Pharmacia & Upjohn Co Llc | Zusammensetzungen zur behandlung baktrieller infektionen, welche ein oxazolidinonderivat, sulbactam und ampicillin enthalten |
| DOP2002000333A (es) | 2001-02-14 | 2002-09-30 | Warner Lambert Co | Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz |
| ES2268011T3 (es) | 2001-04-07 | 2007-03-16 | Astrazeneca Ab | Oxazolidinonas que contienen un grupo sulfonimida como antibioticos. |
| GB0108793D0 (en) | 2001-04-07 | 2001-05-30 | Astrazeneca Ab | Chemical compounds |
| WO2003006447A2 (en) | 2001-07-09 | 2003-01-23 | Pharmacia Italia Spa | Interaction inhibitors of tcf-4 with beta-catenin |
| EP1409464A4 (en) | 2001-07-16 | 2005-11-02 | Ranbaxy Lab Ltd | OXAZOLIDINONE DERIVATIVES AS POTENTIAL ANTIMICROBIALS |
| AR038536A1 (es) | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
| BR0310074A (pt) | 2002-05-15 | 2005-03-08 | Ranbaxy Lab Ltd | Formas polimórficas de derivados de fenil oxazolidinona |
| WO2003097640A1 (en) | 2002-05-22 | 2003-11-27 | Orchid Chemicals & Pharmaceuticals Ltd. | Oxazolidinone derivatives as antibacterial agents |
| WO2004009587A1 (en) | 2002-07-22 | 2004-01-29 | Orchid Chemicals & Pharmaceuticals Ltd | Oxazolidinone derivatives as antibacterial agents |
| EA200500283A1 (ru) | 2002-07-29 | 2005-08-25 | Рэнбакси Лабораториз Лимитед | Производные оксазолидинона как противомикробные средства |
| AU2003253141A1 (en) * | 2002-08-22 | 2004-03-11 | Orchid Chemicals And Pharmaceuticals Ltd | Novel antibacterial agents |
| US6875784B2 (en) | 2002-10-09 | 2005-04-05 | Pharmacia & Upjohn Company | Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives |
| DE60309504T2 (de) | 2002-11-21 | 2007-05-16 | Pharmacia & Upjohn Co. Llc, Kalamazoo | N-(4-(piperazin-1-yl)-phenyl-2-oxazolidinon-5-carbosäureamid-derivate und verwandte verbindungen als antibakterielle mittel |
| GB0229526D0 (en) | 2002-12-19 | 2003-01-22 | Astrazeneca Ab | Chemical compounds |
| GB0229518D0 (en) | 2002-12-19 | 2003-01-22 | Astrazeneca Ab | Chemical compounds |
| CN1237056C (zh) | 2002-12-25 | 2006-01-18 | 中国科学院上海药物研究所 | 噁唑烷酮类化合物、其制备方法和用途 |
| AU2003215861A1 (en) * | 2003-04-07 | 2004-11-01 | Ranbaxy Laboratories Limited | Oxazolidinone derivatives as antimicrobials |
| CA2521685A1 (en) | 2003-04-09 | 2004-10-21 | Pharmacia & Upjohn Company Llc | Antimicrobial [3.1.0] bicyclohexylphenyl-oxazolidinone derivatives and analogues |
| WO2004113329A1 (en) | 2003-06-20 | 2004-12-29 | Orchid Chemicals And Pharmaceuticals Ltd. | Oxazole derivatives as antibacterial agents |
| WO2005003087A2 (en) | 2003-07-01 | 2005-01-13 | Orchid Chemicals And Pharmaceuticals Ltd. | Oxazole derivatives as antibacterial agents |
| US20070293493A1 (en) | 2003-07-02 | 2007-12-20 | Milton Hammond | Oxazolidinone antibiotics and derivatives thereof |
| EP1656357A1 (en) | 2003-07-02 | 2006-05-17 | Merck & Co., Inc. | Oxazolidinone antibiotics and derivatives thereof |
| WO2005036169A2 (en) * | 2003-10-03 | 2005-04-21 | Cumbre Inc. | Fluorescent probes for ribosomes and method of use |
| KR100854211B1 (ko) | 2003-12-18 | 2008-08-26 | 동아제약주식회사 | 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물 |
| WO2005082897A1 (en) | 2004-01-28 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Oxazolidinone antibacterial agents |
| WO2005082900A2 (en) | 2004-01-28 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Oxazolidinone amidoximes as antibacterial agents |
| US20080064689A1 (en) | 2004-05-25 | 2008-03-13 | Astrazeneca Ab | 3-[4-(6-Pyridin-3-Yl)-3-Phenyl] -5-(1H-1,2,3-Triazol-1-Ylmethyl)-1,3-Oxazolidin-2-Ones as Antibacterial Agents |
| MXPA06013540A (es) | 2004-05-25 | 2007-01-26 | Astrazeneca Ab | Derivados de 3-(4-(2 -dihidroisoxasol -3-ilpiridin-5-il) fenil)-5- triazol-1- ilmetiloxazolidin -2-ona como inhibidores de mao para el tratamiento de infecciones bacterianas. |
| WO2006035283A1 (en) | 2004-09-27 | 2006-04-06 | Ranbaxy Laboratories Limited | Oxazolidinone derivatives as antimicrobials |
| WO2006043121A1 (en) | 2004-10-20 | 2006-04-27 | Ranbaxy Laboratories Limited | Oxazolidinone derivatives as antimicrobials |
| WO2006109056A1 (en) | 2005-04-12 | 2006-10-19 | Vicore Pharma Ab | New tricyclic angiotensin ii agonists |
| EP1745784A1 (en) | 2005-06-27 | 2007-01-24 | Ferrer Internacional, S.A. | Oxazolidinone derivatives and use thereof as antibiotics |
| JP2009500389A (ja) | 2005-07-06 | 2009-01-08 | ファルマシア・アンド・アップジョン・カンパニー・エルエルシー | 抗菌剤としてのアゼチジンおよびシクロブタンを含むオキサゾリジノンカルボキサミド |
| KR20070038236A (ko) | 2005-10-05 | 2007-04-10 | 일동제약주식회사 | 신규 옥사졸리디논 포름 아미드 유도체 및 그 제조방법 |
| WO2007082910A1 (en) | 2006-01-19 | 2007-07-26 | Laboratorios Salvat, S.A. | Dicarbonylic compounds with antibacterial activity |
| EP1987025B1 (en) | 2006-02-14 | 2009-09-16 | Pfizer Products Inc. | Benzoxazinone and benzoxazepinone oxazolidinones as antibacterial agents |
| CN100406455C (zh) | 2006-02-20 | 2008-07-30 | 中国科学院上海药物研究所 | 含三氮唑基的噁唑烷酮类化合物及其制备方法和用途 |
| CN101460495B (zh) | 2006-03-31 | 2013-08-14 | 财团法人乙卯研究所 | 具有杂环的化合物 |
| EP2170874A4 (en) | 2007-06-22 | 2011-08-31 | Orchid Res Lab Ltd | NEW COMPOUNDS AND THEIR USE |
| CN101434584A (zh) | 2007-11-15 | 2009-05-20 | 中山大学 | 具有抗菌活性的手性噁唑烷酮类化合物 |
-
2009
- 2009-11-18 AU AU2009318783A patent/AU2009318783A1/en not_active Abandoned
- 2009-11-18 JP JP2011537013A patent/JP5662940B2/ja not_active Expired - Fee Related
- 2009-11-18 EP EP09827270.1A patent/EP2367820B1/en not_active Not-in-force
- 2009-11-18 KR KR1020117013609A patent/KR20110092309A/ko not_active Ceased
- 2009-11-18 RU RU2011124795/04A patent/RU2522582C2/ru not_active IP Right Cessation
- 2009-11-18 MX MX2011005365A patent/MX2011005365A/es not_active Application Discontinuation
- 2009-11-18 CN CN2009801465662A patent/CN102224151A/zh active Pending
- 2009-11-18 WO PCT/IN2009/000658 patent/WO2010058423A2/en not_active Ceased
- 2009-11-18 US US13/130,440 patent/US8841306B2/en not_active Expired - Fee Related
- 2009-11-18 CA CA2743971A patent/CA2743971A1/en not_active Abandoned
- 2009-11-20 AR ARP090104485A patent/AR074387A1/es not_active Application Discontinuation
-
2011
- 2011-05-30 ZA ZA2011/03978A patent/ZA201103978B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2743971A1 (en) | 2010-05-27 |
| MX2011005365A (es) | 2011-06-24 |
| US20110245258A1 (en) | 2011-10-06 |
| WO2010058423A2 (en) | 2010-05-27 |
| RU2011124795A (ru) | 2012-12-27 |
| AR074387A1 (es) | 2011-01-12 |
| CN102224151A (zh) | 2011-10-19 |
| EP2367820A2 (en) | 2011-09-28 |
| JP2012509313A (ja) | 2012-04-19 |
| US8841306B2 (en) | 2014-09-23 |
| KR20110092309A (ko) | 2011-08-17 |
| WO2010058423A3 (en) | 2010-12-09 |
| RU2522582C2 (ru) | 2014-07-20 |
| JP5662940B2 (ja) | 2015-02-04 |
| EP2367820A4 (en) | 2012-06-20 |
| WO2010058423A9 (en) | 2011-04-28 |
| AU2009318783A1 (en) | 2011-06-23 |
| EP2367820B1 (en) | 2016-09-21 |
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