ZA200707568B - Crystal forms of an imidazole derivative - Google Patents

Crystal forms of an imidazole derivative

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Publication number
ZA200707568B
ZA200707568B ZA200707568A ZA200707568A ZA200707568B ZA 200707568 B ZA200707568 B ZA 200707568B ZA 200707568 A ZA200707568 A ZA 200707568A ZA 200707568 A ZA200707568 A ZA 200707568A ZA 200707568 B ZA200707568 B ZA 200707568B
Authority
ZA
South Africa
Prior art keywords
crystal forms
imidazole derivative
imidazole
derivative
crystal
Prior art date
Application number
ZA200707568A
Other languages
English (en)
Inventor
Haruta Naoaki
Li Zheng Jane
Trask Andrew Vincent
Kato Tomoki
Numata Toyoharu
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of ZA200707568B publication Critical patent/ZA200707568B/xx

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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ZA200707568A 2005-03-11 2007-09-03 Crystal forms of an imidazole derivative ZA200707568B (en)

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US66059205P 2005-03-11 2005-03-11

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ZA200707568B true ZA200707568B (en) 2009-09-30

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US (1) US7960407B2 (es)
EP (1) EP1861400B1 (es)
JP (1) JP5069415B2 (es)
KR (1) KR100911073B1 (es)
CN (1) CN101137656B (es)
AR (1) AR055567A1 (es)
AT (1) ATE469150T1 (es)
AU (1) AU2006221699A1 (es)
BR (1) BRPI0608819B8 (es)
CA (1) CA2600510C (es)
DE (1) DE602006014516D1 (es)
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IL (1) IL185145A0 (es)
IN (1) IN2014DN09939A (es)
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TW (1) TW200643021A (es)
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AU2009295308A1 (en) 2008-09-25 2010-04-01 Merck Canada Inc. Beta-carboline sulphonylurea derivatives as EP4 receptor antagonists
CA2754702C (en) 2009-04-22 2016-06-07 Yukinori Take Selective ep4 antagonistic substance for treatment of cancer
JP6152643B2 (ja) * 2010-02-22 2017-06-28 株式会社ＡｓｋＡｔ Ｉｌ−２３媒介疾患を治療するためのｅｐ４受容体拮抗薬の使用
RU2451680C1 (ru) 2011-02-21 2012-05-27 Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" Клатратный комплекс циклодекстрина или арабиногалактана с 9-фенил-симм-октагидроселеноксантеном, способ его получения (варианты), фармацевтическая композиция и лекарственное средство
RU2464042C1 (ru) * 2011-03-31 2012-10-20 Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" КЛАТРАТНЫЙ КОМПЛЕКС β-ЦИКЛОДЕКСТРИНА С ПРОИЗВОДНЫМ 5-ГИДРОКСИ-4-АМИНОМЕТИЛ-1-ЦИКЛОГЕКСИЛ(ИЛИ ЦИКЛОГЕПТИЛ)-3-АЛКОКСИКАРБОНИЛИНДОЛА, СПОСОБ ЕГО ПОЛУЧЕНИЯ (ВАРИАНТЫ), ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ И ЛЕКАРСТВЕННОЕ СРЕДСТВО
MX2015013328A (es) 2013-03-19 2016-02-26 Askat Inc Uso de antagonistas del receptor de ep4 en el tratamiento de enfermedad de cartilago.
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BRPI0608819B8 (pt) 2021-05-25
US7960407B2 (en) 2011-06-14
ATE469150T1 (de) 2010-06-15
RU2357968C1 (ru) 2009-06-10
IN2014DN09939A (es) 2015-08-14
CA2600510C (en) 2010-11-02
BRPI0608819A8 (pt) 2017-10-10
WO2006095268A1 (en) 2006-09-14
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MX2007011110A (es) 2008-02-21
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AU2006221699A1 (en) 2006-09-14
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IL185145A0 (en) 2007-12-03
DE602006014516D1 (es) 2010-07-08
BRPI0608819B1 (pt) 2019-11-12
CN101137656B (zh) 2010-12-22
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US20090018158A1 (en) 2009-01-15
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