ZA200510450B - Methanesulfonic acid salt of pyrazolopyrimidine compound, crystal thereof, and process for producing the same - Google Patents

Methanesulfonic acid salt of pyrazolopyrimidine compound, crystal thereof, and process for producing the same Download PDF

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Publication number
ZA200510450B
ZA200510450B ZA200510450A ZA200510450A ZA200510450B ZA 200510450 B ZA200510450 B ZA 200510450B ZA 200510450 A ZA200510450 A ZA 200510450A ZA 200510450 A ZA200510450 A ZA 200510450A ZA 200510450 B ZA200510450 B ZA 200510450B
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ZA
South Africa
Prior art keywords
disorder
compound
chloro
methyl
cyclopenta
Prior art date
Application number
ZA200510450A
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English (en)
Inventor
Hasegawa Tomoyuki
Araki Hiroshi
Obitsu Tetsuo
Gemba Yuichi
Matsui Toskiaki
Saito Tetsuji
Okamoto Masaki
Mikami Yutaka
Original Assignee
Ono Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ono Pharmaceutical Co filed Critical Ono Pharmaceutical Co
Publication of ZA200510450B publication Critical patent/ZA200510450B/en

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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ZA200510450A 2003-06-25 2005-12-22 Methanesulfonic acid salt of pyrazolopyrimidine compound, crystal thereof, and process for producing the same ZA200510450B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2003181908 2003-06-25

Publications (1)

Publication Number Publication Date
ZA200510450B true ZA200510450B (en) 2006-12-27

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ID=33535237

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ZA200510450A ZA200510450B (en) 2003-06-25 2005-12-22 Methanesulfonic acid salt of pyrazolopyrimidine compound, crystal thereof, and process for producing the same

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Country Link
US (1) US7947697B1 (ru)
EP (1) EP1637531B1 (ru)
JP (1) JP4655276B2 (ru)
KR (1) KR101082227B1 (ru)
CN (1) CN100422186C (ru)
AT (1) ATE478873T1 (ru)
AU (1) AU2004249629B2 (ru)
BR (1) BRPI0411923A (ru)
CA (1) CA2529561C (ru)
DE (1) DE602004028820D1 (ru)
ES (1) ES2349393T3 (ru)
IL (1) IL172697A (ru)
MX (1) MXPA05013917A (ru)
NO (1) NO332186B1 (ru)
NZ (1) NZ544301A (ru)
RU (1) RU2345995C2 (ru)
TW (1) TWI356058B (ru)
WO (1) WO2004113344A1 (ru)
ZA (1) ZA200510450B (ru)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005061508A1 (ja) * 2003-12-22 2005-07-07 Ono Pharmaceutical Co., Ltd. 三環式複素環化合物およびその化合物を有効成分とする医薬
WO2005087775A1 (ja) * 2004-03-15 2005-09-22 Ono Pharmaceutical Co., Ltd. 三環式複素環化合物およびその化合物を有効成分として含有する医薬組成物
CN112225732B (zh) * 2019-07-15 2024-01-09 四川科瑞德制药股份有限公司 一种盐酸哌罗匹隆水合物晶型及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU639615B2 (en) 1990-10-09 1993-07-29 Otsuka Pharmaceutical Co., Ltd. Pyrimidine derivative, production thereof, and androgen inhibitor
CN1030768C (zh) * 1990-10-09 1996-01-24 大塚制药株式会社 嘧啶衍生物或其药用盐的制备方法
JPH05112571A (ja) * 1990-10-19 1993-05-07 Otsuka Pharmaceut Co Ltd ピリミジン誘導体
CN1169149A (zh) * 1995-09-28 1997-12-31 株式会社大制药工场 止痛组合物
WO1999064422A1 (en) 1998-06-09 1999-12-16 Neurogen Corporation Pyrido[2,3-b]indolizine derivatives and aza analogues thereof; crf1 specific ligands
DK1129091T3 (da) 1998-11-12 2002-11-04 Neurocrine Biosciences Inc Antagonister for CRF-receptorer og fremgangsmåder med relation dertil
CA2349904A1 (en) 1998-11-12 2000-05-18 Neurocrine Biosciences, Inc. Crf receptor antagonists and methods relating thereto
US6531475B1 (en) 1998-11-12 2003-03-11 Neurocrine Biosciences, Inc. CRF receptor antagonists and methods relating thereto
CN1896076A (zh) 2000-12-28 2007-01-17 小野药品工业株式会社 三杂环化合物和包括其作为活性组分的药物

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AU2004249629A1 (en) 2004-12-29
IL172697A0 (en) 2006-04-10
MXPA05013917A (es) 2006-03-09
KR101082227B1 (ko) 2011-11-09
JPWO2004113344A1 (ja) 2006-07-27
CA2529561A1 (en) 2004-12-29
US7947697B1 (en) 2011-05-24
RU2345995C2 (ru) 2009-02-10
BRPI0411923A (pt) 2006-08-15
JP4655276B2 (ja) 2011-03-23
IL172697A (en) 2013-05-30
KR20060026060A (ko) 2006-03-22
RU2006101986A (ru) 2006-07-27
NO332186B1 (no) 2012-07-23
EP1637531A1 (en) 2006-03-22
DE602004028820D1 (de) 2010-10-07
ES2349393T3 (es) 2010-12-30
CN1842530A (zh) 2006-10-04
CA2529561C (en) 2012-05-29
ATE478873T1 (de) 2010-09-15
NZ544301A (en) 2008-08-29
EP1637531A4 (en) 2008-09-03
WO2004113344A1 (ja) 2004-12-29
TWI356058B (en) 2012-01-11
TW200504064A (en) 2005-02-01
NO20056093L (no) 2006-03-24
CN100422186C (zh) 2008-10-01
EP1637531B1 (en) 2010-08-25
AU2004249629B2 (en) 2009-07-30

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