TWI356058B - Methanesulfonate salt of pyrazolo-pyrimidine compo - Google Patents

Methanesulfonate salt of pyrazolo-pyrimidine compo Download PDF

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Publication number
TWI356058B
TWI356058B TW093118239A TW93118239A TWI356058B TW I356058 B TWI356058 B TW I356058B TW 093118239 A TW093118239 A TW 093118239A TW 93118239 A TW93118239 A TW 93118239A TW I356058 B TWI356058 B TW I356058B
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TW
Taiwan
Prior art keywords
group
pentylamino
disorders
compound
dihydro
Prior art date
Application number
TW093118239A
Other languages
English (en)
Chinese (zh)
Other versions
TW200504064A (en
Inventor
Tomoyuki Hasegawa
Toshiaki Matsui
Hiroshi Araki
Tetsuji Saito
Tetsuo Obitsu
Masaki Okamoto
Yuichi Gemba
Yutaka Mikami
Original Assignee
Ono Pharmaceutical Co
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Publication date
Application filed by Ono Pharmaceutical Co filed Critical Ono Pharmaceutical Co
Publication of TW200504064A publication Critical patent/TW200504064A/zh
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Publication of TWI356058B publication Critical patent/TWI356058B/zh

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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  • Obesity (AREA)
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TW093118239A 2003-06-25 2004-06-24 Methanesulfonate salt of pyrazolo-pyrimidine compo TWI356058B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2003181908 2003-06-25

Publications (2)

Publication Number Publication Date
TW200504064A TW200504064A (en) 2005-02-01
TWI356058B true TWI356058B (en) 2012-01-11

Family

ID=33535237

Family Applications (1)

Application Number Title Priority Date Filing Date
TW093118239A TWI356058B (en) 2003-06-25 2004-06-24 Methanesulfonate salt of pyrazolo-pyrimidine compo

Country Status (19)

Country Link
US (1) US7947697B1 (ru)
EP (1) EP1637531B1 (ru)
JP (1) JP4655276B2 (ru)
KR (1) KR101082227B1 (ru)
CN (1) CN100422186C (ru)
AT (1) ATE478873T1 (ru)
AU (1) AU2004249629B2 (ru)
BR (1) BRPI0411923A (ru)
CA (1) CA2529561C (ru)
DE (1) DE602004028820D1 (ru)
ES (1) ES2349393T3 (ru)
IL (1) IL172697A (ru)
MX (1) MXPA05013917A (ru)
NO (1) NO332186B1 (ru)
NZ (1) NZ544301A (ru)
RU (1) RU2345995C2 (ru)
TW (1) TWI356058B (ru)
WO (1) WO2004113344A1 (ru)
ZA (1) ZA200510450B (ru)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPWO2005061508A1 (ja) * 2003-12-22 2007-07-12 小野薬品工業株式会社 三環式複素環化合物およびその化合物を有効成分とする医薬
WO2005087775A1 (ja) * 2004-03-15 2005-09-22 Ono Pharmaceutical Co., Ltd. 三環式複素環化合物およびその化合物を有効成分として含有する医薬組成物
CN112225732B (zh) * 2019-07-15 2024-01-09 四川科瑞德制药股份有限公司 一种盐酸哌罗匹隆水合物晶型及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1030768C (zh) * 1990-10-09 1996-01-24 大塚制药株式会社 嘧啶衍生物或其药用盐的制备方法
US5420128A (en) 1990-10-09 1995-05-30 Otsuka Pharmaceutical Co., Ltd. Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor
JPH05112571A (ja) 1990-10-19 1993-05-07 Otsuka Pharmaceut Co Ltd ピリミジン誘導体
EP0795555A4 (en) 1995-09-28 1998-01-07 Otsuka Pharma Co Ltd ANALGETICS
WO1999064422A1 (en) 1998-06-09 1999-12-16 Neurogen Corporation Pyrido[2,3-b]indolizine derivatives and aza analogues thereof; crf1 specific ligands
US6531475B1 (en) 1998-11-12 2003-03-11 Neurocrine Biosciences, Inc. CRF receptor antagonists and methods relating thereto
WO2000027850A2 (en) 1998-11-12 2000-05-18 Neurocrine Biosciences, Inc. Crf receptor antagonists and methods relating thereto
PT1129091E (pt) 1998-11-12 2003-02-28 Neurocrine Biosciences Inc Antagonistas de receptor de crf e metodos relacionados
CA2432148C (en) 2000-12-28 2011-01-18 Ono Pharmaceutical Co., Ltd. Tri-heterocyclic compounds and a pharmaceutical comprising them as an active ingredient

Also Published As

Publication number Publication date
NZ544301A (en) 2008-08-29
KR20060026060A (ko) 2006-03-22
KR101082227B1 (ko) 2011-11-09
RU2006101986A (ru) 2006-07-27
ATE478873T1 (de) 2010-09-15
NO20056093L (no) 2006-03-24
CA2529561A1 (en) 2004-12-29
MXPA05013917A (es) 2006-03-09
ES2349393T3 (es) 2010-12-30
IL172697A (en) 2013-05-30
CN1842530A (zh) 2006-10-04
WO2004113344A1 (ja) 2004-12-29
US7947697B1 (en) 2011-05-24
CN100422186C (zh) 2008-10-01
NO332186B1 (no) 2012-07-23
EP1637531A1 (en) 2006-03-22
JPWO2004113344A1 (ja) 2006-07-27
ZA200510450B (en) 2006-12-27
CA2529561C (en) 2012-05-29
AU2004249629B2 (en) 2009-07-30
EP1637531A4 (en) 2008-09-03
RU2345995C2 (ru) 2009-02-10
EP1637531B1 (en) 2010-08-25
TW200504064A (en) 2005-02-01
IL172697A0 (en) 2006-04-10
JP4655276B2 (ja) 2011-03-23
AU2004249629A1 (en) 2004-12-29
BRPI0411923A (pt) 2006-08-15
DE602004028820D1 (de) 2010-10-07

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