NO332186B1 - Metansulfonsyresalt av pyrazolpyrimidinforbindelse, krystall derav, fremgangsmate for fremstilling av det samme, farmasoytisk preparat samt anvendelse derav - Google Patents
Metansulfonsyresalt av pyrazolpyrimidinforbindelse, krystall derav, fremgangsmate for fremstilling av det samme, farmasoytisk preparat samt anvendelse derav Download PDFInfo
- Publication number
- NO332186B1 NO332186B1 NO20056093A NO20056093A NO332186B1 NO 332186 B1 NO332186 B1 NO 332186B1 NO 20056093 A NO20056093 A NO 20056093A NO 20056093 A NO20056093 A NO 20056093A NO 332186 B1 NO332186 B1 NO 332186B1
- Authority
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- Norway
- Prior art keywords
- crystal
- chloro
- disorder
- methoxyphenyl
- methyl
- Prior art date
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- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
- A61P5/16—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4 for decreasing, blocking or antagonising the activity of the thyroid hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Pulmonology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Rheumatology (AREA)
- Hospice & Palliative Care (AREA)
- Dermatology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Addiction (AREA)
- Psychology (AREA)
- Otolaryngology (AREA)
- Emergency Medicine (AREA)
- Vascular Medicine (AREA)
- Reproductive Health (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2003181908 | 2003-06-25 | ||
PCT/JP2004/009263 WO2004113344A1 (ja) | 2003-06-25 | 2004-06-24 | ピラゾロピリミジン化合物のメタンスルホン酸塩、その結晶およびその製造方法 |
Publications (2)
Publication Number | Publication Date |
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NO20056093L NO20056093L (no) | 2006-03-24 |
NO332186B1 true NO332186B1 (no) | 2012-07-23 |
Family
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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NO20056093A NO332186B1 (no) | 2003-06-25 | 2005-12-21 | Metansulfonsyresalt av pyrazolpyrimidinforbindelse, krystall derav, fremgangsmate for fremstilling av det samme, farmasoytisk preparat samt anvendelse derav |
Country Status (19)
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US (1) | US7947697B1 (ru) |
EP (1) | EP1637531B1 (ru) |
JP (1) | JP4655276B2 (ru) |
KR (1) | KR101082227B1 (ru) |
CN (1) | CN100422186C (ru) |
AT (1) | ATE478873T1 (ru) |
AU (1) | AU2004249629B2 (ru) |
BR (1) | BRPI0411923A (ru) |
CA (1) | CA2529561C (ru) |
DE (1) | DE602004028820D1 (ru) |
ES (1) | ES2349393T3 (ru) |
IL (1) | IL172697A (ru) |
MX (1) | MXPA05013917A (ru) |
NO (1) | NO332186B1 (ru) |
NZ (1) | NZ544301A (ru) |
RU (1) | RU2345995C2 (ru) |
TW (1) | TWI356058B (ru) |
WO (1) | WO2004113344A1 (ru) |
ZA (1) | ZA200510450B (ru) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
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JPWO2005061508A1 (ja) * | 2003-12-22 | 2007-07-12 | 小野薬品工業株式会社 | 三環式複素環化合物およびその化合物を有効成分とする医薬 |
WO2005087775A1 (ja) * | 2004-03-15 | 2005-09-22 | Ono Pharmaceutical Co., Ltd. | 三環式複素環化合物およびその化合物を有効成分として含有する医薬組成物 |
CN112225732B (zh) * | 2019-07-15 | 2024-01-09 | 四川科瑞德制药股份有限公司 | 一种盐酸哌罗匹隆水合物晶型及其制备方法 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0503099A4 (en) | 1990-10-09 | 1993-12-01 | Otsuka Pharmaceutical Co., Ltd. | Pyrimidine derivative, production thereof, and androgen inhibitor |
CN1030768C (zh) * | 1990-10-09 | 1996-01-24 | 大塚制药株式会社 | 嘧啶衍生物或其药用盐的制备方法 |
JPH05112571A (ja) | 1990-10-19 | 1993-05-07 | Otsuka Pharmaceut Co Ltd | ピリミジン誘導体 |
WO1997011946A1 (fr) | 1995-09-28 | 1997-04-03 | Otsuka Pharmaceutical Factory, Inc. | Analgesiques |
JP2002517501A (ja) | 1998-06-09 | 2002-06-18 | ニューロゲン コーポレイション | ピリド[2,3−b]インドリジン誘導体およびそのアザ類似化合物;CRF1特異的リガンド |
US6531475B1 (en) | 1998-11-12 | 2003-03-11 | Neurocrine Biosciences, Inc. | CRF receptor antagonists and methods relating thereto |
TR200102178T2 (tr) | 1998-11-12 | 2002-01-21 | Neurocrine Biosciences, Inc. | CRF reseptör antagonistleri ve bunlarla ilgili yöntemler. |
JP2002529465A (ja) | 1998-11-12 | 2002-09-10 | ニューロクライン バイオサイエンシーズ, インコーポレイテッド | Crfレセプターアンタゴニストおよびcrfレセプターアンタゴニストに関する方法 |
ATE526330T1 (de) | 2000-12-28 | 2011-10-15 | Ono Pharmaceutical Co | Heterotrizyklische verbindungen als antagonisten des crf-rezeptors |
-
2004
- 2004-06-24 DE DE602004028820T patent/DE602004028820D1/de not_active Expired - Lifetime
- 2004-06-24 BR BRPI0411923-1A patent/BRPI0411923A/pt not_active IP Right Cessation
- 2004-06-24 RU RU2006101986/04A patent/RU2345995C2/ru not_active IP Right Cessation
- 2004-06-24 CN CNB2004800243652A patent/CN100422186C/zh not_active Expired - Fee Related
- 2004-06-24 JP JP2005507336A patent/JP4655276B2/ja not_active Expired - Fee Related
- 2004-06-24 CA CA2529561A patent/CA2529561C/en not_active Expired - Fee Related
- 2004-06-24 WO PCT/JP2004/009263 patent/WO2004113344A1/ja active Application Filing
- 2004-06-24 NZ NZ544301A patent/NZ544301A/en not_active IP Right Cessation
- 2004-06-24 EP EP04746732A patent/EP1637531B1/en not_active Expired - Lifetime
- 2004-06-24 MX MXPA05013917A patent/MXPA05013917A/es active IP Right Grant
- 2004-06-24 AU AU2004249629A patent/AU2004249629B2/en not_active Ceased
- 2004-06-24 ES ES04746732T patent/ES2349393T3/es not_active Expired - Lifetime
- 2004-06-24 AT AT04746732T patent/ATE478873T1/de not_active IP Right Cessation
- 2004-06-24 US US10/561,214 patent/US7947697B1/en not_active Expired - Fee Related
- 2004-06-24 TW TW093118239A patent/TWI356058B/zh not_active IP Right Cessation
-
2005
- 2005-12-20 IL IL172697A patent/IL172697A/en not_active IP Right Cessation
- 2005-12-21 NO NO20056093A patent/NO332186B1/no not_active IP Right Cessation
- 2005-12-22 ZA ZA200510450A patent/ZA200510450B/en unknown
- 2005-12-23 KR KR1020057024807A patent/KR101082227B1/ko not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
NO20056093L (no) | 2006-03-24 |
TW200504064A (en) | 2005-02-01 |
KR101082227B1 (ko) | 2011-11-09 |
RU2006101986A (ru) | 2006-07-27 |
BRPI0411923A (pt) | 2006-08-15 |
CA2529561C (en) | 2012-05-29 |
MXPA05013917A (es) | 2006-03-09 |
KR20060026060A (ko) | 2006-03-22 |
AU2004249629A1 (en) | 2004-12-29 |
JP4655276B2 (ja) | 2011-03-23 |
TWI356058B (en) | 2012-01-11 |
JPWO2004113344A1 (ja) | 2006-07-27 |
WO2004113344A1 (ja) | 2004-12-29 |
EP1637531A4 (en) | 2008-09-03 |
RU2345995C2 (ru) | 2009-02-10 |
EP1637531B1 (en) | 2010-08-25 |
CA2529561A1 (en) | 2004-12-29 |
NZ544301A (en) | 2008-08-29 |
CN1842530A (zh) | 2006-10-04 |
DE602004028820D1 (de) | 2010-10-07 |
ATE478873T1 (de) | 2010-09-15 |
US7947697B1 (en) | 2011-05-24 |
IL172697A0 (en) | 2006-04-10 |
AU2004249629B2 (en) | 2009-07-30 |
ES2349393T3 (es) | 2010-12-30 |
EP1637531A1 (en) | 2006-03-22 |
CN100422186C (zh) | 2008-10-01 |
ZA200510450B (en) | 2006-12-27 |
IL172697A (en) | 2013-05-30 |
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