YU80700A - Novi 17-halogenizovani 19-nor steroidi, postupak i međuproizvodi za njihovo pripremanje, njihova primena kao medikamenata i farmaceutske kompozicije koje ih sadrže - Google Patents
Novi 17-halogenizovani 19-nor steroidi, postupak i međuproizvodi za njihovo pripremanje, njihova primena kao medikamenata i farmaceutske kompozicije koje ih sadržeInfo
- Publication number
- YU80700A YU80700A YU80700A YU80700A YU80700A YU 80700 A YU80700 A YU 80700A YU 80700 A YU80700 A YU 80700A YU 80700 A YU80700 A YU 80700A YU 80700 A YU80700 A YU 80700A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- same
- medicines
- intermediates
- pharmaceutical compositions
- steroids
- Prior art date
Links
- 229940079593 drug Drugs 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title abstract 2
- 239000000543 intermediate Substances 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
- C07J41/0083—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Reproductive Health (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Pronalazak se odnosi na jedinjenje formule (I) kod kojih je posebno X = halogen, Y = jednostruka veza, O, NH, S, SO ili SO2, Z = vodonik ili halogen, n, R1 R2, R3 i R4 su kako su definisani u opisu. Pronalazak se dalje odnosi na postupak i na medjurpoizvode za pripremanje ovih jedinjenja, na njihovu primenu kao medikamenata i na farmaceutske kompozicije koje ih sadrže.[The invention concerns compounds of formula (I) wherein, in particular: X = halogen; Y = single bond, O, NH, S, SO or SO2; Z = hydrogen or halogen; n, R1, R2, R3 and R4 are as defined in the description. The invention also concerns the method and intermediates for preparing said compounds, their use as medicines and pharmaceutical compositions containing them.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9807898A FR2780060B1 (fr) | 1998-06-23 | 1998-06-23 | Nouveaux 19-nor steroides 17-halogenes, procede et intermediaires de preparation, application comme medicaments et compositions pharmaceutiques les renfermant |
Publications (1)
Publication Number | Publication Date |
---|---|
YU80700A true YU80700A (sh) | 2003-10-31 |
Family
ID=9527717
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
YU80700A YU80700A (sh) | 1998-06-23 | 1999-06-22 | Novi 17-halogenizovani 19-nor steroidi, postupak i međuproizvodi za njihovo pripremanje, njihova primena kao medikamenata i farmaceutske kompozicije koje ih sadrže |
Country Status (37)
Country | Link |
---|---|
US (2) | US6423700B1 (sh) |
EP (1) | EP1090027B1 (sh) |
JP (1) | JP4509380B2 (sh) |
KR (1) | KR20010034919A (sh) |
CN (1) | CN1313862A (sh) |
AP (1) | AP1579A (sh) |
AR (1) | AR018916A1 (sh) |
AT (1) | ATE237628T1 (sh) |
AU (1) | AU771369B2 (sh) |
BR (1) | BR9912206A (sh) |
CA (1) | CA2336167A1 (sh) |
CZ (1) | CZ296246B6 (sh) |
DE (1) | DE69906972T2 (sh) |
DK (1) | DK1090027T3 (sh) |
DZ (1) | DZ2827A1 (sh) |
EA (1) | EA003325B1 (sh) |
ES (1) | ES2196879T3 (sh) |
FR (1) | FR2780060B1 (sh) |
HK (1) | HK1039945A1 (sh) |
HR (1) | HRP20000893A2 (sh) |
HU (1) | HUP0103194A3 (sh) |
ID (1) | ID27410A (sh) |
IL (1) | IL140416A (sh) |
MA (1) | MA26656A1 (sh) |
MY (1) | MY118101A (sh) |
NO (1) | NO318381B1 (sh) |
NZ (1) | NZ508535A (sh) |
PL (1) | PL345073A1 (sh) |
PT (1) | PT1090027E (sh) |
SK (1) | SK19492000A3 (sh) |
TN (1) | TNSN99130A1 (sh) |
TR (1) | TR200003857T2 (sh) |
TW (1) | TW550077B (sh) |
UA (1) | UA66867C2 (sh) |
WO (1) | WO1999067274A1 (sh) |
YU (1) | YU80700A (sh) |
ZA (1) | ZA200007355B (sh) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP3922104B2 (ja) * | 2002-06-07 | 2007-05-30 | 富士通株式会社 | ポイント管理装置、ポイント管理システム、ポイント管理方法、およびポイント管理プログラム |
FR2854402B1 (fr) * | 2003-04-29 | 2008-07-04 | Aventis Pharma Sa | Nouveau procede et intermediaires de preparation de composes 19-nor-steroides |
FR2854403B1 (fr) * | 2003-04-29 | 2008-07-11 | Aventis Pharma Sa | Nouveau procede et intermediaires de preparation de composes 19-nor-steroides 17-halogenes |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3079408A (en) * | 1963-02-26 | Ig-bisoxygenated iy-haloestra- | ||
US3264327A (en) * | 1962-07-27 | 1966-08-02 | Syntex Corp | 17alpha-fluoro-, 17beta-chlorofluoroacetoxy- and 17beta-methyl-delta4-and delta5-androstene derivatives |
US3413321A (en) * | 1966-06-03 | 1968-11-26 | Du Pont | Selected 17-fluoro-delta16 steroids |
FR2528434B1 (fr) * | 1982-06-11 | 1985-07-19 | Roussel Uclaf | Nouveaux 19-nor steroides substitues en 11b et eventuellement en 2, leur procede de preparation et leur application comme medicament |
FR2640977A2 (en) * | 1982-06-11 | 1990-06-29 | Roussel Uclaf | New position-11 substituted 19-norsteroids and their application as medicinal products. |
FR2685332A1 (fr) * | 1991-12-20 | 1993-06-25 | Roussel Uclaf | Nouveaux 19-nor sterouides ayant en position 11beta une chaine thiocarbonee, leur procede de preparation et les intermediaires et leur application a titre de medicaments. |
FR2757519B1 (fr) * | 1996-12-23 | 1999-06-11 | Hoechst Marion Roussel Inc | Steroides substitues en position 11, leur procede de preparation, leur application comme medicament et les compositions pharmaceutiques les renfermant |
FR2761992B1 (fr) * | 1997-04-09 | 1999-06-11 | Hoechst Marion Roussel Inc | Nouveaux steroides 4-halogenes, leur procede et intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant |
FR2771096B1 (fr) * | 1997-11-17 | 2000-08-11 | Hoechst Marion Roussel Inc | Nouveaux 19-nor steroides, substitues en position 11beta, procede et intermediaires de preparation, application comme medicaments et compositions pharmaceutiques les renfermant |
-
1998
- 1998-06-23 FR FR9807898A patent/FR2780060B1/fr not_active Expired - Lifetime
-
1999
- 1999-06-07 TW TW088109436A patent/TW550077B/zh not_active IP Right Cessation
- 1999-06-21 MA MA25638A patent/MA26656A1/fr unknown
- 1999-06-21 MY MYPI99002542A patent/MY118101A/en unknown
- 1999-06-22 TN TNTNSN99130A patent/TNSN99130A1/fr unknown
- 1999-06-22 DZ DZ990127A patent/DZ2827A1/xx active
- 1999-06-22 IL IL14041699A patent/IL140416A/xx not_active IP Right Cessation
- 1999-06-22 HU HU0103194A patent/HUP0103194A3/hu unknown
- 1999-06-22 WO PCT/FR1999/001491 patent/WO1999067274A1/fr not_active Application Discontinuation
- 1999-06-22 AR ARP990102991A patent/AR018916A1/es not_active Application Discontinuation
- 1999-06-22 ES ES99957166T patent/ES2196879T3/es not_active Expired - Lifetime
- 1999-06-22 DE DE69906972T patent/DE69906972T2/de not_active Expired - Lifetime
- 1999-06-22 AT AT99957166T patent/ATE237628T1/de not_active IP Right Cessation
- 1999-06-22 BR BR9912206-5A patent/BR9912206A/pt not_active IP Right Cessation
- 1999-06-22 SK SK1949-2000A patent/SK19492000A3/sk unknown
- 1999-06-22 PL PL99345073A patent/PL345073A1/xx not_active Application Discontinuation
- 1999-06-22 CZ CZ20004834A patent/CZ296246B6/cs not_active IP Right Cessation
- 1999-06-22 AU AU42705/99A patent/AU771369B2/en not_active Ceased
- 1999-06-22 AP APAP/P/2000/002007A patent/AP1579A/en active
- 1999-06-22 CA CA002336167A patent/CA2336167A1/fr not_active Abandoned
- 1999-06-22 US US09/720,565 patent/US6423700B1/en not_active Expired - Lifetime
- 1999-06-22 JP JP2000555925A patent/JP4509380B2/ja not_active Expired - Lifetime
- 1999-06-22 ID IDW20002721A patent/ID27410A/id unknown
- 1999-06-22 NZ NZ508535A patent/NZ508535A/xx unknown
- 1999-06-22 KR KR1020007014649A patent/KR20010034919A/ko not_active Application Discontinuation
- 1999-06-22 UA UA2001010468A patent/UA66867C2/uk unknown
- 1999-06-22 PT PT99957166T patent/PT1090027E/pt unknown
- 1999-06-22 YU YU80700A patent/YU80700A/sh unknown
- 1999-06-22 DK DK99957166T patent/DK1090027T3/da active
- 1999-06-22 CN CN99809983A patent/CN1313862A/zh active Pending
- 1999-06-22 EP EP99957166A patent/EP1090027B1/fr not_active Expired - Lifetime
- 1999-06-22 TR TR2000/03857T patent/TR200003857T2/xx unknown
- 1999-06-22 EA EA200100069A patent/EA003325B1/ru unknown
-
2000
- 2000-12-11 ZA ZA200007355A patent/ZA200007355B/en unknown
- 2000-12-21 HR HR20000893A patent/HRP20000893A2/hr not_active Application Discontinuation
- 2000-12-21 NO NO20006573A patent/NO318381B1/no unknown
-
2002
- 2002-02-28 HK HK02101559.9A patent/HK1039945A1/zh unknown
- 2002-06-18 US US10/173,914 patent/US6566542B2/en not_active Expired - Lifetime
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