YU40258B - Process for obtaining new 4-(3-subt.-4-methoxy-phenyl)-2-pyrrolidones - Google Patents
Process for obtaining new 4-(3-subt.-4-methoxy-phenyl)-2-pyrrolidonesInfo
- Publication number
- YU40258B YU40258B YU632/75A YU63275A YU40258B YU 40258 B YU40258 B YU 40258B YU 632/75 A YU632/75 A YU 632/75A YU 63275 A YU63275 A YU 63275A YU 40258 B YU40258 B YU 40258B
- Authority
- YU
- Yugoslavia
- Prior art keywords
- subt
- pyrrolidones
- methoxy
- phenyl
- obtaining new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
- C07D207/273—2-Pyrrolidones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
- C07D207/277—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
- C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
- C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C47/00—Compounds having —CHO groups
- C07C47/52—Compounds having —CHO groups bound to carbon atoms of six—membered aromatic rings
- C07C47/575—Compounds having —CHO groups bound to carbon atoms of six—membered aromatic rings containing ether groups, groups, groups, or groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Psychiatry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pyrrole Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE2413935A DE2413935A1 (de) | 1974-03-20 | 1974-03-20 | 4-(polyalkoxy-phenyl)-2-pyrrolidone |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| YU63275A YU63275A (en) | 1982-06-30 |
| YU40258B true YU40258B (en) | 1985-10-31 |
Family
ID=5910915
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| YU632/75A YU40258B (en) | 1974-03-20 | 1975-03-17 | Process for obtaining new 4-(3-subt.-4-methoxy-phenyl)-2-pyrrolidones |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US4012495A (cs) |
| JP (1) | JPS6011028B2 (cs) |
| AT (1) | AT347931B (cs) |
| BE (1) | BE826923A (cs) |
| CA (1) | CA1069517A (cs) |
| CH (1) | CH621338A5 (cs) |
| CS (1) | CS214738B2 (cs) |
| DD (1) | DD119229A5 (cs) |
| DE (1) | DE2413935A1 (cs) |
| DK (1) | DK139965C (cs) |
| ES (1) | ES435750A1 (cs) |
| FR (1) | FR2264531B1 (cs) |
| GB (1) | GB1498705A (cs) |
| HU (1) | HU174074B (cs) |
| IE (1) | IE40865B1 (cs) |
| IL (1) | IL46883A (cs) |
| NL (1) | NL7503367A (cs) |
| SE (1) | SE402010B (cs) |
| SU (1) | SU649312A3 (cs) |
| YU (1) | YU40258B (cs) |
Families Citing this family (114)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4193926A (en) | 1974-03-20 | 1980-03-18 | Schering Aktiengesellschaft | 4-(Polyalkoxy phenyl)-2-pyrrolidones |
| DE2541855A1 (de) * | 1975-09-18 | 1977-03-31 | Schering Ag | 4-(polyalkoxy-phenyl)-2-pyrrolidone ii |
| CU21107A3 (es) | 1978-02-10 | 1988-02-01 | Hoffmann La Roche | Pyrrolidines derivatives |
| IL57266A (en) * | 1978-06-12 | 1982-12-31 | Mundipharma Ag | Production of pyrrolidin-2-ones and of 3-pyrrolin-2-ones |
| CA1124247A (en) * | 1979-08-09 | 1982-05-25 | Hoffmann-La Roche Limited | Pyrrolidine derivatives |
| GB2123288A (en) * | 1982-07-16 | 1984-02-01 | Wellcome Found | Anti-thrombotic agent |
| US4584313A (en) * | 1984-05-07 | 1986-04-22 | Warner-Lambert Company | (Substituted-phenyl)-5-oxo-2-pyrrolidinepropanoic acids and esters thereof, and use for reversing electroconvulsive shock-induced amnesia |
| US4548947A (en) * | 1984-05-07 | 1985-10-22 | Warner-Lambert Company | 1-(Substituted-aryl)-dihydro-1H-pyrrolizine-3,5-[2H,6H-]diones and use for reversing amnesia |
| DE3438839A1 (de) * | 1984-10-19 | 1986-04-24 | Schering AG, 1000 Berlin und 4709 Bergkamen | Pharmazeutische praeparate |
| US5783591A (en) * | 1984-10-19 | 1998-07-21 | Schering Aktiengesellschaft | Administration of oxazolidinone and pyrolidinone compounds for the treatment of inflammation |
| US5459145A (en) * | 1988-01-19 | 1995-10-17 | Pfizer Inc. | Calcium independent camp phosphodiesterase inhibitor antidepressant |
| FI875724A7 (fi) * | 1986-04-29 | 1987-12-28 | Pfizer | Kalsiumista riippumaton cAMP fosfodiesteraasi-inhibiittori-masennukse nvastainen lääke. |
| FI875101A7 (fi) * | 1986-12-03 | 1988-06-04 | Tanabe Seiyaku Co | Laktaamijohdannaiset ja niitä sisältävät valmisteet. |
| US4971959A (en) * | 1987-04-14 | 1990-11-20 | Warner-Lambert Company | Trisubstituted phenyl analogs having activity for congestive heart failure |
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| US4960457A (en) * | 1988-12-27 | 1990-10-02 | Ici Americas Inc. | Substituted 1,3-diphenyl pyrrolidones and their use as herbicides |
| DE3921593A1 (de) * | 1989-06-28 | 1991-01-10 | Schering Ag | Verfahren zur racemattrennung von 4-aryl-2-oxo-pyrrolidin-3-carbonsaeure-ester |
| JP2578001B2 (ja) * | 1989-12-11 | 1997-02-05 | 明治製菓株式会社 | 抗痴呆薬 |
| DE3943385A1 (de) * | 1989-12-27 | 1991-07-04 | Schering Ag | Mittel zur transdermalen applikation enthaltend rolipram |
| DD299058A5 (de) * | 1990-01-31 | 1992-03-26 | Arzneimittelwerk Dresden Gmbh,De | Verfahren zur herstellung von n-acyl-4-phenyl-pyrrolidin-2-onen mit cerebroprotektiver wirkung |
| GB9009395D0 (en) * | 1990-04-26 | 1990-06-20 | Orion Yhtymae Oy | Cyclic hydroxamic acids and their use |
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| CN107090016A (zh) | 2011-03-01 | 2017-08-25 | 辛纳吉制药公司 | 制备鸟苷酸环化酶c激动剂的方法 |
| ES2395801B1 (es) | 2011-06-23 | 2014-06-06 | María Carmen PARDINA PALLEJÀ | "pentoxifilina por vía transvaginal para el tratamiento de la infertilidad" |
| US9545446B2 (en) | 2013-02-25 | 2017-01-17 | Synergy Pharmaceuticals, Inc. | Agonists of guanylate cyclase and their uses |
| AU2014235209B2 (en) | 2013-03-15 | 2018-06-14 | Bausch Health Ireland Limited | Guanylate cyclase receptor agonists combined with other drugs |
| US9708367B2 (en) | 2013-03-15 | 2017-07-18 | Synergy Pharmaceuticals, Inc. | Agonists of guanylate cyclase and their uses |
| CN105764916B (zh) | 2013-06-05 | 2021-05-18 | 博士医疗爱尔兰有限公司 | 鸟苷酸环化酶c的超纯激动剂、制备和使用所述激动剂的方法 |
| CN114404588A (zh) | 2013-08-09 | 2022-04-29 | 阿德利克斯公司 | 用于抑制磷酸盐转运的化合物和方法 |
| EP3972599B1 (en) | 2019-05-21 | 2025-10-22 | Ardelyx, Inc. | Combination for lowering serum phosphate in a patient |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1516776A (fr) | 1966-07-21 | 1968-03-15 | Rhone Poulenc Sa | Nouveaux dérivés du pyrrole et leur préparation |
| GB1350582A (en) * | 1970-07-24 | 1974-04-18 | Ucb Sa | Cerivatives of 2-pyrrolidinone |
-
1974
- 1974-03-20 DE DE2413935A patent/DE2413935A1/de active Granted
-
1975
- 1975-03-10 SU SU752111302A patent/SU649312A3/ru active
- 1975-03-17 YU YU632/75A patent/YU40258B/xx unknown
- 1975-03-18 CH CH345775A patent/CH621338A5/de not_active IP Right Cessation
- 1975-03-18 DK DK110675A patent/DK139965C/da not_active IP Right Cessation
- 1975-03-18 ES ES435750A patent/ES435750A1/es not_active Expired
- 1975-03-18 DD DD184858A patent/DD119229A5/xx unknown
- 1975-03-19 SE SE7503157A patent/SE402010B/xx not_active IP Right Cessation
- 1975-03-19 AT AT210975A patent/AT347931B/de not_active IP Right Cessation
- 1975-03-19 CS CS751860A patent/CS214738B2/cs unknown
- 1975-03-19 HU HU75SCHE514A patent/HU174074B/hu unknown
- 1975-03-20 IE IE611/75A patent/IE40865B1/xx unknown
- 1975-03-20 NL NL7503367A patent/NL7503367A/xx not_active Application Discontinuation
- 1975-03-20 CA CA222,720A patent/CA1069517A/en not_active Expired
- 1975-03-20 JP JP50034220A patent/JPS6011028B2/ja not_active Expired
- 1975-03-20 BE BE154536A patent/BE826923A/xx not_active IP Right Cessation
- 1975-03-20 US US05/560,193 patent/US4012495A/en not_active Expired - Lifetime
- 1975-03-20 GB GB11686/75A patent/GB1498705A/en not_active Expired
- 1975-03-20 FR FR7508701A patent/FR2264531B1/fr not_active Expired
- 1975-03-20 IL IL46883A patent/IL46883A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FR2264531B1 (cs) | 1978-07-28 |
| ATA210975A (de) | 1978-06-15 |
| SE7503157L (sv) | 1975-11-28 |
| AT347931B (de) | 1979-01-25 |
| NL7503367A (nl) | 1975-09-23 |
| US4012495A (en) | 1977-03-15 |
| IL46883A0 (en) | 1975-05-22 |
| SE402010B (sv) | 1978-06-12 |
| CS214738B2 (en) | 1982-05-28 |
| DK139965B (da) | 1979-05-28 |
| DK110675A (cs) | 1975-09-21 |
| BE826923A (fr) | 1975-09-22 |
| DK139965C (da) | 1979-10-29 |
| IL46883A (en) | 1979-09-30 |
| CH621338A5 (cs) | 1981-01-30 |
| YU63275A (en) | 1982-06-30 |
| SU649312A3 (ru) | 1979-02-25 |
| GB1498705A (en) | 1978-01-25 |
| DE2413935A1 (de) | 1975-10-16 |
| DD119229A5 (cs) | 1976-04-12 |
| ES435750A1 (es) | 1976-12-16 |
| AU7931075A (en) | 1976-09-23 |
| HU174074B (hu) | 1979-10-28 |
| CA1069517A (en) | 1980-01-08 |
| DE2413935C2 (cs) | 1988-05-26 |
| JPS50157360A (cs) | 1975-12-19 |
| IE40865L (en) | 1975-09-20 |
| JPS6011028B2 (ja) | 1985-03-22 |
| IE40865B1 (en) | 1979-08-29 |
| FR2264531A1 (cs) | 1975-10-17 |
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