YU35361B - Process for obtaining base-substituted benzyl-phthalazone derivatives - Google Patents

Process for obtaining base-substituted benzyl-phthalazone derivatives

Info

Publication number
YU35361B
YU35361B YU112/72A YU11272A YU35361B YU 35361 B YU35361 B YU 35361B YU 112/72 A YU112/72 A YU 112/72A YU 11272 A YU11272 A YU 11272A YU 35361 B YU35361 B YU 35361B
Authority
YU
Yugoslavia
Prior art keywords
substituted benzyl
obtaining base
phthalazone derivatives
phthalazone
derivatives
Prior art date
Application number
YU112/72A
Other languages
English (en)
Other versions
YU11272A (en
Inventor
Vogelsang Dietrich
Dietrich Vogelsang
Scheffler Gerhard
Gerhard Scheffler
Brock Norbert
Norbert Brock
Original Assignee
Asta Werke Ag Chem Fab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asta Werke Ag Chem Fab filed Critical Asta Werke Ag Chem Fab
Publication of YU11272A publication Critical patent/YU11272A/xx
Publication of YU35361B publication Critical patent/YU35361B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
YU112/72A 1971-01-22 1972-01-17 Process for obtaining base-substituted benzyl-phthalazone derivatives YU35361B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH101271A CH572914A5 (fr) 1971-01-22 1971-01-22

Publications (2)

Publication Number Publication Date
YU11272A YU11272A (en) 1980-06-30
YU35361B true YU35361B (en) 1980-12-31

Family

ID=4200381

Family Applications (1)

Application Number Title Priority Date Filing Date
YU112/72A YU35361B (en) 1971-01-22 1972-01-17 Process for obtaining base-substituted benzyl-phthalazone derivatives

Country Status (21)

Country Link
AR (1) AR197293A1 (fr)
AT (1) AT313288B (fr)
AU (1) AU3767472A (fr)
BE (1) BE778269A (fr)
CA (1) CA1010041A (fr)
CH (1) CH572914A5 (fr)
DE (1) DE2164058C3 (fr)
DK (1) DK136981B (fr)
ES (1) ES398949A1 (fr)
FI (1) FI53704C (fr)
FR (1) FR2122517B1 (fr)
GB (1) GB1377231A (fr)
HK (1) HK62577A (fr)
HU (1) HU163979B (fr)
IL (1) IL38496A (fr)
NL (1) NL177116C (fr)
OA (1) OA04087A (fr)
PL (1) PL88930B1 (fr)
SE (1) SE404604B (fr)
YU (1) YU35361B (fr)
ZA (1) ZA718712B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE49205T1 (de) * 1984-09-14 1990-01-15 Asta Pharma Ag Substituierte benzylphthalazinon-derivate.
PT88984B (pt) * 1987-11-13 1993-01-29 Asta Medica Ag Processo para a preparação de embonato de azelastina e de composições earmacâutxcas que 0 contêm como ingrediente activo
ATE84968T1 (de) * 1987-11-13 1993-02-15 Asta Medica Ag Azelastin enthaltende arzneimittel zur anwendung in der nase und/oder am auge.
DE3836579A1 (de) * 1987-11-13 1989-05-24 Asta Pharma Ag Azelastin enthaltende arzneimittel zur anwendung in der nase und/oder am auge
EP0316639B1 (fr) * 1987-11-13 1994-06-08 ASTA Medica Aktiengesellschaft Azélastine-embonate, procédé pour sa préparation et préparations pharmaceutiques qui contiennent l'azélastine-embonate comme produit actif
DE3912292A1 (de) * 1988-04-20 1989-11-09 Asta Pharma Ag Azelastin enthaltende arzneimittel mit kontrollierter wirkstoffabgabe
US5110814A (en) * 1989-01-11 1992-05-05 Asta Pharma Ag Azelastine and its salts used to combat psoriasis
ES2055216T3 (es) * 1989-05-05 1994-08-16 Asta Medica Ag Sales de la azelastina con solubilidad mejorada.
DE4207234A1 (de) * 1992-03-07 1993-09-09 Asta Medica Ag Neue aminocarbonsaeure-derivate mit antiallergischer/antiasthmatischer wirkung und verfahren zu deren herstellung
DE4343409C2 (de) * 1993-12-18 1997-03-20 Asta Medica Ag Verbessertes Verfahren zur Herstellung von Hexahydroazepinonen und Hexahydroazepinolen
DE4345224C2 (de) * 1993-12-18 1999-07-01 Asta Medica Ag Verfahren zur Herstellung von Säureadditionssalzen des Azelastins und Flezelastins
GB2389530B (en) 2002-06-14 2007-01-10 Cipla Ltd Pharmaceutical compositions
US20070020330A1 (en) 2004-11-24 2007-01-25 Medpointe Healthcare Inc. Compositions comprising azelastine and methods of use thereof
DK2522365T3 (en) 2004-11-24 2017-02-06 Meda Pharmaceuticals Inc Compositions comprising azelastine and methods for its use
US8758816B2 (en) 2004-11-24 2014-06-24 Meda Pharmaceuticals Inc. Compositions comprising azelastine and methods of use thereof
DE602007010118D1 (de) * 2006-04-20 2010-12-09 Glaxo Group Ltd 2-substituierte 4-benzylphthalazinonderivate als histamin-h1- und h3-antagonisten

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1046625B (de) * 1957-08-15 1958-12-18 Hydrierwerk Rodleben Veb Verfahren zur Herstellung basisch substituierter Phthalazone
GB1100911A (en) * 1963-08-20 1968-01-24 Benger Lab Ltd Phthalazine derivatives
FR1512879A (fr) * 1966-10-28 1968-02-09 Hydrierwerk Rodleben Veb Procédé pour la fabrication de phtalazones avec substituants basiques

Also Published As

Publication number Publication date
CA1010041A (en) 1977-05-10
SU440838A3 (fr) 1974-08-25
GB1377231A (en) 1974-12-11
DE2164058B2 (de) 1980-10-23
NL177116B (nl) 1985-03-01
SE404604B (sv) 1978-10-16
OA04087A (fr) 1979-10-30
DK136981C (fr) 1978-06-05
NL177116C (nl) 1985-08-01
FI53704C (fi) 1978-07-10
YU11272A (en) 1980-06-30
NL7200400A (fr) 1972-07-25
IL38496A0 (en) 1972-03-28
PL88930B1 (fr) 1976-10-30
BE778269A (fr) 1972-07-19
FI53704B (fr) 1978-03-31
HU163979B (fr) 1973-12-28
HK62577A (en) 1977-12-30
CH572914A5 (fr) 1976-02-27
DE2164058C3 (de) 1981-08-13
AT313288B (de) 1974-02-11
FR2122517A1 (fr) 1972-09-01
AU3767472A (en) 1973-07-12
DE2164058A1 (de) 1972-07-27
FR2122517B1 (fr) 1975-08-01
IL38496A (en) 1975-05-22
DK136981B (da) 1977-12-27
ZA718712B (en) 1972-09-27
ES398949A1 (es) 1975-06-01
AR197293A1 (es) 1974-03-29

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