WO1996016954A1 - Derives de l'acide anthranilique utiles en tant que fongicides - Google Patents

Derives de l'acide anthranilique utiles en tant que fongicides Download PDF

Info

Publication number
WO1996016954A1
WO1996016954A1 PCT/EP1995/004800 EP9504800W WO9616954A1 WO 1996016954 A1 WO1996016954 A1 WO 1996016954A1 EP 9504800 W EP9504800 W EP 9504800W WO 9616954 A1 WO9616954 A1 WO 9616954A1
Authority
WO
WIPO (PCT)
Prior art keywords
optionally substituted
heterocyclyl
alkyl
cycloalkenyl
alkenyl
Prior art date
Application number
PCT/EP1995/004800
Other languages
English (en)
Inventor
Peter Dominic Riordan
Peter John West
Ian Kenneth Boddy
Original Assignee
Agrevo Uk Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Agrevo Uk Limited filed Critical Agrevo Uk Limited
Priority to EP95941681A priority Critical patent/EP0794950A1/fr
Priority to AU43028/96A priority patent/AU4302896A/en
Publication of WO1996016954A1 publication Critical patent/WO1996016954A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/06—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/36—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A01N43/52—1,3-Diazoles; Hydrogenated 1,3-diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/04—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • C07D249/06—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles with aryl radicals directly attached to ring atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/06—1,2,3-Thiadiazoles; Hydrogenated 1,2,3-thiadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/70—Nitro radicals
    • C07D307/71—Nitro radicals attached in position 5
    • C07D307/72—Nitro radicals attached in position 5 with hydrocarbon radicals, substituted by nitrogen-containing radicals, attached in position 2
    • C07D307/73—Nitro radicals attached in position 5 with hydrocarbon radicals, substituted by nitrogen-containing radicals, attached in position 2 by amino or imino, or substituted amino or imino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/84—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/42—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms with nitro or nitroso radicals directly attached to ring carbon atoms
    • C07D333/44—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms with nitro or nitroso radicals directly attached to ring carbon atoms attached in position 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/72—Benzo[c]thiophenes; Hydrogenated benzo[c]thiophenes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Composés de la formule (I) dans laquelle A représente un groupe hétéroaryle à 5 chaînons, éventuellement substitué, comprenant au moins un hétéroatome choisi parmi azote, soufre et oxygène, lequel est éventuellement substitué par un ou plusieurs substituants du groupe R2; R1 représente alkyle, cycloalkyle, cycloalcényle, alcényle, alcynyle ou amino (chacun de ceux-ci étant éventuellement substitué), Y1-X-, halogène, cyano, nitro, acyle, acyloxy, hétérocyclyle éventuellement substitué ou phényle éventuellement substitué; ou il représente deux groupes adjacents qui, avec les atomes de carbone auxquels ils sont attachés, peuvent former un noyau benzo éventuellement substitué; R2 possède les mêmes notations que R1, ou il représente deux groupes adjacents qui, avec les atomes de carbone auxquels ils sont attachés, peuvent former un noyau hétérocyclique éventuellement substitué; Y représente alkyle, cycloalkyle, cycloalcényle, alcényle ou alcynyle, chacun étant éventuellement substitué, hydrogène ou acyle; Y1 possède la même notation que Y ou il représente phényle éventuellement substitué ou hétérocyclyle éventuellement substitué; Z représente C(=X?1)-X2-R3¿, cyano, nitro, amino, acyle, hétérocyclyle éventuellement substitué, -C(R?5)=N-OR6¿ ou -C(R?5)=N-NR6R7; R3¿ représente alkyle, cycloalkyle, cycloalcényle, alcényle, alcynyle, phényle ou hétérocyclyle, chacun étant éventuellement substitué, hydrogène ou un groupe cationique inorganique ou organique; X1 et X2 qui peuvent être semblables ou différents, représentent O ou S; R?5, R6 et R7¿, qui peuvent être semblables ou différents, représentent alkyle, cycloalkyle, cycloalcényle, alcényle, alcynyle, phényle ou hétérocyclyle, chacun étant éventuellement substitué, ou hydrogène, ou bien R6 et R7, ensemble avec l'atome (les atomes) auquel (auxquels) ils sont attachés, peuvent former un noyau; et n vaut 0 à 4. Ces composés possèdent une activité fongicide.
PCT/EP1995/004800 1994-12-02 1995-12-01 Derives de l'acide anthranilique utiles en tant que fongicides WO1996016954A1 (fr)

Priority Applications (2)

Application Number Priority Date Filing Date Title
EP95941681A EP0794950A1 (fr) 1994-12-02 1995-12-01 Derives de l'acide anthranilique utiles en tant que fongicides
AU43028/96A AU4302896A (en) 1994-12-02 1995-12-01 Derivatives of anthranilic acid useful as fungicides

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9424379.7 1994-12-02
GB9424379A GB9424379D0 (en) 1994-12-02 1994-12-02 Fungicides

Publications (1)

Publication Number Publication Date
WO1996016954A1 true WO1996016954A1 (fr) 1996-06-06

Family

ID=10765345

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP1995/004800 WO1996016954A1 (fr) 1994-12-02 1995-12-01 Derives de l'acide anthranilique utiles en tant que fongicides

Country Status (6)

Country Link
EP (1) EP0794950A1 (fr)
AU (1) AU4302896A (fr)
GB (1) GB9424379D0 (fr)
IL (1) IL116234A0 (fr)
WO (1) WO1996016954A1 (fr)
ZA (1) ZA9510223B (fr)

Cited By (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997030047A1 (fr) * 1996-02-17 1997-08-21 Agrevo Uk Limited 1,2,4 oxadiazoles fongicides et analogues
WO1998018792A1 (fr) * 1996-10-28 1998-05-07 Merck Sharp & Dohme Limited DERIVES DE LA THIENYLCYCLOHEXANONE UTILISES COMME LIGANDS DU SOUS-TYPE α-5 DE RECEPTEUR DU GABA¿A?
GB2336588A (en) * 1998-04-23 1999-10-27 Merck Sharp & Dohme Benzo[c]thiophene Derivatives for Enhancing Cognition
US6143773A (en) * 1998-04-23 2000-11-07 Merck Sharp & Dohme Limited Substituted thienobenzisoxazole derivatives for enhancing cognition
US6156761A (en) * 1998-04-23 2000-12-05 Merck Sharpe & Dohme Limited Substituted tetralone derivatives for enhancing cognition
WO2001058879A1 (fr) * 2000-02-09 2001-08-16 The Procter & Gamble Company 2-phenylcarbamoyl-benzimidazoles
US6395766B1 (en) 1998-06-04 2002-05-28 Merck Sharp & Dohme Limited Tetrahydroindolone derivatives as gabaaalpha5 ligands for enhancing cognition
JP2002524557A (ja) * 1998-09-16 2002-08-06 バイエル アクチェンゲゼルシャフト イソチアゾールカルボン酸アミド類
WO2003016304A1 (fr) * 2001-08-15 2003-02-27 E. I. Du Pont De Nemours And Company Amides aryle ortho-heterocycliques substitues permettant de lutter contre des ravageurs invertebres
EP1394159A1 (fr) * 2002-08-13 2004-03-03 Warner-Lambert Company LLC Nouveaux dérivés de thiophène, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent
WO2004018461A2 (fr) * 2002-08-23 2004-03-04 Pharmacia & Upjohn Company Llc Derives d'acide benzoique antibacteriens
WO2005004606A2 (fr) * 2003-07-10 2005-01-20 Bayer Cropscience Ag Pyridinylanilides
WO2005085234A3 (fr) * 2004-03-03 2006-01-26 Syngenta Participations Ag Nouveaux insecticides
WO2006068618A1 (fr) * 2004-12-23 2006-06-29 Astrazeneca Ab Nouveaux composés
US7078419B2 (en) 2003-03-10 2006-07-18 Boehringer Ingelheim Pharmaceuticals, Inc. Cytokine inhibitors
US7223782B2 (en) * 2001-11-01 2007-05-29 Icagen, Inc. Pyrazole-amides and -sulfonamides
EP1846388A1 (fr) * 2005-01-25 2007-10-24 Synta Pharmaceuticals Corporation Composes de thiophene utilises contre l'inflammation et les troubles lies a l'immunite
JP2008517944A (ja) * 2004-10-22 2008-05-29 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Ｃ−ｆｍｓキナーゼの阻害剤
WO2009054468A1 (fr) * 2007-10-24 2009-04-30 Astellas Pharma Inc. Composé à base d'azolecarboxamide ou son sel
JP2009535311A (ja) * 2006-04-28 2009-10-01 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト 殺虫化合物
WO2010035886A1 (fr) * 2008-09-25 2010-04-01 住友化学株式会社 Composition à usage agricole qui contrôle ou empêche une maladie botanique provoquée par des agents pathogènes de plante
US8163746B2 (en) 2006-04-19 2012-04-24 Astellas Pharma Inc. Azolecarboxamide derivative
CN104529900A (zh) * 2014-12-31 2015-04-22 南开大学 1-取代-n-取代苯基-5-氨基-1h-吡唑-4-甲酰胺类化合物的杀菌活性
EP3315028A1 (fr) * 2016-10-27 2018-05-02 Kemijski Institut Inhibiteur de nlp proteines comme agent phytopharmaceutiques pour le contrôle d'un agent pathogene vegetal
JP2019507141A (ja) * 2016-02-11 2019-03-14 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 有害生物防除剤としての置換２−オキシイミダゾリル−カルボキサミド類
CN110105347A (zh) * 2019-06-18 2019-08-09 浙江工业大学 一种2-(2-吡啶基)-1,3-恶唑酰胺类衍生物及其制备方法和应用
CN110693869A (zh) * 2019-10-23 2020-01-17 华南理工大学 2-(甲氨基)苯甲酸甲酯的应用
WO2021035258A1 (fr) * 2019-08-21 2021-02-25 The Scripps Research Institute Agonistes bicycliques du simulateur de gènes d'interféron (sting)
RU2800072C1 (ru) * 2019-08-21 2023-07-17 Зе Скриппс Рисерч Инститьют Бициклические агонисты стимулятора генов интерферона sting

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2006471A1 (de) * 1969-02-13 1970-08-27 Uniroyal, Inc., New York, N.Y.(V. St.A.); Uniroyal, Ltd., Montreal, Quebec (Kanada) Schädlingsbekämpfungsmittel
US3725427A (en) * 1966-12-07 1973-04-03 Uniroyal Ltd Certain 2,4-dimethyl-5-carboxamido-thiazoles
EP0279239A1 (fr) * 1987-01-30 1988-08-24 Ciba-Geigy Ag Agents microbicides
WO1992017479A1 (fr) * 1991-04-08 1992-10-15 Zeneca Ltd. Derives antibiotiques de carbapenem

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3725427A (en) * 1966-12-07 1973-04-03 Uniroyal Ltd Certain 2,4-dimethyl-5-carboxamido-thiazoles
DE2006471A1 (de) * 1969-02-13 1970-08-27 Uniroyal, Inc., New York, N.Y.(V. St.A.); Uniroyal, Ltd., Montreal, Quebec (Kanada) Schädlingsbekämpfungsmittel
EP0279239A1 (fr) * 1987-01-30 1988-08-24 Ciba-Geigy Ag Agents microbicides
WO1992017479A1 (fr) * 1991-04-08 1992-10-15 Zeneca Ltd. Derives antibiotiques de carbapenem

Non-Patent Citations (20)

* Cited by examiner, † Cited by third party
Title
CHEMICAL ABSTRACTS, vol. 087, no. 17, 24 October 1977, Columbus, Ohio, US; abstract no. 135197, ARYA V P ET AL: "Antihypertensive agents: Part IV. Synthesis and hypotensive activity of certain 2-substituted 4,5-dihydroimidazoles" *
CHEMICAL ABSTRACTS, vol. 115, no. 23, 9 December 1991, Columbus, Ohio, US; abstract no. 256589, BELOKON Y N ET AL: "A novel application of the chiral reagent (S)-N-(N'-benzylprolyl)am inobenzaldehyde - synthesis of.alpha.-methylvaline and.alpha.-methylglutamic acid in optically pure form" *
CHEMICAL ABSTRACTS, vol. 119, no. 19, 8 November 1993, Columbus, Ohio, US; abstract no. 195098u, YONG WHAN KIM ET AL.: "Quantitative structure-activity relationship of N-substituted phenyl-5-chloro-1,3-dimethylpyrazol-4-carboxamides" page 21; column 1; *
CHEMICAL ABSTRACTS, vol. 121, no. 19, 7 November 1994, Columbus, Ohio, US; abstract no. 230435s, JUNG SUL MOON ET AL.: "Synthesis of N-substituted 5-hydroxyanthranilic acid." page 1058; column 1; *
CHEMICAL ABSTRACTS, vol. 121, no. 21, 21 November 1994, Columbus, Ohio, US; abstract no. 255694, RAJENDRAN S P ET AL: "Synthesis and utilization of 3-(2'-hydroxyethyl)quinolin-2(1H)-ones. Part-II" *
CHEMICAL ABSTRACTS, vol. 121, no. 23, 5 December 1994, Columbus, Ohio, US; abstract no. 271343, LIM J K ET AL: "Analgesic, anti-inflammatory and antiviral effects of melandrin derivatives" *
CHEMICAL ABSTRACTS, vol. 122, no. 13, 27 March 1995, Columbus, Ohio, US; abstract no. 160414, LEE A R ET AL: "Facile synthesis of N-substituted 2-indolecarboxamides" *
CHEMICAL ABSTRACTS, vol. 122, no. 7, 13 February 1995, Columbus, Ohio, US; abstract no. 080950, LIM J K ET AL: "Synthesis of melandrin derivatives" *
CHIN. PHARM. J. (TAIPEI) (CPHJEP);94; VOL.46 (4); PP.307-11, SCHOOL PHARMACY;NATIONAL DEFENSE MEDICAL CENTER; TAIPEI; TAIWAN (TW) *
HAN'GUK NONGHWA HAKHOECHI, vol. 35, no. 3, pages 382 - 388 *
INDIAN J. CHEM., SECT. B (IJSBDB);77; VOL.15B (2); PP.148-53, CIBA-GEIGY RES. CENT.;BOMBAY; INDIA *
IZV. AKAD. NAUK SSSR, SER. KHIM. (IASKA6,00023353);91; (7); PP.1536-42, INST. ELEMENTOORG. SOEDIN. IM. NESMEYANOVA;MOSCOW; USSR (SU) *
J. INDIAN CHEM. SOC. (JICSAH,00194522);93; VOL.70 (10); PP.815-18, BHARATHIAR UNIV.;DEPT. CHEM.; COIMBATORE; 641 046; INDIA (IN) *
LOONEY-DEAN V ET AL: "Synthesis of derivatives of pyrrole using methyl 2-isothiocyanatobenzoate", SYNTHESIS, no. 1, STUTTGART DE, pages 68 - 71 *
PEET N P: "Reactions of 2-isocyanatobenzoyl chloride and 2-carbomethoxyphenyl isocyanate with 5-aminotetrazole", JOURNAL OF HETEROCYCLIC CHEMISTRY, vol. 24, no. 1, PROVO US, pages 223 - 225 *
SIEMION I Z ET AL: "The amide-aromatic-ring system. An inherently dissymmetric chromophore", TETRAHEDRON, (INCL TETRAHEDRON REPORTS), vol. 33, no. 1, OXFORD GB, pages 155 - 157 *
W. GARY PHILLIPS ET AL.: "Thiazole Carboxanilide Fungicides: ...", PESTICIDE SCIENCE, vol. 38, no. 1, BARKING GB, pages 1 - 7, XP000394080 *
YAKHAK HOECHI (YAHOA3,05134234);94; VOL.38 (3); PP.281-5, SUNG KYUN KWAN UNIVERSITY;COLLEGE OF PHARMACY; SUWON; 440-746; S. KOREA (KR) *
YAKHAK HOECHI (YAHOA3,05134234);94; VOL.38 (3); PP.345-50, SUNG KYUN KWAN UNIV.;COLL. PHARM.; SUWON; 440-746; S. KOREA (KR) *
YAKHAK HOECHI, vol. 37, no. 3, pages 243 - 246 *

Cited By (54)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997030047A1 (fr) * 1996-02-17 1997-08-21 Agrevo Uk Limited 1,2,4 oxadiazoles fongicides et analogues
WO1998018792A1 (fr) * 1996-10-28 1998-05-07 Merck Sharp & Dohme Limited DERIVES DE LA THIENYLCYCLOHEXANONE UTILISES COMME LIGANDS DU SOUS-TYPE α-5 DE RECEPTEUR DU GABA¿A?
US6262103B1 (en) 1996-10-28 2001-07-17 Merck Sharp & Dohme Limited Thienycyclohexanone derivatives as ligands of the GABAA α5 receptor subtype
GB2336588A (en) * 1998-04-23 1999-10-27 Merck Sharp & Dohme Benzo[c]thiophene Derivatives for Enhancing Cognition
US6143773A (en) * 1998-04-23 2000-11-07 Merck Sharp & Dohme Limited Substituted thienobenzisoxazole derivatives for enhancing cognition
US6156787A (en) * 1998-04-23 2000-12-05 Merck Sharp & Dohme Limited Substituted thienlycyclohexanone derivatives for enhancing cognition
US6156761A (en) * 1998-04-23 2000-12-05 Merck Sharpe & Dohme Limited Substituted tetralone derivatives for enhancing cognition
US6395766B1 (en) 1998-06-04 2002-05-28 Merck Sharp & Dohme Limited Tetrahydroindolone derivatives as gabaaalpha5 ligands for enhancing cognition
JP4856312B2 (ja) * 1998-09-16 2012-01-18 バイエル アクチェンゲゼルシャフト イソチアゾールカルボン酸アミド類
JP2002524557A (ja) * 1998-09-16 2002-08-06 バイエル アクチェンゲゼルシャフト イソチアゾールカルボン酸アミド類
WO2001058879A1 (fr) * 2000-02-09 2001-08-16 The Procter & Gamble Company 2-phenylcarbamoyl-benzimidazoles
WO2003016304A1 (fr) * 2001-08-15 2003-02-27 E. I. Du Pont De Nemours And Company Amides aryle ortho-heterocycliques substitues permettant de lutter contre des ravageurs invertebres
US7629463B2 (en) 2001-08-15 2009-12-08 E. I. Du Pont De Nemours And Company Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests
US7375232B2 (en) 2001-08-15 2008-05-20 E.I. Du Pont De Nemours And Company Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests
US7223782B2 (en) * 2001-11-01 2007-05-29 Icagen, Inc. Pyrazole-amides and -sulfonamides
WO2004018448A1 (fr) * 2002-08-13 2004-03-04 Warner-Lambert Company Llc Nouveaux derives de thiophene, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
EP1394159A1 (fr) * 2002-08-13 2004-03-03 Warner-Lambert Company LLC Nouveaux dérivés de thiophène, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent
WO2004018461A2 (fr) * 2002-08-23 2004-03-04 Pharmacia & Upjohn Company Llc Derives d'acide benzoique antibacteriens
WO2004018461A3 (fr) * 2002-08-23 2004-08-26 Upjohn Co Derives d'acide benzoique antibacteriens
US7078419B2 (en) 2003-03-10 2006-07-18 Boehringer Ingelheim Pharmaceuticals, Inc. Cytokine inhibitors
WO2005004606A3 (fr) * 2003-07-10 2005-04-21 Bayer Cropscience Ag Pyridinylanilides
JP2009513514A (ja) * 2003-07-10 2009-04-02 バイエル・クロツプサイエンス・アクチエンゲゼルシヤフト ピリジニルアニリド類
WO2005004606A2 (fr) * 2003-07-10 2005-01-20 Bayer Cropscience Ag Pyridinylanilides
WO2005085234A3 (fr) * 2004-03-03 2006-01-26 Syngenta Participations Ag Nouveaux insecticides
US7812170B2 (en) 2004-03-03 2010-10-12 Syngenta Crop Protection, Inc. Insecticides
CN1926129B (zh) * 2004-03-03 2011-06-15 辛根塔参与股份公司 双酰胺杀虫剂
JP2008517944A (ja) * 2004-10-22 2008-05-29 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Ｃ−ｆｍｓキナーゼの阻害剤
WO2006068618A1 (fr) * 2004-12-23 2006-06-29 Astrazeneca Ab Nouveaux composés
EP1846388A1 (fr) * 2005-01-25 2007-10-24 Synta Pharmaceuticals Corporation Composes de thiophene utilises contre l'inflammation et les troubles lies a l'immunite
US8802721B2 (en) 2005-01-25 2014-08-12 Synta Pharmaceuticals Corp. Thiophene compounds for inflammation and immune-related uses
EP1846388A4 (fr) * 2005-01-25 2011-12-07 Synta Pharmaceuticals Corp Composes de thiophene utilises contre l'inflammation et les troubles lies a l'immunite
US8163746B2 (en) 2006-04-19 2012-04-24 Astellas Pharma Inc. Azolecarboxamide derivative
JP2009535311A (ja) * 2006-04-28 2009-10-01 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト 殺虫化合物
US8252936B2 (en) * 2006-04-28 2012-08-28 Syngenta Crop Protection Llc Insecticidal compounds
JP2013216672A (ja) * 2006-04-28 2013-10-24 Syngenta Participations Ag 殺虫化合物
RU2461551C2 (ru) * 2007-10-24 2012-09-20 Астеллас Фарма Инк. Азолкарбоксамидное соединение или его фармацевтически приемлемая соль
US8304547B2 (en) 2007-10-24 2012-11-06 Astellas Pharma Inc. Azolecarboxamide compound or salt thereof
AU2008314922B2 (en) * 2007-10-24 2013-08-29 Astellas Pharma Inc. Azolecarboxamide compound or salt thereof
JP5321467B2 (ja) * 2007-10-24 2013-10-23 アステラス製薬株式会社 アゾールカルボキサミド化合物又はその塩
TWI418557B (zh) * 2007-10-24 2013-12-11 Astellas Pharma Inc 唑系羧醯胺化合物或其鹽
WO2009054468A1 (fr) * 2007-10-24 2009-04-30 Astellas Pharma Inc. Composé à base d'azolecarboxamide ou son sel
KR101504787B1 (ko) * 2007-10-24 2015-03-20 아스테라스 세이야쿠 가부시키가이샤 아졸카복사마이드 화합물 또는 그 염
WO2010035886A1 (fr) * 2008-09-25 2010-04-01 住友化学株式会社 Composition à usage agricole qui contrôle ou empêche une maladie botanique provoquée par des agents pathogènes de plante
CN104529900A (zh) * 2014-12-31 2015-04-22 南开大学 1-取代-n-取代苯基-5-氨基-1h-吡唑-4-甲酰胺类化合物的杀菌活性
JP2019507141A (ja) * 2016-02-11 2019-03-14 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 有害生物防除剤としての置換２−オキシイミダゾリル−カルボキサミド類
EP3315028A1 (fr) * 2016-10-27 2018-05-02 Kemijski Institut Inhibiteur de nlp proteines comme agent phytopharmaceutiques pour le contrôle d'un agent pathogene vegetal
CN110105347A (zh) * 2019-06-18 2019-08-09 浙江工业大学 一种2-(2-吡啶基)-1,3-恶唑酰胺类衍生物及其制备方法和应用
CN110105347B (zh) * 2019-06-18 2021-01-15 浙江工业大学 一种2-(2-吡啶基)-1,3-恶唑酰胺类衍生物及其制备方法和应用
WO2021035258A1 (fr) * 2019-08-21 2021-02-25 The Scripps Research Institute Agonistes bicycliques du simulateur de gènes d'interféron (sting)
CN115003383A (zh) * 2019-08-21 2022-09-02 斯克里普斯研究学院 干扰素基因刺激物sting的双环激动剂
JP2022545006A (ja) * 2019-08-21 2022-10-24 ザ スクリプス リサーチ インスティテュート インターフェロン遺伝子の刺激因子ｓｔｉｎｇの二環式アゴニスト
RU2800072C1 (ru) * 2019-08-21 2023-07-17 Зе Скриппс Рисерч Инститьют Бициклические агонисты стимулятора генов интерферона sting
CN110693869A (zh) * 2019-10-23 2020-01-17 华南理工大学 2-(甲氨基)苯甲酸甲酯的应用
CN110693869B (zh) * 2019-10-23 2022-05-24 华南理工大学 2-(甲氨基)苯甲酸甲酯的应用

Also Published As

Publication number Publication date
EP0794950A1 (fr) 1997-09-17
IL116234A0 (en) 1996-03-31
AU4302896A (en) 1996-06-19
GB9424379D0 (en) 1995-01-18
ZA9510223B (en) 1996-07-29

Similar Documents

Publication Publication Date Title
WO1996016954A1 (fr) Derives de l'acide anthranilique utiles en tant que fongicides
AU1898195A (en) Anilide derivatives as fungicides
JP2688495B2 (ja) アクリル系殺菌剤
JP4749542B2 (ja) 殺菌剤として有用な２−ピリジルメチルアミン誘導体
WO1997030047A1 (fr) 1,2,4 oxadiazoles fongicides et analogues
KR100675539B1 (ko) Ｎ2-페닐아미딘 유도체
US4310590A (en) 3-Isothiazolones as biocides
EP0982992B1 (fr) Utilisation de thienopyrimidines comme fongicides
EP1204322A1 (fr) Compositions fongicides
EP1179528B1 (fr) Dérivés phénylamidines fongicides
US6166054A (en) Agricultural and horticultural disease controller and a method for controlling the diseases
WO1996017840A1 (fr) Derives d'hydroxyacetamide a substitution heterocyclyle fongicides
WO1997007099A1 (fr) Derives de l'acide alpha-methoxyimino-naphtylacetique ou alpha m ethoxymethylene et leur utilisation comme fongicides
WO1998027080A1 (fr) Chromones utiles en tant que fongicides
WO1997010228A1 (fr) Anilides substitues de l'acide benzoique ou thiobenzoique utilises comme fongicides
GB2305173A (en) N-(heterocyclylmethylene)-2-(carboxy or heterocyclyl)aniline derivatives as fungicides
EP1178037B1 (fr) Dérivés de phénylimidates fongicides
KR100297332B1 (ko) 해충구제제로서의피리딜-1,2,4-티아디아졸
EP0390506A1 (fr) Azoles fongicides
JP2002205979A (ja) 殺菌性フェニルイミン誘導体
EP1178035A1 (fr) Dérivés de phénylimines fongicides
EP0245991A2 (fr) Benzothiazolines comme fongicides
WO1998051673A1 (fr) Nouveaux derives de l'imidazole et du pyrrole utiles comme fongicides
GB2225011A (en) Fungicidal acrylates
MXPA00007713A (en) 2-pyridylmethylamine derivatives useful as fungicides

Legal Events

Date Code Title Description
AK Designated states

Kind code of ref document: A1

Designated state(s): AU BG BR CA CN CZ FI HU JP KR KZ MX NO NZ PL RO RU SD SK UA US

AL Designated countries for regional patents

Kind code of ref document: A1

Designated state(s): KE LS MW SD SZ UG AT BE CH DE DK ES FR GB GR IE IT LU MC NL PT SE BF BJ CF CG CI CM GA GN ML MR NE SN TD TG

DFPE Request for preliminary examination filed prior to expiration of 19th month from priority date (pct application filed before 20040101)
121 Ep: the epo has been informed by wipo that ep was designated in this application
WWE Wipo information: entry into national phase

Ref document number: 1995941681

Country of ref document: EP

WWP Wipo information: published in national office

Ref document number: 1995941681

Country of ref document: EP

WWW Wipo information: withdrawn in national office

Ref document number: 1995941681

Country of ref document: EP