UA91677C2 - Макроциклические соединения как ингибиторы вирусной репликации - Google Patents

Макроциклические соединения как ингибиторы вирусной репликации

Info

Publication number
UA91677C2
UA91677C2 UAA200611368A UAA200611368A UA91677C2 UA 91677 C2 UA91677 C2 UA 91677C2 UA A200611368 A UAA200611368 A UA A200611368A UA A200611368 A UAA200611368 A UA A200611368A UA 91677 C2 UA91677 C2 UA 91677C2
Authority
UA
Ukraine
Prior art keywords
methods
inhibitors
hcv replication
macrocyclic compounds
subject compound
Prior art date
Application number
UAA200611368A
Other languages
English (en)
Russian (ru)
Ukrainian (uk)
Inventor
Лоренс М. Блетт
Стивен М. Венгловски
Стивен В. Эндрюс
Кевин Р. Кондроски
Ютонг Джианг
Эйприл Л. Кеннеди
Джордж Э. Догерти
Джон Э. Джоси
Питер Д. Стенджел
Вуддард Бенджамин Т., (умерший)
Мачендер Р. Маддуру
Original Assignee
Интермюн, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Интермюн, Инк. filed Critical Интермюн, Инк.
Priority claimed from PCT/US2005/010494 external-priority patent/WO2005095403A2/en
Publication of UA91677C2 publication Critical patent/UA91677C2/ru

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
UAA200611368A 2004-03-30 2005-03-29 Макроциклические соединения как ингибиторы вирусной репликации UA91677C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US55816104P 2004-03-30 2004-03-30
PCT/US2005/010494 WO2005095403A2 (en) 2004-03-30 2005-03-29 Macrocyclic compounds as inhibitors of viral replication

Publications (1)

Publication Number Publication Date
UA91677C2 true UA91677C2 (ru) 2010-08-25

Family

ID=37955155

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200611368A UA91677C2 (ru) 2004-03-30 2005-03-29 Макроциклические соединения как ингибиторы вирусной репликации

Country Status (5)

Country Link
CN (1) CN1938311A (es)
CU (1) CU20090112A6 (es)
TN (1) TNSN06308A1 (es)
UA (1) UA91677C2 (es)
ZA (1) ZA200608798B (es)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009034055A1 (en) * 2007-09-10 2009-03-19 Novartis Forschungsstiftung, Zweigniederlassung Method for predicting the response of a subject suffering from a viral infection of the liver to an antiviral therapy
CN103965200B (zh) 2008-09-22 2016-06-08 阵列生物制药公司 作为trk激酶抑制剂的取代的咪唑并[1,2-b]哒嗪化合物
RS57221B2 (sr) 2008-10-22 2020-08-31 Array Biopharma Inc Jedinjenja supstituisanog pirazolo[1,5-]pirimidina kao inhibitori trk kinaze
LT2401272T (lt) 2009-02-27 2017-03-27 Janssen Pharmaceuticals, Inc. Hcv makrociklinio slopiklio amorfinė druska
AR077468A1 (es) 2009-07-09 2011-08-31 Array Biopharma Inc Compuestos de pirazolo (1,5 -a) pirimidina sustituidos como inhibidores de trk- quinasa
CA2774387A1 (en) * 2009-09-28 2011-03-31 F. Hoffmann-La Roche Ltd Novel macrocyclic inhibitors of hepatitis c virus replication
PL2528922T3 (pl) * 2010-01-27 2018-01-31 Ab Pharma Ltd Związki poliheterocykliczne jako inhibitory hcv
RU2735545C2 (ru) 2010-05-20 2020-11-03 Эррэй Биофарма Инк. Макроциклические соединения в качестве ингибиторов киназы trk
GB201116559D0 (en) * 2011-09-26 2011-11-09 Univ Leuven Kath Novel viral replication inhibitors
SG11201703962XA (en) 2014-11-16 2017-06-29 Array Biopharma Inc Crystalline form of (s)-n-(5-((r)-2-(2,5-difluorophenyl)-pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine-1-carboxamide hydrogen sulfate
RU2744852C2 (ru) 2015-10-26 2021-03-16 Локсо Онколоджи, Инк. Точечные мутации в устойчивых к ингибитору trk злокачественных опухолях и связанные с ними способы
CN107043405B (zh) * 2016-02-05 2021-11-19 爱博新药研发(上海)有限公司 多环杂环化合物的晶型、其制备方法、应用及组合物
US10045991B2 (en) 2016-04-04 2018-08-14 Loxo Oncology, Inc. Methods of treating pediatric cancers
KR102400423B1 (ko) 2016-04-04 2022-05-19 록쏘 온콜로지, 인코포레이티드 (s)-n-(5-((r)-2-(2,5-디플루오로페닐)-피롤리딘-1-일)-피라졸로[1,5-a]피리미딘-3-일)-3-하이드록시피롤리딘-1-카복사미드의 액체 제형
LT3800189T (lt) 2016-05-18 2023-10-10 Loxo Oncology, Inc. (s)-n-(5-((r)-2-(2,5-difluorfenil)pirolidin-1-il)pirazolo[1,5-a]pirimidin-3- il)-3-hidroksipirolidin-1-karboksamido gavimas
JOP20190092A1 (ar) 2016-10-26 2019-04-25 Array Biopharma Inc عملية لتحضير مركبات بيرازولو[1، 5-a]بيريميدين وأملاح منها
JOP20190213A1 (ar) 2017-03-16 2019-09-16 Array Biopharma Inc مركبات حلقية ضخمة كمثبطات لكيناز ros1

Also Published As

Publication number Publication date
ZA200608798B (en) 2008-06-25
TNSN06308A1 (en) 2007-12-03
CU20090112A6 (es) 2012-03-15
CN1938311A (zh) 2007-03-28

Similar Documents

Publication Publication Date Title
UA91677C2 (ru) Макроциклические соединения как ингибиторы вирусной репликации
WO2005095403A3 (en) Macrocyclic compounds as inhibitors of viral replication
SG166791A1 (en) Novel macrocyclic inhibitors of hepatitis c virus replication
MY144593A (en) Macrocyclic carboxylic acids and acylsulfonamides as inhibitors of hcv replication
WO2007047146A3 (en) Inhibitors of viral replication
MX2009011867A (es) Nuevos inhibidores macrociclicos de la replicacion del virus de hepatitis c.
WO2008005511A3 (en) Novel inhibitors of hepatitis c virus replication
TN2009000481A1 (en) Novel peptide inhibitors of hepatitis c virus replication
WO2009142842A3 (en) Novel macrocyclic inhibitors of hepatitis c virus replication
WO2006039488A3 (en) Hcv ns3-ns4a protease inhibition
WO2008106058A3 (en) Inhibitors of serine proteases
MX2012003171A (es) Novedosos inhibidores macrociclicos de la replicacion del virus de hepatitis c.
WO2009134616A3 (en) Novel inhibitors of hepatitis c virus replication
TNSN06103A1 (en) Macrocyclic carboxylic acids and acylsulfonamides as inhibitors of hcv replication
TW200611905A (en) Macrocyclic compounds as inhibitors of viral replication
UA95455C2 (ru) Макроциклические ингибиторы репликации вируса гепатита с
UA84579C2 (ru) Макроциклические карбоновые кислоты и ацилсульфонамиды как ингибиторы репликации вируса гепатита с
TN2010000468A1 (en) Novel macrocyclic inhibitors of hepatitis c virus replication