UA91677C2 - Макроциклические соединения как ингибиторы вирусной репликации - Google Patents
Макроциклические соединения как ингибиторы вирусной репликацииInfo
- Publication number
- UA91677C2 UA91677C2 UAA200611368A UAA200611368A UA91677C2 UA 91677 C2 UA91677 C2 UA 91677C2 UA A200611368 A UAA200611368 A UA A200611368A UA A200611368 A UAA200611368 A UA A200611368A UA 91677 C2 UA91677 C2 UA 91677C2
- Authority
- UA
- Ukraine
- Prior art keywords
- methods
- inhibitors
- hcv replication
- macrocyclic compounds
- subject compound
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US55816104P | 2004-03-30 | 2004-03-30 | |
PCT/US2005/010494 WO2005095403A2 (en) | 2004-03-30 | 2005-03-29 | Macrocyclic compounds as inhibitors of viral replication |
Publications (1)
Publication Number | Publication Date |
---|---|
UA91677C2 true UA91677C2 (ru) | 2010-08-25 |
Family
ID=37955155
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA200611368A UA91677C2 (ru) | 2004-03-30 | 2005-03-29 | Макроциклические соединения как ингибиторы вирусной репликации |
Country Status (5)
Country | Link |
---|---|
CN (1) | CN1938311A (es) |
CU (1) | CU20090112A6 (es) |
TN (1) | TNSN06308A1 (es) |
UA (1) | UA91677C2 (es) |
ZA (1) | ZA200608798B (es) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2009034055A1 (en) * | 2007-09-10 | 2009-03-19 | Novartis Forschungsstiftung, Zweigniederlassung | Method for predicting the response of a subject suffering from a viral infection of the liver to an antiviral therapy |
CN103965200B (zh) | 2008-09-22 | 2016-06-08 | 阵列生物制药公司 | 作为trk激酶抑制剂的取代的咪唑并[1,2-b]哒嗪化合物 |
RS57221B2 (sr) | 2008-10-22 | 2020-08-31 | Array Biopharma Inc | Jedinjenja supstituisanog pirazolo[1,5-]pirimidina kao inhibitori trk kinaze |
LT2401272T (lt) | 2009-02-27 | 2017-03-27 | Janssen Pharmaceuticals, Inc. | Hcv makrociklinio slopiklio amorfinė druska |
AR077468A1 (es) | 2009-07-09 | 2011-08-31 | Array Biopharma Inc | Compuestos de pirazolo (1,5 -a) pirimidina sustituidos como inhibidores de trk- quinasa |
CA2774387A1 (en) * | 2009-09-28 | 2011-03-31 | F. Hoffmann-La Roche Ltd | Novel macrocyclic inhibitors of hepatitis c virus replication |
PL2528922T3 (pl) * | 2010-01-27 | 2018-01-31 | Ab Pharma Ltd | Związki poliheterocykliczne jako inhibitory hcv |
RU2735545C2 (ru) | 2010-05-20 | 2020-11-03 | Эррэй Биофарма Инк. | Макроциклические соединения в качестве ингибиторов киназы trk |
GB201116559D0 (en) * | 2011-09-26 | 2011-11-09 | Univ Leuven Kath | Novel viral replication inhibitors |
SG11201703962XA (en) | 2014-11-16 | 2017-06-29 | Array Biopharma Inc | Crystalline form of (s)-n-(5-((r)-2-(2,5-difluorophenyl)-pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine-1-carboxamide hydrogen sulfate |
RU2744852C2 (ru) | 2015-10-26 | 2021-03-16 | Локсо Онколоджи, Инк. | Точечные мутации в устойчивых к ингибитору trk злокачественных опухолях и связанные с ними способы |
CN107043405B (zh) * | 2016-02-05 | 2021-11-19 | 爱博新药研发(上海)有限公司 | 多环杂环化合物的晶型、其制备方法、应用及组合物 |
US10045991B2 (en) | 2016-04-04 | 2018-08-14 | Loxo Oncology, Inc. | Methods of treating pediatric cancers |
KR102400423B1 (ko) | 2016-04-04 | 2022-05-19 | 록쏘 온콜로지, 인코포레이티드 | (s)-n-(5-((r)-2-(2,5-디플루오로페닐)-피롤리딘-1-일)-피라졸로[1,5-a]피리미딘-3-일)-3-하이드록시피롤리딘-1-카복사미드의 액체 제형 |
LT3800189T (lt) | 2016-05-18 | 2023-10-10 | Loxo Oncology, Inc. | (s)-n-(5-((r)-2-(2,5-difluorfenil)pirolidin-1-il)pirazolo[1,5-a]pirimidin-3- il)-3-hidroksipirolidin-1-karboksamido gavimas |
JOP20190092A1 (ar) | 2016-10-26 | 2019-04-25 | Array Biopharma Inc | عملية لتحضير مركبات بيرازولو[1، 5-a]بيريميدين وأملاح منها |
JOP20190213A1 (ar) | 2017-03-16 | 2019-09-16 | Array Biopharma Inc | مركبات حلقية ضخمة كمثبطات لكيناز ros1 |
-
2005
- 2005-03-29 CN CN 200580010503 patent/CN1938311A/zh active Pending
- 2005-03-29 UA UAA200611368A patent/UA91677C2/ru unknown
-
2006
- 2006-09-27 TN TNP2006000308A patent/TNSN06308A1/en unknown
- 2006-10-23 ZA ZA200608798A patent/ZA200608798B/xx unknown
-
2009
- 2009-06-24 CU CU20090112A patent/CU20090112A6/es unknown
Also Published As
Publication number | Publication date |
---|---|
ZA200608798B (en) | 2008-06-25 |
TNSN06308A1 (en) | 2007-12-03 |
CU20090112A6 (es) | 2012-03-15 |
CN1938311A (zh) | 2007-03-28 |
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