UA73104C2 - Erectile dysfunction remedy comprising 3(2h)-pyridazinone derivative - Google Patents
Erectile dysfunction remedy comprising 3(2h)-pyridazinone derivative Download PDFInfo
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- UA73104C2 UA73104C2 UA2001074743A UA2001074743A UA73104C2 UA 73104 C2 UA73104 C2 UA 73104C2 UA 2001074743 A UA2001074743 A UA 2001074743A UA 2001074743 A UA2001074743 A UA 2001074743A UA 73104 C2 UA73104 C2 UA 73104C2
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- alkyl group
- hydrogen atom
- atom
- erectile dysfunction
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- 208000010228 Erectile Dysfunction Diseases 0.000 title claims abstract description 36
- 201000001881 impotence Diseases 0.000 title claims abstract description 36
- AAILEWXSEQLMNI-UHFFFAOYSA-N 1h-pyridazin-6-one Chemical class OC1=CC=CN=N1 AAILEWXSEQLMNI-UHFFFAOYSA-N 0.000 title abstract description 7
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- ZEMPKEQAKRGZGQ-XOQCFJPHSA-N glycerol triricinoleate Natural products CCCCCC[C@@H](O)CC=CCCCCCCCC(=O)OC[C@@H](COC(=O)CCCCCCCC=CC[C@@H](O)CCCCCC)OC(=O)CCCCCCCC=CC[C@H](O)CCCCCC ZEMPKEQAKRGZGQ-XOQCFJPHSA-N 0.000 description 1
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- 125000006124 n-propyl sulfonyl group Chemical group 0.000 description 1
- 125000004706 n-propylthio group Chemical group C(CC)S* 0.000 description 1
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- 239000002504 physiological saline solution Substances 0.000 description 1
- 125000003386 piperidinyl group Chemical group 0.000 description 1
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- 229910052697 platinum Inorganic materials 0.000 description 1
- 239000001267 polyvinylpyrrolidone Substances 0.000 description 1
- 229920000036 polyvinylpyrrolidone Polymers 0.000 description 1
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- 125000002572 propoxy group Chemical group [*]OC([H])([H])C(C([H])([H])[H])([H])[H] 0.000 description 1
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- 150000003180 prostaglandins Chemical class 0.000 description 1
- 125000000719 pyrrolidinyl group Chemical group 0.000 description 1
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- 239000011780 sodium chloride Substances 0.000 description 1
- BTURAGWYSMTVOW-UHFFFAOYSA-M sodium dodecanoate Chemical compound [Na+].CCCCCCCCCCCC([O-])=O BTURAGWYSMTVOW-UHFFFAOYSA-M 0.000 description 1
- 229940082004 sodium laurate Drugs 0.000 description 1
- 229940083618 sodium nitroprusside Drugs 0.000 description 1
- 239000000600 sorbitol Substances 0.000 description 1
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- 239000000126 substance Substances 0.000 description 1
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- HHVIBTZHLRERCL-UHFFFAOYSA-N sulfonyldimethane Chemical compound CS(C)(=O)=O HHVIBTZHLRERCL-UHFFFAOYSA-N 0.000 description 1
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- 125000005931 tert-butyloxycarbonyl group Chemical group [H]C([H])([H])C(OC(*)=O)(C([H])([H])[H])C([H])([H])[H] 0.000 description 1
- RWRDLPDLKQPQOW-UHFFFAOYSA-N tetrahydropyrrole Natural products C1CCNC1 RWRDLPDLKQPQOW-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Reproductive Health (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP34679898 | 1998-12-07 | ||
| PCT/JP1999/006693 WO2000033845A1 (fr) | 1998-12-07 | 1999-11-30 | Agent therapeutique pour le traitement de la dyserection |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA73104C2 true UA73104C2 (en) | 2005-06-15 |
Family
ID=18385894
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UA2001074743A UA73104C2 (en) | 1998-12-07 | 1999-11-30 | Erectile dysfunction remedy comprising 3(2h)-pyridazinone derivative |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP1157694A4 (xx) |
| KR (1) | KR100633869B1 (xx) |
| CN (1) | CN1163230C (xx) |
| AU (1) | AU768825B2 (xx) |
| CA (1) | CA2353956C (xx) |
| CZ (1) | CZ20012020A3 (xx) |
| IL (2) | IL143530A0 (xx) |
| NO (1) | NO321797B1 (xx) |
| NZ (1) | NZ512754A (xx) |
| RU (1) | RU2229885C2 (xx) |
| SK (1) | SK286984B6 (xx) |
| TW (1) | TW585767B (xx) |
| UA (1) | UA73104C2 (xx) |
| WO (1) | WO2000033845A1 (xx) |
| ZA (1) | ZA200105429B (xx) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20070117806A1 (en) * | 2003-12-26 | 2007-05-24 | Nissan Chemical Industries, Ltd. | Neutrophilia inhibitor |
| WO2005074938A1 (ja) * | 2004-02-09 | 2005-08-18 | Nissan Chemical Industries, Ltd. | 血管内膜肥厚抑制薬 |
| RU2536425C2 (ru) * | 2013-01-17 | 2014-12-20 | Общество с ограниченной ответственностью "Фармамед" | Фармацевтическая композиция, содержащая силденафил цитрат, и способ ее приготовления |
| JP6865933B2 (ja) | 2018-02-23 | 2021-04-28 | 株式会社Ｍｅｉｓ Ｔｅｃｈｎｏｌｏｇｙ | 勃起不全治療剤 |
| CN113546049B (zh) * | 2021-04-30 | 2023-03-17 | 贵州汉方药业有限公司 | 一种柔性丸剂药物黏合剂及使用该黏合剂制成的柔性丸剂 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ270130A (en) * | 1993-12-16 | 1995-12-21 | Nihon Nohyaku Co Ltd | Pyridazinone derivatives, preparation and pharmaceutical compositions thereof |
| AU1466395A (en) * | 1994-01-25 | 1995-08-08 | Nissan Chemical Industries Ltd. | Pyridazinone derivative |
| IL112695A (en) * | 1994-02-22 | 1999-04-11 | Green Cross Corp | Pharmaceutical compositions containing pyridazinone derivatives |
| CN1121220C (zh) * | 1996-08-20 | 2003-09-17 | 卫材株式会社 | 稠合哒嗪系化合物的勃起机能不全症治疗剂 |
| TW482675B (en) * | 1997-01-31 | 2002-04-11 | Green Cross Corp | Compositions for oral administration containing pyridazinone compounds technical field of the invention |
| AU8886298A (en) * | 1997-08-28 | 1999-03-22 | Nissan Chemical Industries Ltd. | Neovascularization promoters and neovascularization potentiators |
| AU734734B2 (en) * | 1997-10-28 | 2001-06-21 | Vivus, Inc. | Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction |
-
1999
- 1999-11-30 AU AU14131/00A patent/AU768825B2/en not_active Ceased
- 1999-11-30 UA UA2001074743A patent/UA73104C2/uk unknown
- 1999-11-30 CA CA002353956A patent/CA2353956C/en not_active Expired - Fee Related
- 1999-11-30 CN CNB998141860A patent/CN1163230C/zh not_active Expired - Fee Related
- 1999-11-30 CZ CZ20012020A patent/CZ20012020A3/cs unknown
- 1999-11-30 IL IL14353099A patent/IL143530A0/xx active IP Right Grant
- 1999-11-30 KR KR1020017006978A patent/KR100633869B1/ko not_active IP Right Cessation
- 1999-11-30 EP EP99973258A patent/EP1157694A4/en not_active Withdrawn
- 1999-11-30 NZ NZ512754A patent/NZ512754A/xx not_active IP Right Cessation
- 1999-11-30 WO PCT/JP1999/006693 patent/WO2000033845A1/ja active IP Right Grant
- 1999-11-30 SK SK706-2001A patent/SK286984B6/sk not_active IP Right Cessation
- 1999-11-30 RU RU2001118846/15A patent/RU2229885C2/ru not_active IP Right Cessation
- 1999-12-06 TW TW088121327A patent/TW585767B/zh not_active IP Right Cessation
-
2001
- 2001-05-29 NO NO20012616A patent/NO321797B1/no not_active IP Right Cessation
- 2001-06-03 IL IL143530A patent/IL143530A/en not_active IP Right Cessation
- 2001-07-02 ZA ZA200105429A patent/ZA200105429B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NO20012616D0 (no) | 2001-05-29 |
| NO20012616L (no) | 2001-08-07 |
| AU1413100A (en) | 2000-06-26 |
| CA2353956C (en) | 2008-10-28 |
| IL143530A (en) | 2006-12-31 |
| TW585767B (en) | 2004-05-01 |
| CN1329492A (zh) | 2002-01-02 |
| SK7062001A3 (en) | 2001-11-06 |
| NO321797B1 (no) | 2006-07-03 |
| KR20010081067A (ko) | 2001-08-25 |
| CN1163230C (zh) | 2004-08-25 |
| ZA200105429B (en) | 2002-07-02 |
| EP1157694A4 (en) | 2002-08-28 |
| KR100633869B1 (ko) | 2006-10-16 |
| RU2229885C2 (ru) | 2004-06-10 |
| CZ20012020A3 (cs) | 2001-10-17 |
| CA2353956A1 (en) | 2000-06-15 |
| EP1157694A1 (en) | 2001-11-28 |
| IL143530A0 (en) | 2002-04-21 |
| SK286984B6 (sk) | 2009-08-06 |
| NZ512754A (en) | 2002-10-25 |
| WO2000033845A1 (fr) | 2000-06-15 |
| AU768825B2 (en) | 2004-01-08 |
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