NO321797B1 - Anvendelse av et 3(2H)-pyridazinonderivat for fremstilling av et terapeutisk preparat til behandling av erektil malfunksjon - Google Patents
Anvendelse av et 3(2H)-pyridazinonderivat for fremstilling av et terapeutisk preparat til behandling av erektil malfunksjon Download PDFInfo
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- NO321797B1 NO321797B1 NO20012616A NO20012616A NO321797B1 NO 321797 B1 NO321797 B1 NO 321797B1 NO 20012616 A NO20012616 A NO 20012616A NO 20012616 A NO20012616 A NO 20012616A NO 321797 B1 NO321797 B1 NO 321797B1
- Authority
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- Norway
- Prior art keywords
- group
- pyridazinone
- hydroxy
- compound
- atom
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- 238000002651 drug therapy Methods 0.000 description 1
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- 229910000402 monopotassium phosphate Inorganic materials 0.000 description 1
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- 229920001206 natural gum Polymers 0.000 description 1
- 239000002840 nitric oxide donor Substances 0.000 description 1
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- 235000013855 polyvinylpyrrolidone Nutrition 0.000 description 1
- GNSKLFRGEWLPPA-UHFFFAOYSA-M potassium dihydrogen phosphate Chemical compound [K+].OP(O)([O-])=O GNSKLFRGEWLPPA-UHFFFAOYSA-M 0.000 description 1
- 239000003755 preservative agent Substances 0.000 description 1
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- GMVPRGQOIOIIMI-DWKJAMRDSA-N prostaglandin E1 Chemical compound CCCCC[C@H](O)\C=C\[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(O)=O GMVPRGQOIOIIMI-DWKJAMRDSA-N 0.000 description 1
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- 235000017557 sodium bicarbonate Nutrition 0.000 description 1
- 229910000030 sodium bicarbonate Inorganic materials 0.000 description 1
- 239000011780 sodium chloride Substances 0.000 description 1
- BTURAGWYSMTVOW-UHFFFAOYSA-M sodium dodecanoate Chemical compound [Na+].CCCCCCCCCCCC([O-])=O BTURAGWYSMTVOW-UHFFFAOYSA-M 0.000 description 1
- 229940082004 sodium laurate Drugs 0.000 description 1
- 229940083618 sodium nitroprusside Drugs 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Reproductive Health (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP34679898 | 1998-12-07 | ||
| PCT/JP1999/006693 WO2000033845A1 (fr) | 1998-12-07 | 1999-11-30 | Agent therapeutique pour le traitement de la dyserection |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20012616D0 NO20012616D0 (no) | 2001-05-29 |
| NO20012616L NO20012616L (no) | 2001-08-07 |
| NO321797B1 true NO321797B1 (no) | 2006-07-03 |
Family
ID=18385894
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20012616A NO321797B1 (no) | 1998-12-07 | 2001-05-29 | Anvendelse av et 3(2H)-pyridazinonderivat for fremstilling av et terapeutisk preparat til behandling av erektil malfunksjon |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP1157694A4 (xx) |
| KR (1) | KR100633869B1 (xx) |
| CN (1) | CN1163230C (xx) |
| AU (1) | AU768825B2 (xx) |
| CA (1) | CA2353956C (xx) |
| CZ (1) | CZ20012020A3 (xx) |
| IL (2) | IL143530A0 (xx) |
| NO (1) | NO321797B1 (xx) |
| NZ (1) | NZ512754A (xx) |
| RU (1) | RU2229885C2 (xx) |
| SK (1) | SK286984B6 (xx) |
| TW (1) | TW585767B (xx) |
| UA (1) | UA73104C2 (xx) |
| WO (1) | WO2000033845A1 (xx) |
| ZA (1) | ZA200105429B (xx) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1698339A4 (en) * | 2003-12-26 | 2009-06-17 | Nissan Chemical Ind Ltd | INHIBITOR OF NEUTROPHILY |
| US20070161642A1 (en) * | 2004-02-09 | 2007-07-12 | Nissan Chemical Industries Ltd. | Drug for inhibiting vascular intimal hyperplasia |
| RU2536425C2 (ru) * | 2013-01-17 | 2014-12-20 | Общество с ограниченной ответственностью "Фармамед" | Фармацевтическая композиция, содержащая силденафил цитрат, и способ ее приготовления |
| JP6865933B2 (ja) | 2018-02-23 | 2021-04-28 | 株式会社Ｍｅｉｓ Ｔｅｃｈｎｏｌｏｇｙ | 勃起不全治療剤 |
| CN113546049B (zh) * | 2021-04-30 | 2023-03-17 | 贵州汉方药业有限公司 | 一种柔性丸剂药物黏合剂及使用该黏合剂制成的柔性丸剂 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW326041B (en) * | 1993-12-16 | 1998-02-01 | Nippon Nouyaku Kk | Pyridazinone derivatives, their production process and their use for inhibition of platelet aggregation |
| US5750523A (en) * | 1994-01-25 | 1998-05-12 | Nissan Chemical Industries, Ltd. | Pyridazinone derivatives |
| IL112695A (en) * | 1994-02-22 | 1999-04-11 | Green Cross Corp | Pharmaceutical compositions containing pyridazinone derivatives |
| US6288064B1 (en) * | 1996-08-20 | 2001-09-11 | Eisai Co., Ltd. | Remedy for erection failure comprising fused pyridazine compound |
| TW482675B (en) * | 1997-01-31 | 2002-04-11 | Green Cross Corp | Compositions for oral administration containing pyridazinone compounds technical field of the invention |
| JP4352613B2 (ja) * | 1997-08-28 | 2009-10-28 | 日産化学工業株式会社 | 血管新生促進剤及び血管新生作用増強剤 |
| JP2003525845A (ja) * | 1997-10-28 | 2003-09-02 | ヴィヴァス・インコーポレイテッド | 勃起機能不全の処置のためのホスホジエステラーゼインヒビターの局所投与 |
-
1999
- 1999-11-30 CZ CZ20012020A patent/CZ20012020A3/cs unknown
- 1999-11-30 RU RU2001118846/15A patent/RU2229885C2/ru not_active IP Right Cessation
- 1999-11-30 IL IL14353099A patent/IL143530A0/xx active IP Right Grant
- 1999-11-30 SK SK706-2001A patent/SK286984B6/sk not_active IP Right Cessation
- 1999-11-30 UA UA2001074743A patent/UA73104C2/uk unknown
- 1999-11-30 CN CNB998141860A patent/CN1163230C/zh not_active Expired - Fee Related
- 1999-11-30 AU AU14131/00A patent/AU768825B2/en not_active Ceased
- 1999-11-30 KR KR1020017006978A patent/KR100633869B1/ko not_active IP Right Cessation
- 1999-11-30 WO PCT/JP1999/006693 patent/WO2000033845A1/ja active IP Right Grant
- 1999-11-30 NZ NZ512754A patent/NZ512754A/xx not_active IP Right Cessation
- 1999-11-30 CA CA002353956A patent/CA2353956C/en not_active Expired - Fee Related
- 1999-11-30 EP EP99973258A patent/EP1157694A4/en not_active Withdrawn
- 1999-12-06 TW TW088121327A patent/TW585767B/zh not_active IP Right Cessation
-
2001
- 2001-05-29 NO NO20012616A patent/NO321797B1/no not_active IP Right Cessation
- 2001-06-03 IL IL143530A patent/IL143530A/en not_active IP Right Cessation
- 2001-07-02 ZA ZA200105429A patent/ZA200105429B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR20010081067A (ko) | 2001-08-25 |
| CZ20012020A3 (cs) | 2001-10-17 |
| AU1413100A (en) | 2000-06-26 |
| IL143530A0 (en) | 2002-04-21 |
| IL143530A (en) | 2006-12-31 |
| KR100633869B1 (ko) | 2006-10-16 |
| CA2353956C (en) | 2008-10-28 |
| CA2353956A1 (en) | 2000-06-15 |
| SK7062001A3 (en) | 2001-11-06 |
| AU768825B2 (en) | 2004-01-08 |
| EP1157694A4 (en) | 2002-08-28 |
| RU2229885C2 (ru) | 2004-06-10 |
| CN1163230C (zh) | 2004-08-25 |
| CN1329492A (zh) | 2002-01-02 |
| EP1157694A1 (en) | 2001-11-28 |
| TW585767B (en) | 2004-05-01 |
| ZA200105429B (en) | 2002-07-02 |
| SK286984B6 (sk) | 2009-08-06 |
| UA73104C2 (en) | 2005-06-15 |
| NZ512754A (en) | 2002-10-25 |
| WO2000033845A1 (fr) | 2000-06-15 |
| NO20012616D0 (no) | 2001-05-29 |
| NO20012616L (no) | 2001-08-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM1K | Lapsed by not paying the annual fees |