UA71650C2 - Сполуки з аналгетичною дією, фармацевтична композиція на основі цих сполук та спосіб лікування - Google Patents
Сполуки з аналгетичною дією, фармацевтична композиція на основі цих сполук та спосіб лікування Download PDFInfo
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- UA71650C2 UA71650C2 UA2002064617A UA200264617A UA71650C2 UA 71650 C2 UA71650 C2 UA 71650C2 UA 2002064617 A UA2002064617 A UA 2002064617A UA 200264617 A UA200264617 A UA 200264617A UA 71650 C2 UA71650 C2 UA 71650C2
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pulmonology (AREA)
- Anesthesiology (AREA)
- Psychology (AREA)
- Virology (AREA)
- Urology & Nephrology (AREA)
- Communicable Diseases (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Use Of Switch Circuits For Exchanges And Methods Of Control Of Multiplex Exchanges (AREA)
- Furan Compounds (AREA)
- Valve-Gear Or Valve Arrangements (AREA)
- Liquid Crystal (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE9904674A SE9904674D0 (sv) | 1999-12-20 | 1999-12-20 | Novel compounds |
| PCT/SE2000/002562 WO2001046174A1 (en) | 1999-12-20 | 2000-12-15 | Novel compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA71650C2 true UA71650C2 (uk) | 2004-12-15 |
Family
ID=20418210
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UA2002064617A UA71650C2 (uk) | 1999-12-20 | 2000-12-15 | Сполуки з аналгетичною дією, фармацевтична композиція на основі цих сполук та спосіб лікування |
Country Status (31)
| Country | Link |
|---|---|
| US (2) | US6680318B2 (enExample) |
| EP (1) | EP1242410B1 (enExample) |
| JP (1) | JP2003522741A (enExample) |
| KR (2) | KR20070090050A (enExample) |
| CN (1) | CN1608064A (enExample) |
| AT (1) | ATE275143T1 (enExample) |
| AU (1) | AU780799B2 (enExample) |
| BG (1) | BG65457B1 (enExample) |
| BR (1) | BR0016591A (enExample) |
| CA (1) | CA2395300A1 (enExample) |
| CZ (1) | CZ20022124A3 (enExample) |
| DE (1) | DE60013486T2 (enExample) |
| DK (1) | DK1242410T3 (enExample) |
| EE (1) | EE200200337A (enExample) |
| ES (1) | ES2225289T3 (enExample) |
| HK (1) | HK1048308B (enExample) |
| HU (1) | HUP0300020A3 (enExample) |
| IL (2) | IL150125A0 (enExample) |
| IS (1) | IS2143B (enExample) |
| MX (1) | MXPA02006063A (enExample) |
| NO (1) | NO322432B1 (enExample) |
| NZ (1) | NZ519986A (enExample) |
| PL (1) | PL356780A1 (enExample) |
| PT (1) | PT1242410E (enExample) |
| RU (1) | RU2258703C2 (enExample) |
| SE (1) | SE9904674D0 (enExample) |
| SI (1) | SI1242410T1 (enExample) |
| SK (1) | SK8832002A3 (enExample) |
| UA (1) | UA71650C2 (enExample) |
| WO (1) | WO2001046174A1 (enExample) |
| ZA (1) | ZA200204255B (enExample) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20040067950A1 (en) * | 1998-07-27 | 2004-04-08 | Schering-Plough Corporation | High affinity ligands for nociceptin receptor ORL-1 |
| SE9904674D0 (sv) * | 1999-12-20 | 1999-12-20 | Astra Pharma Inc | Novel compounds |
| NZ539828A (en) * | 2001-05-18 | 2007-01-26 | Astrazeneca Ab | 4 (phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders |
| JP4892654B2 (ja) * | 2001-10-29 | 2012-03-07 | マウント クック ファーマ，インコーポレーテッド | デルタレセプターアゴニスト化合物によるうつ病の治療方法 |
| SE0203303D0 (sv) * | 2002-11-07 | 2002-11-07 | Astrazeneca Ab | Novel Compounds |
| SE0203300D0 (sv) | 2002-11-07 | 2002-11-07 | Astrazeneca Ab | Novel Compounds |
| SE0203302D0 (sv) | 2002-11-07 | 2002-11-07 | Astrazeneca Ab | Novel Compounds |
| SE0301441D0 (sv) * | 2003-05-16 | 2003-05-16 | Astrazeneca Ab | Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof |
| CN1890208A (zh) * | 2003-12-12 | 2007-01-03 | 伊莱利利公司 | 类鸦片受体拮抗剂 |
| SE0400027D0 (sv) * | 2004-01-09 | 2004-01-09 | Astrazeneca Ab | Diarylmethyl piperazine derivatives, preparations thereof and uses thereof |
| SE0401968D0 (sv) * | 2004-08-02 | 2004-08-02 | Astrazeneca Ab | Diarylmethyl piperazine derivatives, preparations thereof and uses thereof |
| KR101234421B1 (ko) | 2004-08-02 | 2013-02-18 | 아스트라제네카 아베 | 디아릴메틸 피페라진 유도체, 이의 제조 방법 및 용도 |
| CN101128447A (zh) * | 2005-02-28 | 2008-02-20 | 阿斯利康(瑞典)有限公司 | 二芳基甲基哌嗪衍生物，其制备及其用途 |
| GB0606876D0 (en) * | 2006-04-05 | 2006-05-17 | Glaxo Group Ltd | Compounds |
| EA201001644A1 (ru) * | 2008-05-20 | 2011-06-30 | Астразенека Аб | Способ лечения тревожного большого депрессивного расстройства |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH585209A5 (enExample) | 1973-06-29 | 1977-02-28 | Cermol Sa | |
| DE2900810A1 (de) | 1979-01-11 | 1980-07-24 | Cassella Ag | Substituierte n-benzhydryl-n'-p- hydroxybenzyl-piperazine und verfahren zu ihrer herstellung |
| IT1140978B (it) | 1980-05-23 | 1986-10-10 | Selvi & C Spa | 1-(4-clorobenzidril)-4-(2,3-diidros sipropil)-piperazina, metodi per la sua preparazione e relative composizione farmaceutiche |
| GB8320701D0 (en) | 1983-08-01 | 1983-09-01 | Wellcome Found | Chemotherapeutic agent |
| IT1196150B (it) | 1984-06-19 | 1988-11-10 | Poli Ind Chimica Spa | Derivati di 1-(bis-(4-fluorofenil)metil)-4-(3-fenil-2-propenil)-esaidro-1h-1,4-diazepina ad attivita' calcio antagonista,sua preparazione e composizioni che lo contengono |
| SE8500573D0 (sv) | 1985-02-08 | 1985-02-08 | Ferrosan Ab | Novel piperazinecarboxamides having a phenoxyalkyl or thiophenoxyalkyl side chain |
| US5028610A (en) | 1987-03-18 | 1991-07-02 | Sankyo Company Limited | N-benzhydryl-substituted heterocyclic derivatives, their preparation and their use |
| US4829065A (en) | 1987-04-24 | 1989-05-09 | Syntex Pharmaceuticals, Ltd. | Substituted imidazolyl-alkyl-piperazine and -diazepine derivatives |
| US4826844A (en) | 1987-09-30 | 1989-05-02 | American Home Products Corporation | Substituted 1-(aralkyl-piperazinoalkyl) cycloalkanols |
| RU2093156C1 (ru) | 1989-11-22 | 1997-10-20 | Жансен Фармасетика Н.В. | L-(-)-2-(аминокарбонил)-n-(4-амино-2,6-дихлорфенил-4[5,5-бис(4-фторфенил)пентил]-1-пиперазинацетамид, его фармацевтически приемлемая кислотно-аддитивная соль или гидрат, способ его получения и средство для хранения сердца донора |
| GB9202238D0 (en) | 1992-02-03 | 1992-03-18 | Wellcome Found | Compounds |
| US5681830A (en) | 1992-02-03 | 1997-10-28 | Delta Pharmaceuticals, Inc. | Opioid compounds |
| US5807858A (en) | 1996-06-05 | 1998-09-15 | Delta Pharmaceutical, Inc. | Compositions and methods for reducing respiratory depression |
| US5574159A (en) | 1992-02-03 | 1996-11-12 | Delta Pharmaceuticals, Inc. | Opioid compounds and methods for making therefor |
| FR2696744B1 (fr) | 1992-10-12 | 1994-12-30 | Logeais Labor Jacques | Dérivés de 2-pyrrolidone, leur procédé de préparation et leurs applications en thérapeutique. |
| DK148292D0 (da) * | 1992-12-09 | 1992-12-09 | Lundbeck & Co As H | Forbindelser |
| WO1995004051A1 (en) | 1993-07-30 | 1995-02-09 | The Wellcome Foundation Limited | Piperazine compounds used in therapy |
| JP3352184B2 (ja) | 1993-11-12 | 2002-12-03 | 株式会社アズウェル | ピペラジン不飽和脂肪酸誘導体 |
| SE9504661D0 (sv) | 1995-12-22 | 1995-12-22 | Astra Pharma Inc | New compounds |
| US5693843A (en) * | 1995-12-22 | 1997-12-02 | E. I. Du Pont De Nemours And Company | Process for hydrocyanation of diolefins and isomerization of nonconjugated 2 alkyl-3-monoalkenenitriles |
| SE9604786D0 (sv) * | 1996-12-20 | 1996-12-20 | Astra Pharma Inc | New compounds |
| TW548271B (en) | 1996-12-20 | 2003-08-21 | Astra Pharma Inc | Novel piperidine derivatives having an exocyclic double bond with analgesic effects |
| CA2316341A1 (en) | 1997-12-24 | 1999-07-08 | Ortho-Mcneil Pharmaceutical, Inc. | 4-[aryl(piperidin-4-yl)] aminobenzamides which bind to the delta-opioid receptor |
| SE9904674D0 (sv) * | 1999-12-20 | 1999-12-20 | Astra Pharma Inc | Novel compounds |
-
1999
- 1999-12-20 SE SE9904674A patent/SE9904674D0/xx unknown
-
2000
- 2000-12-15 UA UA2002064617A patent/UA71650C2/uk unknown
- 2000-12-15 AU AU24184/01A patent/AU780799B2/en not_active Ceased
- 2000-12-15 JP JP2001547084A patent/JP2003522741A/ja not_active Abandoned
- 2000-12-15 WO PCT/SE2000/002562 patent/WO2001046174A1/en not_active Ceased
- 2000-12-15 HK HK03100216.5A patent/HK1048308B/en not_active IP Right Cessation
- 2000-12-15 ES ES00987916T patent/ES2225289T3/es not_active Expired - Lifetime
- 2000-12-15 SK SK883-2002A patent/SK8832002A3/sk unknown
- 2000-12-15 CZ CZ20022124A patent/CZ20022124A3/cs unknown
- 2000-12-15 BR BR0016591-3A patent/BR0016591A/pt not_active Application Discontinuation
- 2000-12-15 DE DE60013486T patent/DE60013486T2/de not_active Expired - Fee Related
- 2000-12-15 KR KR1020077019022A patent/KR20070090050A/ko not_active Ceased
- 2000-12-15 IL IL15012500A patent/IL150125A0/xx active IP Right Grant
- 2000-12-15 EP EP00987916A patent/EP1242410B1/en not_active Expired - Lifetime
- 2000-12-15 AT AT00987916T patent/ATE275143T1/de not_active IP Right Cessation
- 2000-12-15 KR KR1020027007836A patent/KR100769814B1/ko not_active Expired - Fee Related
- 2000-12-15 RU RU2002114343/04A patent/RU2258703C2/ru not_active IP Right Cessation
- 2000-12-15 SI SI200030501T patent/SI1242410T1/xx unknown
- 2000-12-15 NZ NZ519986A patent/NZ519986A/en unknown
- 2000-12-15 CA CA002395300A patent/CA2395300A1/en not_active Abandoned
- 2000-12-15 PL PL00356780A patent/PL356780A1/xx not_active IP Right Cessation
- 2000-12-15 HU HU0300020A patent/HUP0300020A3/hu unknown
- 2000-12-15 US US10/149,981 patent/US6680318B2/en not_active Expired - Fee Related
- 2000-12-15 CN CNA008190461A patent/CN1608064A/zh active Pending
- 2000-12-15 EE EEP200200337A patent/EE200200337A/xx unknown
- 2000-12-15 PT PT00987916T patent/PT1242410E/pt unknown
- 2000-12-15 MX MXPA02006063A patent/MXPA02006063A/es active IP Right Grant
- 2000-12-15 DK DK00987916T patent/DK1242410T3/da active
-
2002
- 2002-05-28 ZA ZA200204255A patent/ZA200204255B/en unknown
- 2002-06-10 BG BG106805A patent/BG65457B1/bg unknown
- 2002-06-10 IL IL150125A patent/IL150125A/en not_active IP Right Cessation
- 2002-06-18 NO NO20022920A patent/NO322432B1/no unknown
- 2002-06-18 IS IS6426A patent/IS2143B/is unknown
-
2003
- 2003-11-17 US US10/714,448 patent/US20040138225A1/en not_active Abandoned
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