TWI453029B - 去氧艾克特卡丁b(deoxyactagardine b), 包含其之醫藥組合物及其製造方法 - Google Patents

去氧艾克特卡丁b(deoxyactagardine b), 包含其之醫藥組合物及其製造方法 Download PDF

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Publication number
TWI453029B
TWI453029B TW099100713A TW99100713A TWI453029B TW I453029 B TWI453029 B TW I453029B TW 099100713 A TW099100713 A TW 099100713A TW 99100713 A TW99100713 A TW 99100713A TW I453029 B TWI453029 B TW I453029B
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TW
Taiwan
Prior art keywords
compound
compounds
pharmaceutical composition
treatment
pharmaceutically acceptable
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Application number
TW099100713A
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English (en)
Chinese (zh)
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TW201029661A (en
Inventor
Sjoerd Nicolaas Wadman
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Novacta Biosystems Ltd
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Publication of TW201029661A publication Critical patent/TW201029661A/zh
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Publication of TWI453029B publication Critical patent/TWI453029B/zh

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50—Cyclic peptides containing at least one abnormal peptide link
    • C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
TW099100713A 2009-01-14 2010-01-12 去氧艾克特卡丁b(deoxyactagardine b), 包含其之醫藥組合物及其製造方法 TWI453029B (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US14449009P 2009-01-14 2009-01-14

Publications (2)

Publication Number Publication Date
TW201029661A TW201029661A (en) 2010-08-16
TWI453029B true TWI453029B (zh) 2014-09-21

Family

ID=42110329

Family Applications (1)

Application Number Title Priority Date Filing Date
TW099100713A TWI453029B (zh) 2009-01-14 2010-01-12 去氧艾克特卡丁b(deoxyactagardine b), 包含其之醫藥組合物及其製造方法

Country Status (22)

Country Link
US (2) US8283371B2 (https=)
EP (1) EP2387580B1 (https=)
JP (1) JP5719312B2 (https=)
KR (1) KR20110119699A (https=)
CN (1) CN102348718B (https=)
AU (1) AU2010205472B2 (https=)
CA (1) CA2749278A1 (https=)
DK (1) DK2387580T3 (https=)
EA (1) EA021683B1 (https=)
ES (1) ES2520165T3 (https=)
HR (1) HRP20141084T1 (https=)
IL (1) IL213927A0 (https=)
MX (1) MX2011007313A (https=)
NZ (1) NZ594011A (https=)
PL (1) PL2387580T3 (https=)
PT (1) PT2387580E (https=)
RS (1) RS53586B1 (https=)
SG (1) SG172944A1 (https=)
SI (1) SI2387580T1 (https=)
TW (1) TWI453029B (https=)
WO (1) WO2010082018A1 (https=)
ZA (1) ZA201104991B (https=)

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GB0600928D0 (en) 2006-01-17 2006-02-22 Novacta Biosystems Ltd Improvements relating to lantibiotics
GB0714029D0 (en) * 2007-07-18 2007-08-29 Novacta Biosystems Ltd Lantibiotic-based compounds having antimicrobial activity
GB0714030D0 (en) * 2007-07-18 2007-08-29 Novacta Biosystems Ltd The use of type-B lantibiotic-based compounds having antimicrobial activity
CA2749278A1 (en) 2009-01-14 2010-07-22 Novacta Biosystems Limited Deoxyactagardine derivatives
CN102388060B (zh) 2009-02-04 2014-09-10 诺瓦克塔生物系统有限公司 阿肽加定衍生物
WO2011061748A1 (en) * 2009-11-19 2011-05-26 Strides Arcolab Limited Rifaximin premix
GB201001688D0 (en) 2010-02-02 2010-03-17 Novacta Biosystems Ltd Compounds
GB201013507D0 (en) * 2010-08-11 2010-09-22 Novacta Biosystems Ltd Compounds
GB201013508D0 (en) * 2010-08-11 2010-09-22 Novacta Biosystems Ltd Compounds
GB201013513D0 (en) * 2010-08-11 2010-09-22 Novacta Biosystems Ltd Formulations
GB201013509D0 (en) * 2010-08-11 2010-09-22 Novacta Biosystems Ltd Compounds
GB201213434D0 (en) 2012-07-27 2012-09-12 Novacta Biosystems Ltd The use of type-B lantibiotic-based compounds having antimicrobial activity

Citations (1)

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WO2007083112A2 (en) * 2006-01-17 2007-07-26 Novacta Biosystems Limited Lantibiotic biosynthetic gene clusters from a. garbadinensis and a. liguriae

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WO2007083112A2 (en) * 2006-01-17 2007-07-26 Novacta Biosystems Limited Lantibiotic biosynthetic gene clusters from a. garbadinensis and a. liguriae

Also Published As

Publication number Publication date
IL213927A0 (en) 2011-07-31
TW201029661A (en) 2010-08-16
JP2012515195A (ja) 2012-07-05
HRP20141084T1 (hr) 2015-02-13
US8283371B2 (en) 2012-10-09
CA2749278A1 (en) 2010-07-22
DK2387580T3 (da) 2014-10-13
SI2387580T1 (sl) 2014-11-28
EA201190071A1 (ru) 2012-06-29
MX2011007313A (es) 2011-08-04
AU2010205472A1 (en) 2011-07-28
NZ594011A (en) 2013-12-20
PT2387580E (pt) 2014-10-30
AU2010205472B2 (en) 2013-03-14
KR20110119699A (ko) 2011-11-02
EP2387580A1 (en) 2011-11-23
RS53586B1 (sr) 2015-02-27
EP2387580B1 (en) 2014-08-13
WO2010082018A1 (en) 2010-07-22
US20120277145A1 (en) 2012-11-01
ZA201104991B (en) 2013-10-31
ES2520165T3 (es) 2014-11-11
US20100179207A1 (en) 2010-07-15
CN102348718A (zh) 2012-02-08
PL2387580T3 (pl) 2015-01-30
JP5719312B2 (ja) 2015-05-13
SG172944A1 (en) 2011-08-29
CN102348718B (zh) 2015-06-03
EA021683B1 (ru) 2015-08-31
US8741945B2 (en) 2014-06-03

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