TW201602128A - Ｃ－糖苷衍生物之製造方法 - Google Patents

Ｃ－糖苷衍生物之製造方法 Download PDF

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Publication number
TW201602128A
TW201602128A TW103125071A TW103125071A TW201602128A TW 201602128 A TW201602128 A TW 201602128A TW 103125071 A TW103125071 A TW 103125071A TW 103125071 A TW103125071 A TW 103125071A TW 201602128 A TW201602128 A TW 201602128A
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TW
Taiwan
Prior art keywords
formula
compound
magnesium
magnesium salt
reaction
Prior art date
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TW103125071A
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English (en)
Chinese (zh)
Inventor
Hiroshi Tomiyama
Masayuki Yokota
Original Assignee
Kotobuki Pharmaceutical Co Ltd
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Publication date
Application filed by Kotobuki Pharmaceutical Co Ltd filed Critical Kotobuki Pharmaceutical Co Ltd
Publication of TW201602128A publication Critical patent/TW201602128A/zh

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TW103125071A 2013-07-24 2014-07-22 Ｃ－糖苷衍生物之製造方法 TW201602128A (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2013153374A JP5646706B2 (ja) 2013-07-24 2013-07-24 Ｃ−グリコシド誘導体の製造方法

Publications (1)

Publication Number Publication Date
TW201602128A true TW201602128A (zh) 2016-01-16

Family

ID=49760574

Family Applications (1)

Application Number Title Priority Date Filing Date
TW103125071A TW201602128A (zh) 2013-07-24 2014-07-22 Ｃ－糖苷衍生物之製造方法

Country Status (3)

Country Link
JP (1) JP5646706B2 (enExample)
TW (1) TW201602128A (enExample)
WO (1) WO2015012110A1 (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9902751B2 (en) 2013-12-30 2018-02-27 Mylan Laboratories Limited Process for the preparation of empagliflozin
CN106188022A (zh) * 2015-04-30 2016-12-07 上海医药工业研究院 伊格列净的制备方法
JP2022028986A (ja) * 2018-12-17 2022-02-17 株式会社トクヤマ Ｃ－アリールヒドロキシグリコキシド誘導体の製造方法
TW202039428A (zh) * 2018-12-17 2020-11-01 日商德山股份有限公司 Ｃ－芳基羥基二醇化物（Ｃ－Ａｒｙｌｈｙｄｒｏｘｙｇｌｙｃｏｘｉｄｅ）衍生物之製造方法
JP7738857B2 (ja) 2020-11-18 2025-09-16 株式会社トクヤマ ケトン誘導体の製造方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2567571T3 (es) * 2003-03-14 2016-04-25 Astellas Pharma Inc. Derivados de C-glucósido y sales de los mismos
US8198464B2 (en) * 2006-12-21 2012-06-12 Astellas Pharma Inc. Method for producing C-glycoside derivative and intermediate for synthesis thereof
US7879807B2 (en) * 2007-02-21 2011-02-01 Boehringer Ingelheim International Gmbh Tetrasubstituted glucopyranosylated benzene derivatives, medicaments containing such compounds, their use and process for their manufacture
AR072511A1 (es) * 2008-07-15 2010-09-01 Theracos Inc Derivados deuterados de bencilbenceno y metodos de uso. composicion farmaceutica.

Also Published As

Publication number Publication date
JP5646706B2 (ja) 2014-12-24
JP2013234194A (ja) 2013-11-21
WO2015012110A1 (ja) 2015-01-29

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