TW200825089A - 2-phenoxy pyrimidinone analogues - Google Patents
2-phenoxy pyrimidinone analogues Download PDFInfo
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- TW200825089A TW200825089A TW096131019A TW96131019A TW200825089A TW 200825089 A TW200825089 A TW 200825089A TW 096131019 A TW096131019 A TW 096131019A TW 96131019 A TW96131019 A TW 96131019A TW 200825089 A TW200825089 A TW 200825089A
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- alkyl
- hydrate
- pain
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| EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
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| US10278942B2 (en) | 2015-03-11 | 2019-05-07 | Peloton Therapeutics, Inc. | Compositions for use in treating pulmonary arterial hypertension |
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| US20040242566A1 (en) | 2003-03-25 | 2004-12-02 | Syrrx, Inc. | Dipeptidyl peptidase inhibitors |
| GB0326633D0 (en) | 2003-11-14 | 2003-12-17 | Merck Sharp & Dohme | Therapeutic agents |
| AU2004290626A1 (en) * | 2003-11-14 | 2005-06-02 | Merck Sharp & Dohme Limited | Bicyclic pyrimidin-4-(3H)-ones and analogues and derivatives thereof which modulate the function of the vanilloid-1 receptor (VR1) |
| US7544803B2 (en) * | 2004-01-23 | 2009-06-09 | Amgen Inc. | Vanilloid receptor ligands and their use in treatments |
| GB0412769D0 (en) | 2004-06-08 | 2004-07-07 | Novartis Ag | Organic compounds |
| AR051596A1 (es) * | 2004-10-26 | 2007-01-24 | Irm Llc | Compuestos heterociclicos condensados nitrogenados como inhibidores de la actividad del receptor canabinoide 1; composiciones farmaceuticas que los contienen y su empleo en la preparacion de medicamentos para el tratamiento de trastornos alimentarios |
| GB0509573D0 (en) | 2005-05-11 | 2005-06-15 | Merck Sharp & Dohme | Therapeutic compounds |
| WO2006122200A1 (en) | 2005-05-11 | 2006-11-16 | Merck Sharp & Dohme Limited | 2,3-substituted fused bicyclic pyrimidin-4(3h)-ones modulating the function of the vanilloid-1 receptor (vr1) |
| CN1318429C (zh) * | 2005-07-25 | 2007-05-30 | 华中师范大学 | 具有杀菌活性的取代噻吩并[3',2':5,6]吡啶并[4,3－d]嘧啶－4(3H)－酮及制备 |
| AU2006311883A1 (en) | 2005-11-04 | 2007-05-18 | Hydra Biosciences, Inc. | Compounds for modulating TRPV3 function |
| AU2007288203B2 (en) | 2006-08-23 | 2013-01-17 | Neurogen Corporation | 2-phenoxy pyrimidinone analogues |
| EP2061470A4 (en) | 2006-08-23 | 2010-10-06 | Neurogen Corp | HALOALKYL-SUBSTITUTED PYRIMIDINONE DERIVATIVES |
| CA2668579A1 (en) | 2006-11-06 | 2008-06-05 | Neurogen Corporation | Cis-cyclohexyl substituted pyrimidinone derivatives |
| WO2008156607A1 (en) | 2007-06-12 | 2008-12-24 | Neurogen Corporation | Substituted pyrimidinones |
| WO2009100403A1 (en) | 2008-02-07 | 2009-08-13 | Neurogen Corporation | Substituted aryl pyrimidinones |
| WO2009121036A2 (en) | 2008-03-27 | 2009-10-01 | Neurogen Corporation | Substituted aryl pyrimidinone derivatives |
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2007
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- 2007-08-22 CN CN201410468406.2A patent/CN104292229A/zh active Pending
- 2007-08-22 KR KR1020097005810A patent/KR20090043583A/ko not_active Withdrawn
- 2007-08-22 WO PCT/US2007/018654 patent/WO2008024438A2/en not_active Ceased
- 2007-08-22 JP JP2009525630A patent/JP5421108B2/ja not_active Expired - Fee Related
- 2007-08-22 US US11/895,286 patent/US8003656B2/en active Active
- 2007-08-22 TW TW096131019A patent/TW200825089A/zh unknown
- 2007-08-22 EP EP07811503A patent/EP2061794B1/en active Active
- 2007-08-22 EA EA200900330A patent/EA200900330A1/ru unknown
- 2007-08-22 ES ES07811503T patent/ES2399928T3/es active Active
- 2007-08-22 CN CNA2007800309530A patent/CN101506210A/zh active Pending
- 2007-08-22 MX MX2009002066A patent/MX2009002066A/es unknown
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- 2007-08-22 BR BRPI0716582-0A2A patent/BRPI0716582A2/pt not_active IP Right Cessation
- 2007-08-22 ZA ZA200901163A patent/ZA200901163B/xx unknown
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2009
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- 2009-02-20 SV SV2009003173A patent/SV2009003173A/es not_active Application Discontinuation
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- 2009-03-20 CR CR10675A patent/CR10675A/es not_active Application Discontinuation
- 2009-03-20 NO NO20091182A patent/NO20091182L/no not_active Application Discontinuation
- 2009-03-23 MA MA31732A patent/MA30720B1/fr unknown
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2011
- 2011-08-22 US US13/215,195 patent/US8759361B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| MX2009002066A (es) | 2009-03-06 |
| NI200900023A (es) | 2010-03-05 |
| KR20090043583A (ko) | 2009-05-06 |
| AU2007288203B2 (en) | 2013-01-17 |
| GT200900040A (es) | 2010-03-16 |
| JP2010502576A (ja) | 2010-01-28 |
| CR10675A (es) | 2009-04-17 |
| CN104292229A (zh) | 2015-01-21 |
| CN101506210A (zh) | 2009-08-12 |
| US8003656B2 (en) | 2011-08-23 |
| BRPI0716582A2 (pt) | 2013-10-08 |
| IL197043A0 (en) | 2009-11-18 |
| EP2061794A2 (en) | 2009-05-27 |
| EA200900330A1 (ru) | 2009-08-28 |
| ZA200901163B (en) | 2010-08-25 |
| JP5421108B2 (ja) | 2014-02-19 |
| CA2660957C (en) | 2016-10-11 |
| SV2009003173A (es) | 2010-08-10 |
| WO2008024438A2 (en) | 2008-02-28 |
| MA30720B1 (fr) | 2009-09-01 |
| US20090069347A1 (en) | 2009-03-12 |
| ES2399928T3 (es) | 2013-04-04 |
| EP2061794B1 (en) | 2012-12-05 |
| CA2660957A1 (en) | 2008-02-28 |
| US8759361B2 (en) | 2014-06-24 |
| EP2061794A4 (en) | 2010-09-08 |
| US20120208829A1 (en) | 2012-08-16 |
| AU2007288203A1 (en) | 2008-02-28 |
| WO2008024438A3 (en) | 2008-11-27 |
| CO6150167A2 (es) | 2010-04-20 |
| NO20091182L (no) | 2009-05-14 |
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