MX2009002066A - Analogos de 2-fenoxipirimidinona. - Google Patents
Analogos de 2-fenoxipirimidinona.Info
- Publication number
- MX2009002066A MX2009002066A MX2009002066A MX2009002066A MX2009002066A MX 2009002066 A MX2009002066 A MX 2009002066A MX 2009002066 A MX2009002066 A MX 2009002066A MX 2009002066 A MX2009002066 A MX 2009002066A MX 2009002066 A MX2009002066 A MX 2009002066A
- Authority
- MX
- Mexico
- Prior art keywords
- compound
- alkyl
- fluorophenyl
- purin
- hydrate
- Prior art date
Links
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| GB0509573D0 (en) * | 2005-05-11 | 2005-06-15 | Merck Sharp & Dohme | Therapeutic compounds |
| EA200900330A1 (ru) | 2006-08-23 | 2009-08-28 | Ньюроджен Корпорейшн | Аналоги 2-феноксипиримидинона |
| EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| EP3417851B1 (en) | 2013-09-09 | 2020-07-22 | Peloton Therapeutics, Inc. | Aryl ethers and uses thereof |
| EP3180340B1 (en) * | 2014-08-11 | 2018-10-10 | Hydra Biosciences, Inc. | Pyrido[2,3-d]pyrimidine-2,4(1h,3h)-dione derivatives |
| US10807948B2 (en) | 2015-03-11 | 2020-10-20 | Peloton Therapeutics, Inc. | Aromatic compounds and uses thereof |
| US10512626B2 (en) | 2015-03-11 | 2019-12-24 | Peloton Therapeautics, Inc. | Compositions for use in treating glioblastoma |
| EP3268362B1 (en) | 2015-03-11 | 2021-10-20 | Peloton Therapeutics, Inc. | Substituted pyridines and uses thereof |
| WO2016145032A1 (en) | 2015-03-11 | 2016-09-15 | Peloton Therapeutics, Inc. | Compositions for use in treating pulmonary arterial hypertension |
| US10335388B2 (en) | 2015-04-17 | 2019-07-02 | Peloton Therapeutics, Inc. | Combination therapy of a HIF-2-alpha inhibitor and an immunotherapeutic agent and uses thereof |
| WO2020146449A1 (en) * | 2019-01-08 | 2020-07-16 | Texas Tech University System | Small molecule analogs of the protein e4orf1 in the treatment and prevention of metabolic disorders |
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| EP0364598A4 (en) * | 1988-03-02 | 1992-01-15 | Yoshitomi Pharmaceutical Industries, Ltd. | 3,4-dihydrothieno 2,3-d¨pyrimidine compounds and pharmaceutical application thereof |
| US5202328A (en) * | 1991-03-06 | 1993-04-13 | Merck & Co., Inc. | Substituted fused pyrimidinones |
| ES2184960T3 (es) * | 1996-05-15 | 2003-04-16 | Pfizer | Nuevas pirimidin-4-onas-(5,6)-heteroaril condensadas 2,3 disustituidas. |
| CA2288735A1 (en) | 1997-05-08 | 1998-11-12 | Agrevo Uk Limited | Fungicides |
| US6627755B1 (en) * | 1997-06-09 | 2003-09-30 | Pfizer Inc | Quinazolin-4-one AMPA antagonists |
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| CN1318429C (zh) * | 2005-07-25 | 2007-05-30 | 华中师范大学 | 具有杀菌活性的取代噻吩并[3',2':5,6]吡啶并[4,3－d]嘧啶－4(3H)－酮及制备 |
| US20100152209A1 (en) | 2005-11-04 | 2010-06-17 | Hydra Biosciences Inc. | Compounds for Modulating TRPV3 Function |
| US20080090845A1 (en) * | 2006-08-23 | 2008-04-17 | Neurogen Corporation | Haloalkyl-substituted pyrimidinone derivatives |
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| EP2061794A4 (en) | 2010-09-08 |
| JP5421108B2 (ja) | 2014-02-19 |
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| AU2007288203B2 (en) | 2013-01-17 |
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| CA2660957C (en) | 2016-10-11 |
| ES2399928T3 (es) | 2013-04-04 |
| KR20090043583A (ko) | 2009-05-06 |
| WO2008024438A2 (en) | 2008-02-28 |
| BRPI0716582A2 (pt) | 2013-10-08 |
| EP2061794A2 (en) | 2009-05-27 |
| NI200900023A (es) | 2010-03-05 |
| US20120208829A1 (en) | 2012-08-16 |
| EP2061794B1 (en) | 2012-12-05 |
| AU2007288203A1 (en) | 2008-02-28 |
| CO6150167A2 (es) | 2010-04-20 |
| MA30720B1 (fr) | 2009-09-01 |
| JP2010502576A (ja) | 2010-01-28 |
| SV2009003173A (es) | 2010-08-10 |
| CN104292229A (zh) | 2015-01-21 |
| EA200900330A1 (ru) | 2009-08-28 |
| US20090069347A1 (en) | 2009-03-12 |
| CR10675A (es) | 2009-04-17 |
| NO20091182L (no) | 2009-05-14 |
| ZA200901163B (en) | 2010-08-25 |
| TW200825089A (en) | 2008-06-16 |
| CN101506210A (zh) | 2009-08-12 |
| CA2660957A1 (en) | 2008-02-28 |
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