TW200539867A - Human g protein-coupled receptor and modulators thereof for the treatment of hyperglycemia and related disorders - Google Patents
Human g protein-coupled receptor and modulators thereof for the treatment of hyperglycemia and related disorders Download PDFInfo
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- TW200539867A TW200539867A TW094111561A TW94111561A TW200539867A TW 200539867 A TW200539867 A TW 200539867A TW 094111561 A TW094111561 A TW 094111561A TW 94111561 A TW94111561 A TW 94111561A TW 200539867 A TW200539867 A TW 200539867A
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- G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
- G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
- G01N33/74—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving hormones or other non-cytokine intercellular protein regulatory factors such as growth factors, including receptors to hormones and growth factors
- G01N33/76—Human chorionic gonadotropin including luteinising hormone, follicle stimulating hormone, thyroid stimulating hormone or their receptors
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N2333/00—Assays involving biological materials from specific organisms or of a specific nature
- G01N2333/435—Assays involving biological materials from specific organisms or of a specific nature from animals; from humans
- G01N2333/705—Assays involving receptors, cell surface antigens or cell surface determinants
- G01N2333/72—Assays involving receptors, cell surface antigens or cell surface determinants for hormones
- G01N2333/726—G protein coupled receptor, e.g. TSHR-thyrotropin-receptor, LH/hCG receptor, FSH
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- Health & Medical Sciences (AREA)
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- Life Sciences & Earth Sciences (AREA)
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- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
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- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
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- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Hematology (AREA)
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- Endocrinology (AREA)
- Cardiology (AREA)
- Molecular Biology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Immunology (AREA)
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- Epidemiology (AREA)
- Physics & Mathematics (AREA)
- General Physics & Mathematics (AREA)
- Reproductive Health (AREA)
- Cell Biology (AREA)
- Pathology (AREA)
- Emergency Medicine (AREA)
- Biochemistry (AREA)
- Microbiology (AREA)
- Food Science & Technology (AREA)
- Biotechnology (AREA)
- Analytical Chemistry (AREA)
- Vascular Medicine (AREA)
- Ophthalmology & Optometry (AREA)
- Neurosurgery (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US56195404P | 2004-04-13 | 2004-04-13 |
Publications (1)
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|---|---|
| TW200539867A true TW200539867A (en) | 2005-12-16 |
Family
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| TW094111561A TW200539867A (en) | 2004-04-13 | 2005-04-12 | Human g protein-coupled receptor and modulators thereof for the treatment of hyperglycemia and related disorders |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20080306114A1 (https=) |
| EP (1) | EP1735622A2 (https=) |
| JP (4) | JP2007532135A (https=) |
| CN (1) | CN101027560A (https=) |
| AU (1) | AU2005248722A1 (https=) |
| CA (1) | CA2564139A1 (https=) |
| TW (1) | TW200539867A (https=) |
| WO (1) | WO2005116653A2 (https=) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
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| WO2005023253A1 (en) | 2003-09-05 | 2005-03-17 | Altana Pharma Ag | Use of pde4 inhibitors for the treatment of diabetes mellitus |
| WO2006094942A1 (en) * | 2005-03-08 | 2006-09-14 | Nycomed Gmbh | Roflumilast for the treatment of diabetes mellitus |
| AU2006222060B2 (en) | 2005-03-08 | 2011-09-01 | Takeda Gmbh | Roflumilast for the treatment of diabetes mellitus |
| TW200738701A (en) | 2005-07-26 | 2007-10-16 | Du Pont | Fungicidal carboxamides |
| WO2007100618A2 (en) * | 2006-02-23 | 2007-09-07 | Atto Bioscience | Novel cell-based phosphodiesterase assays |
| WO2007115805A2 (en) * | 2006-04-05 | 2007-10-18 | European Molecular Biology Laboratory (Embl) | Aurora kinase inhibitors |
| WO2008013622A2 (en) | 2006-07-27 | 2008-01-31 | E. I. Du Pont De Nemours And Company | Fungicidal azocyclic amides |
| US9090604B2 (en) | 2006-07-27 | 2015-07-28 | E I Du Pont De Nemours And Company | Fungicidal azocyclic amides |
| US7638541B2 (en) | 2006-12-28 | 2009-12-29 | Metabolex Inc. | 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine |
| JP5337711B2 (ja) | 2007-01-25 | 2013-11-06 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | 殺菌性アミド |
| AU2008279447A1 (en) | 2007-07-19 | 2009-01-29 | Metabolex, Inc. | N-azacyclic substituted pyrrole, pyrazole, imidazole, triazole and tetrazole derivatives as agonists of the RUP3 or GPR119 receptor for the treatment of diabetes and metabolic disorders |
| DE102007047735A1 (de) * | 2007-10-05 | 2009-04-09 | Merck Patent Gmbh | Thiazolderivate |
| TWI428091B (zh) | 2007-10-23 | 2014-03-01 | Du Pont | 殺真菌劑混合物 |
| WO2010117090A1 (en) * | 2009-04-10 | 2010-10-14 | Banyu Pharmaceutical Co.,Ltd. | Novel isoquinolinyloxymethyl heteroaryl derivatives |
| WO2010117084A1 (en) * | 2009-04-10 | 2010-10-14 | Banyu Pharmaceutical Co.,Ltd. | Novel isoquinoline derivatives |
| US8410127B2 (en) | 2009-10-01 | 2013-04-02 | Metabolex, Inc. | Substituted tetrazol-1-yl-phenoxymethyl-thiazol-2-yl-piperidinyl-pyrimidine salts |
| KR20120101019A (ko) | 2009-10-30 | 2012-09-12 | 바이엘 크롭사이언스 아게 | 헤테로아릴피페리딘 및 -피페라진 유도체 |
| US8653047B2 (en) * | 2010-01-08 | 2014-02-18 | Isis Pharmaceuticals, Inc. | Modulation of angiopoietin-like 3 expression |
| AU2017305392A1 (en) | 2016-08-03 | 2019-02-21 | Cymabay Therapeutics, Inc. | Oxymethylene aryl compounds for treating inflammatory gastrointestinal diseases or gastrointestinal conditions |
| CN113082020A (zh) * | 2021-04-08 | 2021-07-09 | 徐州医科大学 | 一种腺苷受体激动剂的增强剂及其应用 |
Family Cites Families (9)
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| US5462856A (en) * | 1990-07-19 | 1995-10-31 | Bunsen Rush Laboratories, Inc. | Methods for identifying chemicals that act as agonists or antagonists for receptors and other proteins involved in signal transduction via pathways that utilize G-proteins |
| US6060465A (en) * | 1997-02-06 | 2000-05-09 | Miljkovic; Dusan | Bile acids and their derivatives as glycoregulatory agents |
| JP2002000281A (ja) | 2000-04-12 | 2002-01-08 | Takeda Chem Ind Ltd | 新規g蛋白質共役型レセプター蛋白質およびそのdna |
| US7198914B2 (en) * | 2000-11-17 | 2007-04-03 | Banyu Pharmaceutical Co., Ltd. | Guanosine triphosphate (GTP)-binding protein-coupled receptor protein, BG37 |
| JP4184697B2 (ja) * | 2001-04-12 | 2008-11-19 | 武田薬品工業株式会社 | スクリーニング方法 |
| US7354726B2 (en) * | 2001-04-12 | 2008-04-08 | Takeda Pharmaceutical Company Limited | Screening method |
| GB0230162D0 (en) * | 2002-12-24 | 2003-02-05 | Metris Therapeutics Ltd | Compounds useful in inhibiting angiogenesis |
| US7625887B2 (en) * | 2003-01-28 | 2009-12-01 | Takeda Pharmaceutical Company Limited | Receptor agonists |
| JP2004346059A (ja) * | 2003-01-28 | 2004-12-09 | Takeda Chem Ind Ltd | 受容体作動薬 |
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2005
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- 2005-04-12 CN CNA2005800187303A patent/CN101027560A/zh not_active Withdrawn
- 2005-04-12 TW TW094111561A patent/TW200539867A/zh unknown
- 2005-04-12 CA CA002564139A patent/CA2564139A1/en not_active Abandoned
- 2005-04-12 EP EP05780020A patent/EP1735622A2/en not_active Withdrawn
- 2005-04-12 US US11/578,257 patent/US20080306114A1/en not_active Abandoned
- 2005-04-12 AU AU2005248722A patent/AU2005248722A1/en not_active Withdrawn
- 2005-04-12 JP JP2007508478A patent/JP2007532135A/ja active Pending
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2008
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2011
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2014
- 2014-10-14 JP JP2014209937A patent/JP2015064359A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| CA2564139A1 (en) | 2005-12-08 |
| CN101027560A (zh) | 2007-08-29 |
| JP2007532135A (ja) | 2007-11-15 |
| JP5769361B2 (ja) | 2015-08-26 |
| US20080306114A1 (en) | 2008-12-11 |
| JP2015064359A (ja) | 2015-04-09 |
| JP2012050454A (ja) | 2012-03-15 |
| AU2005248722A1 (en) | 2005-12-08 |
| EP1735622A2 (en) | 2006-12-27 |
| JP2008263979A (ja) | 2008-11-06 |
| WO2005116653A3 (en) | 2006-05-18 |
| WO2005116653A2 (en) | 2005-12-08 |
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