TW200508240A - Amino avermectin monosaccharide derivatives substituted in the 4'-position having pesticidal properties - Google Patents

Amino avermectin monosaccharide derivatives substituted in the 4'-position having pesticidal properties

Info

Publication number
TW200508240A
TW200508240A TW093102006A TW93102006A TW200508240A TW 200508240 A TW200508240 A TW 200508240A TW 093102006 A TW093102006 A TW 093102006A TW 93102006 A TW93102006 A TW 93102006A TW 200508240 A TW200508240 A TW 200508240A
Authority
TW
Taiwan
Prior art keywords
compounds
derivatives substituted
tautomers
instance
pesticidal properties
Prior art date
Application number
TW093102006A
Other languages
English (en)
Chinese (zh)
Inventor
Thomas Pitterna
Peter Maienfisch
Kessabi Fiona Murphy
Hans Tobler
Jerome Cassayre
Laura Quaranta
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of TW200508240A publication Critical patent/TW200508240A/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
TW093102006A 2003-01-31 2004-01-29 Amino avermectin monosaccharide derivatives substituted in the 4'-position having pesticidal properties TW200508240A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0302309.0A GB0302309D0 (en) 2003-01-31 2003-01-31 Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties

Publications (1)

Publication Number Publication Date
TW200508240A true TW200508240A (en) 2005-03-01

Family

ID=9952240

Family Applications (1)

Application Number Title Priority Date Filing Date
TW093102006A TW200508240A (en) 2003-01-31 2004-01-29 Amino avermectin monosaccharide derivatives substituted in the 4'-position having pesticidal properties

Country Status (28)

Country Link
US (1) US20060205595A1 (enExample)
EP (1) EP1594878B1 (enExample)
JP (1) JP2006518347A (enExample)
KR (1) KR20050097524A (enExample)
CN (1) CN100410259C (enExample)
AR (1) AR042967A1 (enExample)
AT (1) ATE397610T1 (enExample)
AU (1) AU2004207073B2 (enExample)
BR (1) BRPI0406875B1 (enExample)
CA (1) CA2513573C (enExample)
CL (1) CL2004000147A1 (enExample)
CY (1) CY1108295T1 (enExample)
DE (1) DE602004014252D1 (enExample)
DK (1) DK1594878T3 (enExample)
ES (1) ES2308140T3 (enExample)
GB (1) GB0302309D0 (enExample)
IL (1) IL169598A (enExample)
MA (1) MA27587A1 (enExample)
MX (1) MXPA05007923A (enExample)
NZ (1) NZ541252A (enExample)
PL (1) PL218731B1 (enExample)
PT (1) PT1594878E (enExample)
RU (1) RU2329268C2 (enExample)
SI (1) SI1594878T1 (enExample)
TW (1) TW200508240A (enExample)
UA (1) UA81012C2 (enExample)
WO (1) WO2004067534A1 (enExample)
ZA (1) ZA200505545B (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EG23124A (en) 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
CR6574A (es) * 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
AR036486A1 (es) 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
AR040073A1 (es) 2002-05-07 2005-03-16 Syngenta Participations Ag Derivados de 4''-desoxi-4''-(s)-amido avermectina y su uso como plaguicidas
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302310D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302547D0 (en) * 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
GB0320176D0 (en) 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively
US8551914B2 (en) * 2010-08-26 2013-10-08 Dow Agrosciences, Llc. Pesticidal compositions
CN103214532B (zh) * 2013-02-28 2018-07-06 河北威远生物化工有限公司 阿维菌素B2a/2b胺基衍生物、衍生物盐和阿维菌素B2a/2b胺基衍生物盐的制备方法及用途
CN103613625B (zh) * 2013-12-02 2016-03-02 兰州大学 一种阿维菌素类化合物及其制备方法和在农药中的用途
CN104402953B (zh) * 2014-11-28 2017-07-28 大庆志飞生物化工有限公司 阿维菌素单糖化合物及其制备方法和用途
CN104402954A (zh) * 2014-11-28 2015-03-11 大庆志飞生物化工有限公司 甲胺基阿维菌素单糖化合物及其制备方法和用途
CN107501368B (zh) * 2017-09-30 2020-02-21 中国科学院成都生物研究所 一种多拉菌素衍生物的合成及其杀虫应用
CN108690108B (zh) * 2018-07-27 2022-03-11 河北威远生物化工有限公司 一种磺酰胺基取代的阿维菌素B2a/B2b衍生物及其制备方法与应用
CN113150053B (zh) * 2020-01-22 2024-10-01 华东理工大学 偶氮苯类阿维菌素衍生物及其制备方法和应用

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Publication number Priority date Publication date Assignee Title
US4206205A (en) * 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
US4203976A (en) * 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4427663A (en) * 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4622313A (en) * 1985-08-01 1986-11-11 Merck & Co., Inc. O-sulfate derivatives of avermectins and milbemycins having improved water solubility
US4886828A (en) * 1986-09-12 1989-12-12 American Cyanamid Company Δ22 -derivatives of LL-F28249 compounds
US4831016A (en) * 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives
US4895837A (en) * 1988-01-29 1990-01-23 Merck & Co., Inc. Avermectin derivatives
NZ228866A (en) * 1988-05-02 1991-10-25 Merck & Co Inc Fluoro-substituted milbemycins and avermectins for combatting parasites and insects
US5008250A (en) * 1988-05-25 1991-04-16 Merck & Co., Inc. Avermectins with a cleaved furan ring and an 8a hydroxy group
GB2220856A (en) * 1988-07-18 1990-01-24 Merck & Co Inc Novel synergistic agricultural insecticidal and acaricidal combinations containing avermectin derivatives
NZ231773A (en) * 1988-12-23 1992-09-25 Merck & Co Inc Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof
FR2646237B1 (fr) * 1989-04-21 1994-01-07 Fabrication Instruments Mesure Dispositif de jaugeage de gaz haute pression, en particulier pour la reserve d'oxygene gazeux embarquee a bord d'un avion
US5057499A (en) * 1989-06-02 1991-10-15 Merck & Co. Inc. Avermectin derivatives
US5023241A (en) * 1989-07-31 1991-06-11 Merck & Co., Inc. Avermectin derivatives
US5169839A (en) * 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
US5192546A (en) * 1991-01-15 1993-03-09 Mycogen Corporation Synergistic pesticidal compositions
US5346698A (en) * 1991-01-15 1994-09-13 Mycogen Corporation Synergistic pesticidal compositions
US5208222A (en) * 1991-03-28 1993-05-04 Merck & Co., Inc. 4"-and 4'-alkylthio avermectin derivatives
GB9201505D0 (en) * 1992-01-24 1992-03-11 Pfizer Ltd Antiparasitic agents
US5229415A (en) * 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
US5362863A (en) * 1993-09-29 1994-11-08 Merck & Co., Inc. Process for the preparation of 4"-amino avermectin compounds
US5981500A (en) * 1994-01-12 1999-11-09 Pfizer Inc. Antiparasitic agents related to the milbemycins and avermectins
US5436355A (en) * 1994-02-03 1995-07-25 Merck & Co., Inc. Process for making avermectin/zein compositions
TW327125B (en) * 1994-02-07 1998-02-21 Merck & Co Inc Composition and method for protecting against pine exhausted
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US6605595B1 (en) * 1999-02-09 2003-08-12 The Kitasato Institute Avermectin derivatives
WO2002012248A1 (en) * 2000-08-09 2002-02-14 The Kitasato Institute Avermectin derivatives
CR6574A (es) * 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) * 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR037938A1 (es) * 2001-12-21 2004-12-22 Syngenta Participations Ag Derivados de avermectina b1 que tienen un substituyente de aminosulfoniloxilo en la posicion 4''
GB0302308D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302548D0 (en) * 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins substituted in the 4"- and 4' -positions having pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively

Also Published As

Publication number Publication date
US20060205595A1 (en) 2006-09-14
AR042967A1 (es) 2005-07-13
RU2005127321A (ru) 2006-01-27
BRPI0406875A (pt) 2006-01-03
CA2513573A1 (en) 2004-08-12
CA2513573C (en) 2012-03-27
BRPI0406875B1 (pt) 2014-05-27
PT1594878E (pt) 2008-09-10
PL378024A1 (pl) 2006-02-20
CY1108295T1 (el) 2014-02-12
EP1594878A1 (en) 2005-11-16
RU2329268C2 (ru) 2008-07-20
ATE397610T1 (de) 2008-06-15
IL169598A0 (en) 2007-07-04
KR20050097524A (ko) 2005-10-07
EP1594878B1 (en) 2008-06-04
CL2004000147A1 (es) 2005-03-04
CN100410259C (zh) 2008-08-13
AU2004207073B2 (en) 2010-09-16
CN1751049A (zh) 2006-03-22
AU2004207073A1 (en) 2004-08-12
MA27587A1 (fr) 2005-10-03
ZA200505545B (en) 2006-04-26
DK1594878T3 (da) 2008-10-06
SI1594878T1 (sl) 2008-10-31
NZ541252A (en) 2008-05-30
JP2006518347A (ja) 2006-08-10
MXPA05007923A (es) 2005-09-30
WO2004067534A1 (en) 2004-08-12
DE602004014252D1 (de) 2008-07-17
GB0302309D0 (en) 2003-03-05
PL218731B1 (pl) 2015-01-30
IL169598A (en) 2010-05-17
UA81012C2 (en) 2007-11-26
ES2308140T3 (es) 2008-12-01

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