TR201903492T4 - Apomorfin ve organik asitler içeren bileşimler ve bunların kullanım alanları. - Google Patents

Apomorfin ve organik asitler içeren bileşimler ve bunların kullanım alanları. Download PDF

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Publication number
TR201903492T4
TR201903492T4 TR2019/03492T TR201903492T TR201903492T4 TR 201903492 T4 TR201903492 T4 TR 201903492T4 TR 2019/03492 T TR2019/03492 T TR 2019/03492T TR 201903492 T TR201903492 T TR 201903492T TR 201903492 T4 TR201903492 T4 TR 201903492T4
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Prior art keywords
organic acids
compositions containing
apomorphine
containing apomorphine
organic acid
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TR2019/03492T
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English (en)
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Yacoby-Zeevi Oron
Nemas Mara
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Neuroderm Ltd
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Publication of TR201903492T4 publication Critical patent/TR201903492T4/tr

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/473—Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
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    • A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
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    • A61K47/20—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
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    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
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    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone

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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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Abstract

Mevcut buluş, apomorfinin stabil sıvı veya yarı-katı farmasötik bileşimlerini, daha özel olarak, nörolojik veya hareket hastalıklarının veya rahatsızlıklarının, örneğin Parkinson hastalığının veya bununla ilişkili durumların tedavisinde yararlı olan bir organik asit içeren, apomorfin ve organik bir asit bileşimini sağlamaktadır.
TR2019/03492T 2012-06-05 2013-06-05 Apomorfin ve organik asitler içeren bileşimler ve bunların kullanım alanları. TR201903492T4 (tr)

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US201261655633P 2012-06-05 2012-06-05

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TR201903492T4 true TR201903492T4 (tr) 2019-04-22

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TR2019/03492T TR201903492T4 (tr) 2012-06-05 2013-06-05 Apomorfin ve organik asitler içeren bileşimler ve bunların kullanım alanları.

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US (3) US9999674B2 (tr)
EP (2) EP2854764B1 (tr)
JP (2) JP6257604B2 (tr)
CN (2) CN107693486A (tr)
AU (1) AU2013273138B2 (tr)
BR (1) BR112014030265A2 (tr)
CA (1) CA2875446A1 (tr)
DK (1) DK2854764T3 (tr)
ES (1) ES2715028T3 (tr)
HU (1) HUE042425T2 (tr)
MX (1) MX2014014902A (tr)
NZ (1) NZ703341A (tr)
PL (1) PL2854764T3 (tr)
PT (1) PT2854764T (tr)
RU (1) RU2688672C2 (tr)
TR (1) TR201903492T4 (tr)
WO (1) WO2013183055A1 (tr)
ZA (1) ZA201409516B (tr)

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US20180303939A1 (en) 2018-10-25
BR112014030265A2 (pt) 2017-06-27
US10525134B2 (en) 2020-01-07
JP6257604B2 (ja) 2018-01-10
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WO2013183055A1 (en) 2013-12-12
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US9999674B2 (en) 2018-06-19
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