TR201901262T4 - (2S,3R,4R,5S,6R)-2-(4-Kloro-3-(4-Etoksibenzil)Fenil)-6-(Metiltiyo)Tetrahidro-2H-Piran-3,4,5-Triol İçeren Bileşimler - Google Patents
(2S,3R,4R,5S,6R)-2-(4-Kloro-3-(4-Etoksibenzil)Fenil)-6-(Metiltiyo)Tetrahidro-2H-Piran-3,4,5-Triol İçeren Bileşimler Download PDFInfo
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- A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161430027P | 2011-01-05 | 2011-01-05 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR201901262T4 true TR201901262T4 (tr) | 2019-02-21 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2019/01262T TR201901262T4 (tr) | 2011-01-05 | 2012-01-03 | (2S,3R,4R,5S,6R)-2-(4-Kloro-3-(4-Etoksibenzil)Fenil)-6-(Metiltiyo)Tetrahidro-2H-Piran-3,4,5-Triol İçeren Bileşimler |
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Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TR201908247T4 (tr) * | 2012-11-20 | 2019-06-21 | Lexicon Pharmaceuticals Inc | Sodyum glikoz birlikte taşıyıcı 1 inhibitörleri. |
| JP6727419B2 (ja) * | 2016-05-25 | 2020-07-22 | クリスタル ファーマシューティカル（スーチョウ）カンパニー，リミテッド | ナトリウム−グルコース共輸送体阻害薬の新規な結晶形及びその製造方法並びに用途 |
| US11723929B2 (en) | 2017-06-13 | 2023-08-15 | The Regents Of The University Of California | Methods of improving cell-based therapy |
| CN107540685B (zh) * | 2017-09-04 | 2020-05-05 | 杭州科巢生物科技有限公司 | 一种Sotagliflozin的制备方法及其中间体 |
| EP3456320A1 (de) * | 2017-09-15 | 2019-03-20 | Stada Arzneimittel Ag | Dpp-4-inhibitor-mono-zusammensetzung |
| FI3712147T3 (fi) * | 2018-01-05 | 2023-04-04 | Shangdong Danhong Pharmaceutical Co Ltd | Sglts-estäjä ja sen käyttö |
| CN110117304A (zh) * | 2018-04-23 | 2019-08-13 | 中国科学院成都生物研究所 | 一种钠-葡萄糖协同转运蛋白1和2抑制剂的药物用途 |
| CN110818722B (zh) * | 2018-08-14 | 2022-12-02 | 苏州鹏旭医药科技有限公司 | 三种化合物及其制备方法和在合成索格列净中的用途 |
| CN113993865B (zh) | 2019-07-05 | 2023-09-22 | 山东丹红制药有限公司 | 一种SGLTs抑制剂的晶型及其应用 |
| CA3145678C (en) * | 2019-07-26 | 2022-08-23 | Medshine Discovery Inc. | Sglt2/dpp4 inhibitor and application thereof |
| CN114585358B (zh) | 2019-07-26 | 2023-11-10 | 东宝紫星(杭州)生物医药有限公司 | 一种SGLTs/DPP4抑制剂及其应用 |
| EP3771480A1 (en) * | 2019-08-01 | 2021-02-03 | Lexicon Pharmaceuticals, Inc. | Continuous process for preparing the crystalline form ii of sotagliflozin |
| EP4054556A4 (en) * | 2019-11-07 | 2023-11-29 | Increvet, Inc. | SODIUM-GLUCOSE-LINKED TRANSPORTER INHIBITORS FOR THE MANAGEMENT OF CHRONIC KIDNEY DISEASE, HYPERTENSION AND HEART FAILURE IN PETS |
| US20240100013A1 (en) | 2021-01-04 | 2024-03-28 | Lexicon Pharmaceuticals, Inc. | Sotagliflozin for improving left atrial function |
| WO2022155303A1 (en) | 2021-01-14 | 2022-07-21 | Lexicon Pharmaceuticals, Inc. | Sotagliflozin for treating or preventing cardiovascular diseases |
| KR20260083316A (ko) | 2023-09-28 | 2026-06-05 | 렉시컨 파마슈티컬스 인코퍼레이티드 | 제1형 당뇨병 및 신장 질환을 치료하는 방법 |
| US20250114323A1 (en) | 2023-10-06 | 2025-04-10 | Lexicon Pharmaceuticals, Inc. | Methods of reducing the risk of cardiovascular events in patients with left ventricular hypertrophy |
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