TR201809681T4 - N-[(r)-1-[(s)-1-(4-aminometil-benzilkarbamoil)-2-fenil-etilkarbamoil]-2-(4-etoksi-fenil)-etil]-benzamit hidroklorürün polimorfları. - Google Patents
N-[(r)-1-[(s)-1-(4-aminometil-benzilkarbamoil)-2-fenil-etilkarbamoil]-2-(4-etoksi-fenil)-etil]-benzamit hidroklorürün polimorfları. Download PDFInfo
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- TR201809681T4 TR201809681T4 TR2018/09681T TR201809681T TR201809681T4 TR 201809681 T4 TR201809681 T4 TR 201809681T4 TR 2018/09681 T TR2018/09681 T TR 2018/09681T TR 201809681 T TR201809681 T TR 201809681T TR 201809681 T4 TR201809681 T4 TR 201809681T4
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- phenyl
- ethoxy
- solid form
- ethyl
- ethylcarbamoyl
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| US201261668543P | 2012-07-06 | 2012-07-06 | |
| GB201212081A GB201212081D0 (en) | 2012-07-06 | 2012-07-06 | New polymorph |
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| GB2510407A (en) * | 2013-02-04 | 2014-08-06 | Kalvista Pharmaceuticals Ltd | Aqueous suspensions of kallikrein inhibitors for parenteral administration |
| TWI636047B (zh) | 2013-08-14 | 2018-09-21 | 英商卡爾維斯塔製藥有限公司 | 雜環衍生物 |
| GB201421085D0 (en) | 2014-11-27 | 2015-01-14 | Kalvista Pharmaceuticals Ltd | New enzyme inhibitors |
| GB201421083D0 (en) | 2014-11-27 | 2015-01-14 | Kalvista Pharmaceuticals Ltd | Enzyme inhibitors |
| WO2017153567A1 (en) | 2016-03-10 | 2017-09-14 | Thrombogenics Nv | Posterior ocular fibrosis inhibition by antagonizing placental growth factor |
| DK3464271T3 (da) | 2016-05-31 | 2020-06-15 | Kalvista Pharmaceuticals Ltd | Pyrazolderivater som plasma-kallikreininhibitorer |
| GB201609607D0 (en) | 2016-06-01 | 2016-07-13 | Kalvista Pharmaceuticals Ltd | Polymorphs of N-(3-Fluoro-4-methoxypyridin-2-yl)methyl)-3-(methoxymethyl)-1-({4-((2-oxopy ridin-1-yl)methyl)phenyl}methyl)pyrazole-4-carboxamide and salts |
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| PT3716952T (pt) | 2017-11-29 | 2022-04-14 | Kalvista Pharmaceuticals Ltd | Formas de administração que incluem um inibidor de calicreína plasmática |
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| JP7805788B2 (ja) | 2019-05-23 | 2026-01-26 | ヤンセン バイオテツク，インコーポレーテツド | Ｉｌ－２３及びｔｎｆアルファに対する抗体の併用療法による炎症性腸疾患の治療方法 |
| EP4010333A1 (en) | 2019-08-09 | 2022-06-15 | Kalvista Pharmaceuticals Limited | Plasma kallikrein inhibitors |
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| IT1223401B (it) * | 1987-12-02 | 1990-09-19 | Montedison Spa | Poliesteri aromatici liquido cristallini termotropici |
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| IL112795A (en) * | 1994-03-04 | 2001-01-28 | Astrazeneca Ab | Peptide derivatives as antithrombic agents their preparation and pharmaceutical compositions containing them |
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| JP2013121919A (ja) | 2010-03-25 | 2013-06-20 | Astellas Pharma Inc | 血漿カリクレイン阻害剤 |
| WO2012004678A2 (en) | 2010-07-07 | 2012-01-12 | The Medicines Company (Leipzig) Gmbh | Serine protease inhibitors |
| US9290485B2 (en) | 2010-08-04 | 2016-03-22 | Novartis Ag | N-((6-amino-pyridin-3-yl)methyl)-heteroaryl-carboxamides |
| WO2012142308A1 (en) | 2011-04-13 | 2012-10-18 | Activesite Pharmaceuticals, Inc. | Prodrugs of inhibitors of plasma kallikrein |
| GB2494851A (en) | 2011-07-07 | 2013-03-27 | Kalvista Pharmaceuticals Ltd | Plasma kallikrein inhibitors |
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| US9512065B2 (en) | 2016-12-06 |
| WO2014006414A1 (en) | 2014-01-09 |
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| JP2015528798A (ja) | 2015-10-01 |
| HUE039775T2 (hu) | 2019-02-28 |
| EP2870137A1 (en) | 2015-05-13 |
| EP2870137B8 (en) | 2018-07-18 |
| US20150191421A1 (en) | 2015-07-09 |
| EP2870137B1 (en) | 2018-05-16 |
| PL2870137T3 (pl) | 2018-12-31 |
| GB201212081D0 (en) | 2012-08-22 |
| ES2679370T3 (es) | 2018-08-24 |
| CA2878319C (en) | 2021-02-09 |
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