TR201809681T4 - N-[(r)-1-[(s)-1-(4-aminometil-benzilkarbamoil)-2-fenil-etilkarbamoil]-2-(4-etoksi-fenil)-etil]-benzamit hidroklorürün polimorfları. - Google Patents
N-[(r)-1-[(s)-1-(4-aminometil-benzilkarbamoil)-2-fenil-etilkarbamoil]-2-(4-etoksi-fenil)-etil]-benzamit hidroklorürün polimorfları. Download PDFInfo
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- TR201809681T4 TR201809681T4 TR2018/09681T TR201809681T TR201809681T4 TR 201809681 T4 TR201809681 T4 TR 201809681T4 TR 2018/09681 T TR2018/09681 T TR 2018/09681T TR 201809681 T TR201809681 T TR 201809681T TR 201809681 T4 TR201809681 T4 TR 201809681T4
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- phenyl
- ethoxy
- solid form
- ethyl
- ethylcarbamoyl
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| US201261668543P | 2012-07-06 | 2012-07-06 | |
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| TWI636047B (zh) | 2013-08-14 | 2018-09-21 | 英商卡爾維斯塔製藥有限公司 | 雜環衍生物 |
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| GB201421085D0 (en) | 2014-11-27 | 2015-01-14 | Kalvista Pharmaceuticals Ltd | New enzyme inhibitors |
| EP3426685A1 (en) | 2016-03-10 | 2019-01-16 | Oxurion NV | Posterior ocular fibrosis inhibition by antagonizing placental growth factor |
| ME03794B (me) | 2016-05-31 | 2021-04-20 | Kalvista Pharmaceuticals Ltd | Derivati pirazola kao inhibitori kalikreina plazme |
| GB201609603D0 (en) * | 2016-06-01 | 2016-07-13 | Kalvista Pharmaceuticals Ltd | Polymorphs of N-[(6-cyano-2-fluoro-3-methoxyphenyl)Methyl]-3-(methoxymethyl)-1-({4-[(2-ox opyridin-1-YL)Methyl]phenyl}methyl)pyrazole-4-carboxamide |
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| US7453002B2 (en) * | 2004-06-15 | 2008-11-18 | Bristol-Myers Squibb Company | Five-membered heterocycles useful as serine protease inhibitors |
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| JP2013121919A (ja) | 2010-03-25 | 2013-06-20 | Astellas Pharma Inc | 血漿カリクレイン阻害剤 |
| ES2483802T3 (es) | 2010-07-07 | 2014-08-07 | The Medicines Company (Leipzig) Gmbh | Inhibidores de serina proteasa |
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| EP2697196A1 (en) | 2011-04-13 | 2014-02-19 | Activesite Pharmaceuticals, Inc. | Prodrugs of inhibitors of plasma kallikrein |
| GB2494851A (en) * | 2011-07-07 | 2013-03-27 | Kalvista Pharmaceuticals Ltd | Plasma kallikrein inhibitors |
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2012
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- 2013-07-05 US US14/413,086 patent/US9512065B2/en not_active Expired - Fee Related
- 2013-07-05 PL PL13737357T patent/PL2870137T3/pl unknown
- 2013-07-05 HU HUE13737357A patent/HUE039775T2/hu unknown
- 2013-07-05 ES ES13737357.7T patent/ES2679370T3/es active Active
- 2013-07-05 EP EP13737357.7A patent/EP2870137B8/en active Active
- 2013-07-05 CA CA2878319A patent/CA2878319C/en active Active
- 2013-07-05 JP JP2015519357A patent/JP6367187B2/ja not_active Expired - Fee Related
- 2013-07-05 WO PCT/GB2013/051781 patent/WO2014006414A1/en not_active Ceased
- 2013-07-05 TR TR2018/09681T patent/TR201809681T4/tr unknown
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|---|---|
| JP6367187B2 (ja) | 2018-08-01 |
| PL2870137T3 (pl) | 2018-12-31 |
| EP2870137A1 (en) | 2015-05-13 |
| WO2014006414A1 (en) | 2014-01-09 |
| US9512065B2 (en) | 2016-12-06 |
| US20150191421A1 (en) | 2015-07-09 |
| CA2878319C (en) | 2021-02-09 |
| GB201212081D0 (en) | 2012-08-22 |
| EP2870137B8 (en) | 2018-07-18 |
| CA2878319A1 (en) | 2014-01-09 |
| JP2015528798A (ja) | 2015-10-01 |
| HUE039775T2 (hu) | 2019-02-28 |
| EP2870137B1 (en) | 2018-05-16 |
| ES2679370T3 (es) | 2018-08-24 |
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