SMT201400071B - Composizione e procedimenti per l'inibizione dellavia di jak - Google Patents
Composizione e procedimenti per l'inibizione dellavia di jakInfo
- Publication number
- SMT201400071B SMT201400071B SM201400071T SM201400071T SMT201400071B SM T201400071 B SMT201400071 B SM T201400071B SM 201400071 T SM201400071 T SM 201400071T SM 201400071 T SM201400071 T SM 201400071T SM T201400071 B SMT201400071 B SM T201400071B
- Authority
- SM
- San Marino
- Prior art keywords
- inhibition
- procedures
- composition
- jak
- path
- Prior art date
Links
- 230000005764 inhibitory process Effects 0.000 title 1
- 238000000034 method Methods 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61K31/13—Amines
- A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- A61K31/5375—1,4-Oxazines, e.g. morpholine
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- A61K31/5375—1,4-Oxazines, e.g. morpholine
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- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D—HETEROCYCLIC COMPOUNDS
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- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
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- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
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- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Pulmonology (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Transplantation (AREA)
- Gastroenterology & Hepatology (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Saccharide Compounds (AREA)
- Dental Preparations (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US14705909P | 2009-01-23 | 2009-01-23 | |
US24163009P | 2009-09-11 | 2009-09-11 | |
PCT/US2010/021856 WO2010085684A1 (en) | 2009-01-23 | 2010-01-22 | Compositions and methods for inhibition of the jak pathway |
Publications (1)
Publication Number | Publication Date |
---|---|
SMT201400071B true SMT201400071B (it) | 2014-07-07 |
Family
ID=42091548
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SM201400071T SMT201400071B (it) | 2009-01-23 | 2014-06-13 | Composizione e procedimenti per l'inibizione dellavia di jak |
SM201500308T SMT201500308B (it) | 2009-01-23 | 2015-12-09 | Composizioni e procedimenti per l’inibizione della via di jak |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SM201500308T SMT201500308B (it) | 2009-01-23 | 2015-12-09 | Composizioni e procedimenti per l’inibizione della via di jak |
Country Status (24)
Country | Link |
---|---|
US (13) | US8324200B2 (es) |
EP (2) | EP2565193B1 (es) |
JP (1) | JP5802136B2 (es) |
KR (1) | KR101762967B1 (es) |
CN (1) | CN102356075B (es) |
AU (1) | AU2010206683B2 (es) |
BR (1) | BRPI1006942A2 (es) |
CA (1) | CA2749217C (es) |
DK (2) | DK2389372T3 (es) |
EA (1) | EA022802B1 (es) |
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