SK902004A3 - Kryštály obsahujúce soľ N-[2-(dietylamino)etyl]-5-[(5-fluór-2- oxo-3H-indol-3-ylidén)metyl]-2,4,dimetyl-1H-pyrrol-3-karboxamidu s kyselinou jablčnou, spôsob ich výroby a kompozície na ich báze - Google Patents

Kryštály obsahujúce soľ N-[2-(dietylamino)etyl]-5-[(5-fluór-2- oxo-3H-indol-3-ylidén)metyl]-2,4,dimetyl-1H-pyrrol-3-karboxamidu s kyselinou jablčnou, spôsob ich výroby a kompozície na ich báze Download PDF

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Publication number
SK902004A3
SK902004A3 SK90-2004A SK902004A SK902004A3 SK 902004 A3 SK902004 A3 SK 902004A3 SK 902004 A SK902004 A SK 902004A SK 902004 A3 SK902004 A3 SK 902004A3
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SK
Slovakia
Prior art keywords
crystal
malic acid
pyrrole
diethylamino
fluoro
Prior art date
Application number
SK90-2004A
Other languages
English (en)
Slovak (sk)
Inventor
Michael Hawley
Thomas J. Fleck
Stephen P. Prescott
Mark T. Maloney
Original Assignee
Pharmacia & Upjohn Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23211067&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK902004(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacia & Upjohn Company filed Critical Pharmacia & Upjohn Company
Publication of SK902004A3 publication Critical patent/SK902004A3/sk

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SK90-2004A 2001-08-15 2002-08-13 Kryštály obsahujúce soľ N-[2-(dietylamino)etyl]-5-[(5-fluór-2- oxo-3H-indol-3-ylidén)metyl]-2,4,dimetyl-1H-pyrrol-3-karboxamidu s kyselinou jablčnou, spôsob ich výroby a kompozície na ich báze SK902004A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31235301P 2001-08-15 2001-08-15
PCT/US2002/025649 WO2003016305A1 (en) 2001-08-15 2002-08-13 Crystals including a malic acid salt of n-[2-(diethylamino) ethyl]-5-[(5-fluoro-2-oxo-3h-indole-3-ylidene) methyl]-2, 4-dimethyl-1h-pyrrole-3-carboxamide, processes for its preparation and compositions thereof

Publications (1)

Publication Number Publication Date
SK902004A3 true SK902004A3 (sk) 2005-03-04

Family

ID=23211067

Family Applications (1)

Application Number Title Priority Date Filing Date
SK90-2004A SK902004A3 (sk) 2001-08-15 2002-08-13 Kryštály obsahujúce soľ N-[2-(dietylamino)etyl]-5-[(5-fluór-2- oxo-3H-indol-3-ylidén)metyl]-2,4,dimetyl-1H-pyrrol-3-karboxamidu s kyselinou jablčnou, spôsob ich výroby a kompozície na ich báze

Country Status (43)

Country Link
US (2) US20030069298A1 (hu)
EP (3) EP3168218B1 (hu)
JP (1) JP4159988B2 (hu)
KR (1) KR100639281B1 (hu)
CN (2) CN100439360C (hu)
AP (1) AP1660A (hu)
AR (1) AR036261A1 (hu)
AU (1) AU2002324684B2 (hu)
BG (1) BG108553A (hu)
BR (1) BR0211612A (hu)
CA (1) CA2455050C (hu)
CO (1) CO5550431A2 (hu)
CU (1) CU23713B7 (hu)
CY (1) CY1121552T1 (hu)
CZ (1) CZ2004196A3 (hu)
DK (2) DK1419151T3 (hu)
EA (1) EA006445B9 (hu)
EC (1) ECSP044975A (hu)
ES (3) ES2453164T3 (hu)
GE (1) GEP20063777B (hu)
HK (2) HK1066542A1 (hu)
HR (1) HRP20040112B1 (hu)
HU (1) HU229206B1 (hu)
IL (1) IL160097A0 (hu)
IS (1) IS7147A (hu)
MA (1) MA27058A1 (hu)
ME (1) ME00414B (hu)
MX (1) MXPA04001452A (hu)
MY (1) MY139383A (hu)
NO (1) NO326508B1 (hu)
NZ (1) NZ531232A (hu)
OA (1) OA12650A (hu)
PL (1) PL216524B1 (hu)
PT (2) PT1419151E (hu)
RS (1) RS53251B (hu)
SI (2) SI1419151T1 (hu)
SK (1) SK902004A3 (hu)
TN (1) TNSN04028A1 (hu)
TR (1) TR201900509T4 (hu)
TW (1) TWI269796B (hu)
UA (1) UA76483C2 (hu)
WO (1) WO2003016305A1 (hu)
ZA (1) ZA200400706B (hu)

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AP1660A (en) 2006-09-09
MXPA04001452A (es) 2004-05-20
PL216524B1 (pl) 2014-04-30
IL160097A0 (en) 2004-06-20
NO326508B1 (no) 2008-12-15
KR100639281B1 (ko) 2006-10-31
CU23713B7 (es) 2011-10-05
BR0211612A (pt) 2004-08-24
CZ2004196A3 (cs) 2005-01-12
AP2004002976A0 (en) 2004-03-31
EA200400183A1 (ru) 2004-08-26
NZ531232A (en) 2004-11-26
CN1789264A (zh) 2006-06-21
EP2332934A1 (en) 2011-06-15
CN1543462A (zh) 2004-11-03
CO5550431A2 (es) 2005-08-31
JP2005503386A (ja) 2005-02-03
NO20041054L (no) 2004-03-12
PT1419151E (pt) 2014-03-27
EP1419151B1 (en) 2014-02-26
PL368317A1 (en) 2005-03-21
MY139383A (en) 2009-09-30
US7435832B2 (en) 2008-10-14
HUP0700036A2 (en) 2008-10-28
HRP20040112A2 (en) 2004-06-30
HK1088008A1 (en) 2006-10-27
CA2455050A1 (en) 2003-02-27
CU20040029A7 (es) 2008-03-14
UA76483C2 (en) 2006-08-15
ECSP044975A (es) 2004-03-23
BG108553A (bg) 2005-04-30
AR036261A1 (es) 2004-08-25
TR201900509T4 (tr) 2019-02-21
DK1419151T3 (da) 2014-03-31
DK3168218T3 (en) 2019-01-14
JP4159988B2 (ja) 2008-10-01
US20070191458A1 (en) 2007-08-16
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