SK74494A3 - Pharmaceutical composition and process for the preparation thereof - Google Patents
Pharmaceutical composition and process for the preparation thereof Download PDFInfo
- Publication number
- SK74494A3 SK74494A3 SK744-94A SK74494A SK74494A3 SK 74494 A3 SK74494 A3 SK 74494A3 SK 74494 A SK74494 A SK 74494A SK 74494 A3 SK74494 A3 SK 74494A3
- Authority
- SK
- Slovakia
- Prior art keywords
- inhibitor
- mao
- phenyl
- composition
- uptake
- Prior art date
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- 238000000034 method Methods 0.000 title claims description 25
- 238000002360 preparation method Methods 0.000 title description 18
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- 230000000144 pharmacologic effect Effects 0.000 description 1
- 230000001817 pituitary effect Effects 0.000 description 1
- 229920003023 plastic Polymers 0.000 description 1
- 239000004033 plastic Substances 0.000 description 1
- 229920001282 polysaccharide Polymers 0.000 description 1
- 239000005017 polysaccharide Substances 0.000 description 1
- 239000001267 polyvinylpyrrolidone Substances 0.000 description 1
- 230000003389 potentiating effect Effects 0.000 description 1
- 239000000843 powder Substances 0.000 description 1
- 230000002265 prevention Effects 0.000 description 1
- 230000003449 preventive effect Effects 0.000 description 1
- 238000011084 recovery Methods 0.000 description 1
- 230000002829 reductive effect Effects 0.000 description 1
- 238000011160 research Methods 0.000 description 1
- 230000000979 retarding effect Effects 0.000 description 1
- 239000012266 salt solution Substances 0.000 description 1
- 238000005070 sampling Methods 0.000 description 1
- 230000035945 sensitivity Effects 0.000 description 1
- 239000011734 sodium Substances 0.000 description 1
- 229910052708 sodium Inorganic materials 0.000 description 1
- 239000007787 solid Substances 0.000 description 1
- 241000894007 species Species 0.000 description 1
- 210000000278 spinal cord Anatomy 0.000 description 1
- 230000004083 survival effect Effects 0.000 description 1
- 208000024891 symptom Diseases 0.000 description 1
- 238000003786 synthesis reaction Methods 0.000 description 1
- 238000012360 testing method Methods 0.000 description 1
- 230000001988 toxicity Effects 0.000 description 1
- 231100000419 toxicity Toxicity 0.000 description 1
- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
- HRXKRNGNAMMEHJ-UHFFFAOYSA-K trisodium citrate Chemical compound [Na+].[Na+].[Na+].[O-]C(=O)CC(O)(CC([O-])=O)C([O-])=O HRXKRNGNAMMEHJ-UHFFFAOYSA-K 0.000 description 1
- 210000002268 wool Anatomy 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Organic Chemistry (AREA)
- Psychiatry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU914060A HUT63579A (en) | 1991-12-20 | 1991-12-20 | Process for producing double-phase pharmaceutical compositions suitable for treating diseases occurring during neurodegenerative processes |
| PCT/HU1992/000060 WO1993012775A1 (en) | 1991-12-20 | 1992-12-18 | Pharmaceutical composition and process for the preparation thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK74494A3 true SK74494A3 (en) | 1995-01-12 |
Family
ID=10966728
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK744-94A SK74494A3 (en) | 1991-12-20 | 1992-12-18 | Pharmaceutical composition and process for the preparation thereof |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US5589513A (lt) |
| EP (1) | EP0617615A1 (lt) |
| JP (1) | JPH07502730A (lt) |
| KR (1) | KR940703655A (lt) |
| AU (1) | AU677170B2 (lt) |
| BG (1) | BG98827A (lt) |
| BR (1) | BR9206950A (lt) |
| CA (1) | CA2125776A1 (lt) |
| CZ (1) | CZ147494A3 (lt) |
| EC (1) | ECSP930933A (lt) |
| EE (1) | EE03015B1 (lt) |
| FI (1) | FI942932A (lt) |
| HU (2) | HUT63579A (lt) |
| IL (1) | IL104150A (lt) |
| LT (1) | LT3119B (lt) |
| LV (1) | LV10386B (lt) |
| MY (1) | MY111055A (lt) |
| NO (1) | NO942303D0 (lt) |
| NZ (1) | NZ246384A (lt) |
| PH (1) | PH31073A (lt) |
| PL (1) | PL172048B1 (lt) |
| RO (1) | RO115785B1 (lt) |
| RU (1) | RU2125448C1 (lt) |
| SI (1) | SI9200404A (lt) |
| SK (1) | SK74494A3 (lt) |
| WO (1) | WO1993012775A1 (lt) |
| ZA (1) | ZA929883B (lt) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5844003A (en) * | 1991-04-04 | 1998-12-01 | Innovations Foundation | Use of deprenyl compounds to maintain, prevent loss, or recover nerve cell function |
| US5817336A (en) * | 1993-04-02 | 1998-10-06 | Orion-Yhtyma Oy | Composition containing selegiline |
| DE4432610C1 (de) * | 1994-09-13 | 1996-02-01 | Knoll Ag | Verfahren zur Herstellung von Selegilin-Hydrochlorid |
| AU723047B2 (en) | 1995-02-10 | 2000-08-17 | University Of Toronto Innovations Foundation, The | Deprenyl compounds for treatment of glaucoma |
| JP4499208B2 (ja) * | 1998-10-29 | 2010-07-07 | 株式会社フジモト・コーポレーション | 新規な光学活性アミノペンタン誘導体 |
| US7374779B2 (en) * | 1999-02-26 | 2008-05-20 | Lipocine, Inc. | Pharmaceutical formulations and systems for improved absorption and multistage release of active agents |
| HUP9902482A2 (hu) * | 1999-07-22 | 2002-04-29 | Chinoin Gyógyszer és Vegyészeti Termékek Gyára Rt. | P-fluoro-selegilin alkalmazása neuroprotektív gyógyszerkészítmények előállítására |
| EP2053033A1 (en) * | 2007-10-26 | 2009-04-29 | Bayer Schering Pharma AG | Compounds for use in imaging, diagnosing and/or treatment of diseases of the central nervous system or of tumors |
| US11304960B2 (en) | 2009-01-08 | 2022-04-19 | Chandrashekar Giliyar | Steroidal compositions |
| DE102009045056A1 (de) * | 2009-09-28 | 2011-03-31 | Henkel Ag & Co. Kgaa | Fleckenvorbehandlungsmittel |
| US9034858B2 (en) | 2010-11-30 | 2015-05-19 | Lipocine Inc. | High-strength testosterone undecanoate compositions |
| US9358241B2 (en) | 2010-11-30 | 2016-06-07 | Lipocine Inc. | High-strength testosterone undecanoate compositions |
| US20180153904A1 (en) | 2010-11-30 | 2018-06-07 | Lipocine Inc. | High-strength testosterone undecanoate compositions |
| US20120148675A1 (en) | 2010-12-10 | 2012-06-14 | Basawaraj Chickmath | Testosterone undecanoate compositions |
| WO2016033556A1 (en) | 2014-08-28 | 2016-03-03 | Lipocine Inc. | BIOAVAILABLE SOLID STATE (17-β)-HYDROXY-4-ANDROSTEN-3-ONE ESTERS |
| WO2016033549A2 (en) | 2014-08-28 | 2016-03-03 | Lipocine Inc. | (17-ß)-3-OXOANDROST-4-EN-17-YL TRIDECANOATE COMPOSITIONS AND METHODS OF THEIR PREPARATION AND USE |
| JP2020503269A (ja) | 2016-11-28 | 2020-01-30 | リポカイン インコーポレーテッド | 経口ウンデカン酸テストステロン療法 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1227447B (de) * | 1962-03-30 | 1966-10-27 | Chinoin Gyogyszer Es Vegyeszet | Verfahren zur Herstellung von Phenylisopropylaminen |
| HU193662B (en) * | 1983-12-20 | 1987-11-30 | Chinoin Gyogyszer Es Vegyeszet | Process for producing synergetic pharmaceutical composition of antidepressive aktivity |
| HU207282B (en) * | 1984-05-31 | 1993-03-29 | Chinoin Gyogyszer Es Vegyeszet | Process for producing phenyl-alkyl-amine derivatives and pharmaceutical compositions containing them |
| DE3764144D1 (de) * | 1986-04-16 | 1990-09-13 | Asta Pharma Ag | Synergistische kombination von amantadin und selegilin. |
| HU207280B (en) * | 1986-09-25 | 1993-03-29 | Chinoin Gyogyszer Es Vegyeszet | Process for producing new phenyl-alkyl-amines and pharmaceutical compositions containing them |
| HU197510B (en) * | 1986-12-19 | 1989-04-28 | Chinoin Gyogyszer Es Vegyeszet | Process for producing pharmaceutical composition containing phenyl-alkyl-amine derivatives, against motion-sick |
| US4861800A (en) * | 1987-08-18 | 1989-08-29 | Buyske Donald A | Method for administering the drug deprenyl so as to minimize the danger of side effects |
| GB8807504D0 (en) * | 1988-03-29 | 1988-05-05 | Sandoz Ltd | Improvements in/relating to organic compounds |
| HU208484B (en) * | 1988-08-17 | 1993-11-29 | Chinoin Gyogyszer Es Vegyeszet | Process for producing pharmaceutical composition containing acid additional salt of selegilin as active component for treating schisofrenia |
| CA2037178A1 (en) * | 1990-02-28 | 1991-08-29 | Albert Walter Brzeczko | Deprenyl/l-dopa/carbidopa pharmaceutical composition |
| GB9011767D0 (en) * | 1990-05-25 | 1990-07-18 | Britannia Pharmaceuticals Ltd | Pharmaceutical compositions |
| US5169868A (en) * | 1991-03-01 | 1992-12-08 | University Of Saskatchewan | Aliphatic propargylamines as specific mao-b inhibitors |
| US5444095A (en) * | 1991-04-04 | 1995-08-22 | University Of Toronto, Innovations Foundation | Use of deprenyl to rescue damaged nerve cells |
| HU209605B (en) * | 1991-04-15 | 1994-09-28 | Chinoin Gyogyszer Es Vegyeszet | Process for production of wather-free transdermal preparation |
| US5326770A (en) * | 1992-07-17 | 1994-07-05 | The Du Pont Merck Pharmaceutical Company | Monoamine oxidase-B (MAO-B) inhibitory 5-substituted 2,4-thiazolidinediones useful in treating memory disorders of mammals |
-
1991
- 1991-12-20 HU HU914060A patent/HUT63579A/hu unknown
-
1992
- 1992-12-18 CZ CZ941474A patent/CZ147494A3/cs unknown
- 1992-12-18 RO RO94-01015A patent/RO115785B1/ro unknown
- 1992-12-18 AU AU32652/93A patent/AU677170B2/en not_active Ceased
- 1992-12-18 JP JP5510411A patent/JPH07502730A/ja active Pending
- 1992-12-18 EP EP93901880A patent/EP0617615A1/en not_active Withdrawn
- 1992-12-18 ZA ZA929883A patent/ZA929883B/xx unknown
- 1992-12-18 US US08/256,128 patent/US5589513A/en not_active Expired - Fee Related
- 1992-12-18 PL PL92304116A patent/PL172048B1/pl unknown
- 1992-12-18 BR BR9206950A patent/BR9206950A/pt not_active Application Discontinuation
- 1992-12-18 KR KR1019940702143A patent/KR940703655A/ko active IP Right Grant
- 1992-12-18 PH PH45474A patent/PH31073A/en unknown
- 1992-12-18 NZ NZ246384A patent/NZ246384A/en unknown
- 1992-12-18 SK SK744-94A patent/SK74494A3/sk unknown
- 1992-12-18 MY MYPI92002341A patent/MY111055A/en unknown
- 1992-12-18 SI SI9200404A patent/SI9200404A/sl unknown
- 1992-12-18 IL IL104150A patent/IL104150A/xx not_active IP Right Cessation
- 1992-12-18 CA CA002125776A patent/CA2125776A1/en not_active Abandoned
- 1992-12-18 RU RU94031161A patent/RU2125448C1/ru active
- 1992-12-18 WO PCT/HU1992/000060 patent/WO1993012775A1/en not_active Application Discontinuation
- 1992-12-20 LV LVP-92-547A patent/LV10386B/en unknown
- 1992-12-21 LT LTIP249A patent/LT3119B/lt not_active IP Right Cessation
-
1993
- 1993-05-25 EC EC1993000933A patent/ECSP930933A/es unknown
-
1994
- 1994-06-02 BG BG98827A patent/BG98827A/xx unknown
- 1994-06-17 FI FI942932A patent/FI942932A/fi unknown
- 1994-06-17 NO NO942303A patent/NO942303D0/no unknown
- 1994-08-10 EE EE9400117A patent/EE03015B1/xx unknown
-
1995
- 1995-06-16 HU HU95P/P00218P patent/HU211478A9/hu unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI942932A0 (fi) | 1994-06-17 |
| CZ147494A3 (en) | 1995-01-18 |
| LV10386A (lv) | 1995-02-20 |
| HU914060D0 (en) | 1992-03-30 |
| RO115785B1 (ro) | 2000-06-30 |
| HUT63579A (en) | 1993-09-28 |
| US5589513A (en) | 1996-12-31 |
| ECSP930933A (es) | 1994-04-20 |
| ZA929883B (en) | 1994-05-16 |
| BR9206950A (pt) | 1995-11-28 |
| PH31073A (en) | 1998-02-05 |
| CA2125776A1 (en) | 1993-07-08 |
| EE03015B1 (et) | 1997-08-15 |
| IL104150A (en) | 1997-11-20 |
| NZ246384A (en) | 1996-02-27 |
| AU3265293A (en) | 1993-07-28 |
| RU2125448C1 (ru) | 1999-01-27 |
| PL172048B1 (pl) | 1997-07-31 |
| JPH07502730A (ja) | 1995-03-23 |
| LTIP249A (en) | 1994-07-15 |
| HU211478A9 (en) | 1995-11-28 |
| LT3119B (en) | 1994-12-27 |
| SI9200404A (en) | 1993-06-30 |
| WO1993012775A1 (en) | 1993-07-08 |
| NO942303D0 (no) | 1994-06-17 |
| MY111055A (en) | 1999-08-30 |
| FI942932A (fi) | 1994-06-17 |
| LV10386B (en) | 1995-12-20 |
| KR940703655A (ko) | 1994-12-12 |
| BG98827A (en) | 1995-06-30 |
| AU677170B2 (en) | 1997-04-17 |
| EP0617615A1 (en) | 1994-10-05 |
| NO942303L (lt) | 1994-08-17 |
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