SK47695A3 - Boropeptide derivatives, method of their preparation and pharmaceutical agents containing these derivatives - Google Patents

Boropeptide derivatives, method of their preparation and pharmaceutical agents containing these derivatives Download PDF

Info

Publication number
SK47695A3
SK47695A3 SK476-95A SK47695A SK47695A3 SK 47695 A3 SK47695 A3 SK 47695A3 SK 47695 A SK47695 A SK 47695A SK 47695 A3 SK47695 A3 SK 47695A3
Authority
SK
Slovakia
Prior art keywords
formula
compound
carbon atoms
straight
alkyl
Prior art date
Application number
SK476-95A
Other languages
English (en)
Slovak (sk)
Inventor
Sergio Mallart
Gilbert Lassalle
Thomas A Purcell
Jean-Claude Muller
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of SK47695A3 publication Critical patent/SK47695A3/sk

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06191Dipeptides containing heteroatoms different from O, S, or N
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biophysics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SK476-95A 1994-04-12 1995-04-11 Boropeptide derivatives, method of their preparation and pharmaceutical agents containing these derivatives SK47695A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9404288A FR2718451B1 (fr) 1994-04-12 1994-04-12 Dérivés de peptides boroniques, leur préparation et leur application en thérapeutique.

Publications (1)

Publication Number Publication Date
SK47695A3 true SK47695A3 (en) 1995-12-06

Family

ID=9461981

Family Applications (1)

Application Number Title Priority Date Filing Date
SK476-95A SK47695A3 (en) 1994-04-12 1995-04-11 Boropeptide derivatives, method of their preparation and pharmaceutical agents containing these derivatives

Country Status (17)

Country Link
EP (1) EP0677531A1 (no)
JP (1) JPH07285990A (no)
KR (1) KR950032225A (no)
CN (1) CN1113493A (no)
AU (1) AU1638095A (no)
CA (1) CA2146833A1 (no)
CZ (1) CZ92295A3 (no)
FI (1) FI951726A (no)
FR (1) FR2718451B1 (no)
HU (1) HUT71617A (no)
IL (1) IL113332A0 (no)
NO (1) NO951418L (no)
NZ (1) NZ270913A (no)
PL (1) PL308074A1 (no)
RU (1) RU95105419A (no)
SK (1) SK47695A3 (no)
ZA (1) ZA952983B (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5726159A (en) * 1994-03-04 1998-03-10 Eli Lilly And Company Antithrombotic agents
CA2143533A1 (en) * 1994-03-04 1995-09-05 Kenneth D. Kurz Antithrombotic agents
US5602101A (en) * 1994-03-04 1997-02-11 Eli Lilly And Company Antithrombotic agents
US5707966A (en) * 1994-03-04 1998-01-13 Eli Lilly And Company Antithrombotic agents
ZA951618B (en) * 1994-03-04 1996-08-27 Lilly Co Eli Antithrombotic agents
US5885967A (en) * 1994-03-04 1999-03-23 Eli Lilly And Company Antithrombotic agents
US5705487A (en) * 1994-03-04 1998-01-06 Eli Lilly And Company Antithrombotic agents
US5710130A (en) * 1995-02-27 1998-01-20 Eli Lilly And Company Antithrombotic agents
US5914319A (en) * 1995-02-27 1999-06-22 Eli Lilly And Company Antithrombotic agents
US5639739A (en) * 1995-03-24 1997-06-17 The Dupont Merck Pharmaceutical Company Imidazole containing aminoboronic acids
FR2739858B1 (fr) * 1995-10-11 1997-11-14 Synthelabo Derives de n-sulfonyl- et n-sulfamoylpeptidylprolinamide, leur preparation et leur application en therapeutique
US5811402A (en) * 1996-03-22 1998-09-22 Eli Lilly And Company Antithrombotic diamides
FR2758329B1 (fr) * 1997-01-16 1999-02-12 Synthelabo Derives d'imidazole-4-butane boronique, leur preparation et leur utilisation en therapeutique

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides
US5187157A (en) * 1987-06-05 1993-02-16 Du Pont Merck Pharmaceutical Company Peptide boronic acid inhibitors of trypsin-like proteases
EP0315574A3 (de) * 1987-11-05 1990-08-22 Hoechst Aktiengesellschaft Renin-Inhibitoren

Also Published As

Publication number Publication date
IL113332A0 (en) 1995-07-31
CZ92295A3 (en) 1995-11-15
AU1638095A (en) 1995-10-19
RU95105419A (ru) 1997-01-10
JPH07285990A (ja) 1995-10-31
CN1113493A (zh) 1995-12-20
FI951726A0 (fi) 1995-04-11
HUT71617A (en) 1996-01-29
CA2146833A1 (fr) 1995-10-13
NZ270913A (en) 1996-05-28
FR2718451A1 (fr) 1995-10-13
PL308074A1 (en) 1995-10-16
ZA952983B (en) 1996-01-11
KR950032225A (ko) 1995-12-20
NO951418D0 (no) 1995-04-11
EP0677531A1 (fr) 1995-10-18
FR2718451B1 (fr) 1996-05-10
HU9501041D0 (en) 1995-06-28
FI951726A (fi) 1995-10-13
NO951418L (no) 1995-10-13

Similar Documents

Publication Publication Date Title
JP3273515B2 (ja) 抗血栓剤としてのペプチドアルデヒド類
EP0012845B1 (en) Tetrahydroisoquinoline compounds, process for preparing same and pharmaceutical compositions containing them
US5444049A (en) Peptide compounds derived from boronic acid
TW234717B (en) 1-[2-(arylsulfonylamine)-1-oxoethyl]piperidine derivatives, their preparation and therapeutic applications
JP2018536702A (ja) Tlr7アゴニストとしての7−(チアゾール−5−イル)ピロロピリミジン化合物
WO2004076433A1 (en) Dipeptidyl peptidase inhibitors
SK47695A3 (en) Boropeptide derivatives, method of their preparation and pharmaceutical agents containing these derivatives
CN102532198A (zh) 抗病毒的次膦酸酯化合物
WO2004076434A1 (en) Dipeptidyl peptidase inhibitors
CN101379059A (zh) N-羟基丙烯酰胺化合物
HU181087B (en) Process for producing mercapto-acyl-dipeptides
CN111606970B (zh) 一种1,5-二氮杂双环[5,3,0]十烷酮氨基酸衍生物及其制备方法和应用
TW201030011A (en) Imidazothiazole derivatives bearing the proline ring structure
NO329543B1 (no) Diketopiperazinderivater, farmasoytiske sammensetninger samt anvendelser derav
JP6333825B2 (ja) インドリン
CA2021944A1 (en) Antiherpetic agents
CA3090646A1 (en) Co-crystal forms of a novobiocin analog and proline
RU2259997C2 (ru) Ингибиторы фарнезилтрансферазы
US4206122A (en) Derivatives of pyrrolidinecarboxaldehyde and piperidinecarboxaldehyde and intermediates therefor
AU2012309556A1 (en) Pyrrolidine-3-ylacetic acid derivative
JP2023549187A (ja) 貧血およびがんの処置のためのvhl阻害剤としての1-(2-(4-シクロプロピル-1h-1,2,3-トリアゾール-1-イル)アセチル)-4-ヒドロキシ-n-(ベンジル)ピロリジンe-2-カルボキサミド誘導体
US6262060B1 (en) Azacycloalkane derivatives, preparation and therapeutic application
EP0533241A2 (en) Substituted alkyl derivatives of piperazinylcamphorsulfonyl oxytocin antagonists
JPH07121908B2 (ja) 新規置換アミノ酸誘導体、その製法およびそれを含有する医薬組成物
JPS59141544A (ja) ラクタムペプチド及びその製造方法、並びに該ペプチドを含有する医薬