SK19092001A3 - Indanylsubstituované benzénkarboxamidy, spôsob ich prípravy, ich použitie ako liečiva, a farmaceutické prostriedky, ktoré ich obsahujú - Google Patents

Indanylsubstituované benzénkarboxamidy, spôsob ich prípravy, ich použitie ako liečiva, a farmaceutické prostriedky, ktoré ich obsahujú Download PDF

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Publication number
SK19092001A3
SK19092001A3 SK1909-2001A SK19092001A SK19092001A3 SK 19092001 A3 SK19092001 A3 SK 19092001A3 SK 19092001 A SK19092001 A SK 19092001A SK 19092001 A3 SK19092001 A3 SK 19092001A3
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SK
Slovakia
Prior art keywords
group
carbon atoms
hydrogen
alkyl
atom
Prior art date
Application number
SK1909-2001A
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English (en)
Slovak (sk)
Inventor
Joachim Brendel
Uwe Gerlach
Hans Ulrich Stilz
Hans Jochen Lang
Original Assignee
Aventis Pharma Deutschland Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Deutschland Gmbh filed Critical Aventis Pharma Deutschland Gmbh
Publication of SK19092001A3 publication Critical patent/SK19092001A3/sk

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/16—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/20—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/21—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/22—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms
    • C07C311/23—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms having the sulfur atoms of the sulfonamide groups bound to acyclic carbon atoms
    • C07C311/26—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms having the sulfur atoms of the sulfonamide groups bound to acyclic carbon atoms of an acyclic unsaturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/04—Systems containing only non-condensed rings with a four-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/08—One of the condensed rings being a six-membered aromatic ring the other ring being five-membered, e.g. indane

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
SK1909-2001A 1999-06-25 2000-06-10 Indanylsubstituované benzénkarboxamidy, spôsob ich prípravy, ich použitie ako liečiva, a farmaceutické prostriedky, ktoré ich obsahujú SK19092001A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19929076A DE19929076A1 (de) 1999-06-25 1999-06-25 Indanylsubstituierte Benzolcarbonamide, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament sowie sie enthaltende pharmazeutische Zubereitungen
PCT/EP2000/005370 WO2001000573A1 (de) 1999-06-25 2000-06-10 Indanylsubstituierte benzolcarbonamide, verfahren zu ihrer herstellung, ihre verwendung als medikament sowie sie enthaltende pharmazeutische zubereitungen

Publications (1)

Publication Number Publication Date
SK19092001A3 true SK19092001A3 (sk) 2002-06-04

Family

ID=7912468

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1909-2001A SK19092001A3 (sk) 1999-06-25 2000-06-10 Indanylsubstituované benzénkarboxamidy, spôsob ich prípravy, ich použitie ako liečiva, a farmaceutické prostriedky, ktoré ich obsahujú

Country Status (31)

Country Link
US (1) US6221866B1 (tr)
EP (1) EP1194403B1 (tr)
JP (1) JP4527918B2 (tr)
KR (1) KR20020023962A (tr)
CN (1) CN1157372C (tr)
AR (1) AR024443A1 (tr)
AT (1) ATE248811T1 (tr)
AU (1) AU771601B2 (tr)
BR (1) BR0011938A (tr)
CA (1) CA2377087A1 (tr)
CZ (1) CZ20014523A3 (tr)
DE (2) DE19929076A1 (tr)
DK (1) DK1194403T3 (tr)
EE (1) EE04464B1 (tr)
ES (1) ES2200886T3 (tr)
HK (1) HK1047575B (tr)
HU (1) HUP0201711A3 (tr)
IL (1) IL147220A0 (tr)
MX (1) MXPA01012281A (tr)
NO (1) NO20015816D0 (tr)
NZ (1) NZ516347A (tr)
PL (1) PL352985A1 (tr)
PT (1) PT1194403E (tr)
RU (1) RU2238934C2 (tr)
SI (1) SI1194403T1 (tr)
SK (1) SK19092001A3 (tr)
TR (1) TR200103701T2 (tr)
TW (1) TWI256950B (tr)
WO (1) WO2001000573A1 (tr)
YU (1) YU88801A (tr)
ZA (1) ZA200109732B (tr)

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DE10121003A1 (de) * 2001-04-28 2002-12-19 Aventis Pharma Gmbh Anthranilsäureamide, Verfahren zur Herstellung, ihrer Verwendung als Medikament sowie sie enthaltende pharmazeutische Zubereitungen
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GB0412986D0 (en) 2004-06-10 2004-07-14 Xention Discovery Ltd Compounds
US7569589B2 (en) 2004-07-29 2009-08-04 Merck & Co., Inc. Potassium channel inhibitors
US7576212B2 (en) 2004-12-09 2009-08-18 Xention Limited Thieno[2,3-B] pyridines as potassium channel inhibitors
DE102005028845A1 (de) * 2005-06-22 2006-12-28 Sanofi-Aventis Deutschland Gmbh Substituierte Heterocyclen, ihre Verwendung als Medikament sowie enthaltende pharmazeutische Zubereitungen
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JP5749162B2 (ja) * 2008-07-10 2015-07-15 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｂ２受容体を調節するスルホン化合物
GB0815784D0 (en) 2008-08-29 2008-10-08 Xention Ltd Novel potassium channel blockers
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GB0815782D0 (en) 2008-08-29 2008-10-08 Xention Ltd Novel potassium channel blockers
CN102164917A (zh) * 2008-09-25 2011-08-24 贝林格尔.英格海姆国际有限公司 选择性调节cb2受体的磺酰基化合物
US8299103B2 (en) * 2009-06-15 2012-10-30 Boehringer Ingelheim International Gmbh Compounds which selectively modulate the CB2 receptor
US8383615B2 (en) 2009-06-16 2013-02-26 Boehringer Ingelheim International Gmbh Azetidine 2-carboxamide derivatives which modulate the CB2 receptor
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EP2523936A1 (en) 2010-01-15 2012-11-21 Boehringer Ingelheim International GmbH Compounds which modulate the cb2 receptor
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Also Published As

Publication number Publication date
PL352985A1 (en) 2003-09-22
AR024443A1 (es) 2002-10-02
BR0011938A (pt) 2002-03-19
DK1194403T3 (da) 2003-12-08
HK1047575B (zh) 2004-12-31
MXPA01012281A (es) 2002-07-30
KR20020023962A (ko) 2002-03-29
NO20015816L (no) 2001-11-29
PT1194403E (pt) 2004-01-30
CA2377087A1 (en) 2001-01-04
YU88801A (sh) 2004-09-03
ZA200109732B (en) 2002-08-30
HUP0201711A3 (en) 2005-05-30
EP1194403A1 (de) 2002-04-10
NZ516347A (en) 2004-01-30
IL147220A0 (en) 2002-08-14
JP4527918B2 (ja) 2010-08-18
CN1358172A (zh) 2002-07-10
JP2003503385A (ja) 2003-01-28
US6221866B1 (en) 2001-04-24
TWI256950B (en) 2006-06-21
ES2200886T3 (es) 2004-03-16
TR200103701T2 (tr) 2002-05-21
HK1047575A1 (en) 2003-02-28
AU5531800A (en) 2001-01-31
NO20015816D0 (no) 2001-11-29
EE04464B1 (et) 2005-04-15
AU771601B2 (en) 2004-03-25
DE19929076A1 (de) 2000-12-28
RU2238934C2 (ru) 2004-10-27
CN1157372C (zh) 2004-07-14
CZ20014523A3 (cs) 2002-04-17
SI1194403T1 (en) 2003-12-31
EE200100684A (et) 2003-04-15
DE50003555D1 (de) 2003-10-09
HUP0201711A2 (en) 2002-09-28
ATE248811T1 (de) 2003-09-15
EP1194403B1 (de) 2003-09-03
WO2001000573A1 (de) 2001-01-04

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