SK12822002A3 - Perličky s trvalým uvoľňovaním obsahujúce stavudín - Google Patents

Perličky s trvalým uvoľňovaním obsahujúce stavudín Download PDF

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Publication number
SK12822002A3
SK12822002A3 SK1282-2002A SK12822002A SK12822002A3 SK 12822002 A3 SK12822002 A3 SK 12822002A3 SK 12822002 A SK12822002 A SK 12822002A SK 12822002 A3 SK12822002 A3 SK 12822002A3
Authority
SK
Slovakia
Prior art keywords
stavudine
beads
spherical beads
extruded
drug
Prior art date
Application number
SK1282-2002A
Other languages
English (en)
Slovak (sk)
Inventor
Rober Abramowitz
Denise M. O'donoghue
Nemichand B. Jain
Original Assignee
Bristol-Myers Squibb Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Company filed Critical Bristol-Myers Squibb Company
Publication of SK12822002A3 publication Critical patent/SK12822002A3/sk

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
    • A61K31/7072—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Biophysics (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SK1282-2002A 2000-03-30 2001-03-29 Perličky s trvalým uvoľňovaním obsahujúce stavudín SK12822002A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US19358800P 2000-03-30 2000-03-30
PCT/US2001/010078 WO2001074329A2 (en) 2000-03-30 2001-03-29 Sustained release beadlets containing stavudine

Publications (1)

Publication Number Publication Date
SK12822002A3 true SK12822002A3 (sk) 2003-02-04

Family

ID=22714247

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1282-2002A SK12822002A3 (sk) 2000-03-30 2001-03-29 Perličky s trvalým uvoľňovaním obsahujúce stavudín

Country Status (26)

Country Link
US (1) US7135465B2 (lt)
EP (1) EP1267879A2 (lt)
JP (1) JP2003528905A (lt)
KR (1) KR20030011805A (lt)
CN (1) CN1187052C (lt)
AR (1) AR027748A1 (lt)
AU (1) AU2001249591A1 (lt)
BG (1) BG107157A (lt)
BR (1) BR0109602A (lt)
CA (1) CA2404687A1 (lt)
CZ (1) CZ20023003A3 (lt)
EE (1) EE200200564A (lt)
GE (1) GEP20043285B (lt)
HU (1) HUP0302631A2 (lt)
IL (1) IL151475A0 (lt)
LT (1) LT5045B (lt)
LV (1) LV12939B (lt)
MX (1) MXPA02009534A (lt)
NO (1) NO20024645L (lt)
NZ (1) NZ522250A (lt)
PE (1) PE20011179A1 (lt)
PL (1) PL366089A1 (lt)
RU (1) RU2239435C2 (lt)
SK (1) SK12822002A3 (lt)
WO (1) WO2001074329A2 (lt)
ZA (1) ZA200207760B (lt)

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US20060024361A1 (en) * 2004-07-28 2006-02-02 Isa Odidi Disintegrant assisted controlled release technology
US10624858B2 (en) 2004-08-23 2020-04-21 Intellipharmaceutics Corp Controlled release composition using transition coating, and method of preparing same
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Also Published As

Publication number Publication date
NO20024645D0 (no) 2002-09-27
EP1267879A2 (en) 2003-01-02
EE200200564A (et) 2004-06-15
WO2001074329A2 (en) 2001-10-11
NO20024645L (no) 2002-09-27
CN1187052C (zh) 2005-02-02
PE20011179A1 (es) 2001-12-06
MXPA02009534A (es) 2003-05-14
ZA200207760B (en) 2004-01-30
LT2002099A (lt) 2003-04-25
LV12939B (en) 2003-04-20
RU2239435C2 (ru) 2004-11-10
AR027748A1 (es) 2003-04-09
HUP0302631A2 (hu) 2003-11-28
AU2001249591A1 (en) 2001-10-15
KR20030011805A (ko) 2003-02-11
RU2002126540A (ru) 2004-03-27
PL366089A1 (en) 2005-01-24
BR0109602A (pt) 2004-06-29
GEP20043285B (en) 2004-07-26
LT5045B (lt) 2003-08-25
NZ522250A (en) 2004-09-24
CN1420774A (zh) 2003-05-28
WO2001074329A3 (en) 2002-05-10
CA2404687A1 (en) 2001-10-11
CZ20023003A3 (cs) 2002-11-13
US7135465B2 (en) 2006-11-14
US20020002147A1 (en) 2002-01-03
IL151475A0 (en) 2003-04-10
JP2003528905A (ja) 2003-09-30
BG107157A (en) 2003-06-30

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