SK11002001A3 - Heteroarylom substituované chinolin-2-ónové deriváty použiteľné ako protinádorové prostriedky - Google Patents

Heteroarylom substituované chinolin-2-ónové deriváty použiteľné ako protinádorové prostriedky Download PDF

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Publication number
SK11002001A3
SK11002001A3 SK1100-2001A SK11002001A SK11002001A3 SK 11002001 A3 SK11002001 A3 SK 11002001A3 SK 11002001 A SK11002001 A SK 11002001A SK 11002001 A3 SK11002001 A3 SK 11002001A3
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SK
Slovakia
Prior art keywords
group
aryl
methyl
substituents
alkyl
Prior art date
Application number
SK1100-2001A
Other languages
English (en)
Slovak (sk)
Inventor
Bingwei Vera Yang
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of SK11002001A3 publication Critical patent/SK11002001A3/sk

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Virology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SK1100-2001A 1999-02-11 2000-02-04 Heteroarylom substituované chinolin-2-ónové deriváty použiteľné ako protinádorové prostriedky SK11002001A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11970299P 1999-02-11 1999-02-11
PCT/IB2000/000121 WO2000047574A1 (en) 1999-02-11 2000-02-04 Heteroaryl-substituted quinolin-2-one derivatives useful as anticancer agents

Publications (1)

Publication Number Publication Date
SK11002001A3 true SK11002001A3 (sk) 2002-05-09

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Family Applications (1)

Application Number Title Priority Date Filing Date
SK1100-2001A SK11002001A3 (sk) 1999-02-11 2000-02-04 Heteroarylom substituované chinolin-2-ónové deriváty použiteľné ako protinádorové prostriedky

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Country Link
US (3) US6258824B1 (OSRAM)
EP (1) EP1150973B1 (OSRAM)
JP (3) JP4090200B2 (OSRAM)
KR (1) KR20010102073A (OSRAM)
CN (1) CN1340051A (OSRAM)
AP (1) AP2001002241A0 (OSRAM)
AR (1) AR028985A1 (OSRAM)
AT (1) ATE297916T1 (OSRAM)
AU (1) AU2124800A (OSRAM)
BG (1) BG105860A (OSRAM)
BR (1) BR0008202A (OSRAM)
CA (1) CA2362394C (OSRAM)
CO (1) CO5140097A1 (OSRAM)
CZ (1) CZ20012910A3 (OSRAM)
DE (1) DE60020812T2 (OSRAM)
DZ (1) DZ3009A1 (OSRAM)
EA (1) EA200100766A1 (OSRAM)
EE (1) EE200100425A (OSRAM)
ES (1) ES2243228T3 (OSRAM)
GT (1) GT200000014A (OSRAM)
HK (1) HK1042096A1 (OSRAM)
HN (1) HN2000000019A (OSRAM)
HR (1) HRP20010574A2 (OSRAM)
HU (1) HUP0105231A3 (OSRAM)
ID (1) ID29584A (OSRAM)
IL (1) IL144307A0 (OSRAM)
IS (1) IS5997A (OSRAM)
MA (1) MA26718A1 (OSRAM)
NO (1) NO20013909L (OSRAM)
OA (1) OA11833A (OSRAM)
PA (1) PA8490601A1 (OSRAM)
PE (1) PE20001464A1 (OSRAM)
PL (1) PL349839A1 (OSRAM)
SK (1) SK11002001A3 (OSRAM)
SV (1) SV2001000020A (OSRAM)
TN (1) TNSN00028A1 (OSRAM)
TR (2) TR200201296T2 (OSRAM)
WO (1) WO2000047574A1 (OSRAM)
ZA (1) ZA200106520B (OSRAM)

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JP4216740B2 (ja) 2009-01-28
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