TW200504057A - Benzothiophene derivative - Google Patents
Benzothiophene derivativeInfo
- Publication number
- TW200504057A TW200504057A TW093105203A TW93105203A TW200504057A TW 200504057 A TW200504057 A TW 200504057A TW 093105203 A TW093105203 A TW 093105203A TW 93105203 A TW93105203 A TW 93105203A TW 200504057 A TW200504057 A TW 200504057A
- Authority
- TW
- Taiwan
- Prior art keywords
- benzothiophene derivative
- compound
- whixh
- berepresented
- prodrug
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
This invention relates to a compound useful as an antitumor agent ,a process for producing the same and a medicine containing the compound whixh could berepresented by the formula (I): (wherein R1 represents nitro group, etc.; R2 represents hydrogen atom, etc.; R3 represents C1-4 linear or branched alkyl group), its salt, prodrug or solvate.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2003050369 | 2003-02-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
TW200504057A true TW200504057A (en) | 2005-02-01 |
Family
ID=32923343
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TW093105203A TW200504057A (en) | 2003-02-27 | 2004-02-27 | Benzothiophene derivative |
Country Status (2)
Country | Link |
---|---|
TW (1) | TW200504057A (en) |
WO (1) | WO2004076446A1 (en) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1756085B1 (en) * | 2004-05-03 | 2010-06-16 | Janssen Pharmaceutica N.V. | Diastereoselective synthesis process with 6-bromo-4-(3-chlorophenyl)-2-methoxy-quinoline |
CN100567290C (en) * | 2004-05-03 | 2009-12-09 | 詹森药业有限公司 | The cis-selectivity addition of lithiated n-methylimidazole on sulfinimines |
WO2006101454A1 (en) * | 2005-03-21 | 2006-09-28 | S*Bio Pte Ltd | Benzothiophene derivatives: preparation and pharmaceutical applications |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA200100766A1 (en) * | 1999-02-11 | 2002-02-28 | Пфайзер Продактс Инк. | QUINOLIN-2-ON-SUBSTITUTED HETEROAARYNE DERIVATIVES USED AS ANTI-TUMOR AGENTS |
JP4974438B2 (en) * | 2000-09-25 | 2012-07-11 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | 6-Heterocyclylmethylquinoline and quinazoline derivatives that inhibit farnesyltransferase |
-
2004
- 2004-02-27 WO PCT/JP2004/002427 patent/WO2004076446A1/en not_active Application Discontinuation
- 2004-02-27 TW TW093105203A patent/TW200504057A/en unknown
Also Published As
Publication number | Publication date |
---|---|
WO2004076446A1 (en) | 2004-09-10 |
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