BR0008202A - Derivados de quinolin-2-ona substituìdos com heteroarilas úteis como agentes contra o câncer - Google Patents
Derivados de quinolin-2-ona substituìdos com heteroarilas úteis como agentes contra o câncerInfo
- Publication number
- BR0008202A BR0008202A BR0008202-3A BR0008202A BR0008202A BR 0008202 A BR0008202 A BR 0008202A BR 0008202 A BR0008202 A BR 0008202A BR 0008202 A BR0008202 A BR 0008202A
- Authority
- BR
- Brazil
- Prior art keywords
- quinolin
- compounds
- formula
- useful
- agents against
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US11970299P | 1999-02-11 | 1999-02-11 | |
PCT/IB2000/000121 WO2000047574A1 (en) | 1999-02-11 | 2000-02-04 | Heteroaryl-substituted quinolin-2-one derivatives useful as anticancer agents |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0008202A true BR0008202A (pt) | 2002-02-19 |
Family
ID=22385869
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0008202-3A BR0008202A (pt) | 1999-02-11 | 2000-02-04 | Derivados de quinolin-2-ona substituìdos com heteroarilas úteis como agentes contra o câncer |
Country Status (39)
Country | Link |
---|---|
US (3) | US6258824B1 (pt) |
EP (1) | EP1150973B1 (pt) |
JP (3) | JP4090200B2 (pt) |
KR (1) | KR20010102073A (pt) |
CN (1) | CN1340051A (pt) |
AP (1) | AP2001002241A0 (pt) |
AR (1) | AR028985A1 (pt) |
AT (1) | ATE297916T1 (pt) |
AU (1) | AU2124800A (pt) |
BG (1) | BG105860A (pt) |
BR (1) | BR0008202A (pt) |
CA (1) | CA2362394C (pt) |
CO (1) | CO5140097A1 (pt) |
CZ (1) | CZ20012910A3 (pt) |
DE (1) | DE60020812T2 (pt) |
DZ (1) | DZ3009A1 (pt) |
EA (1) | EA200100766A1 (pt) |
EE (1) | EE200100425A (pt) |
ES (1) | ES2243228T3 (pt) |
GT (1) | GT200000014A (pt) |
HK (1) | HK1042096A1 (pt) |
HN (1) | HN2000000019A (pt) |
HR (1) | HRP20010574A2 (pt) |
HU (1) | HUP0105231A3 (pt) |
ID (1) | ID29584A (pt) |
IL (1) | IL144307A0 (pt) |
IS (1) | IS5997A (pt) |
MA (1) | MA26718A1 (pt) |
NO (1) | NO20013909L (pt) |
OA (1) | OA11833A (pt) |
PA (1) | PA8490601A1 (pt) |
PE (1) | PE20001464A1 (pt) |
PL (1) | PL349839A1 (pt) |
SK (1) | SK11002001A3 (pt) |
SV (1) | SV2001000020A (pt) |
TN (1) | TNSN00028A1 (pt) |
TR (2) | TR200201297T2 (pt) |
WO (1) | WO2000047574A1 (pt) |
ZA (1) | ZA200106520B (pt) |
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DE60008574T2 (de) * | 1999-11-05 | 2009-10-01 | Cytovia, Inc., San Diego | Substituierte 4H-Chromene und Analoga als Caspase-Aktivatoren und Apoptose-Induktoren und deren Verwendung |
EP1106612B1 (en) * | 1999-11-30 | 2004-02-11 | Pfizer Products Inc. | Quinoline derivatives useful for inhibiting farnesyl protein transferase |
HN2000000266A (es) * | 2000-01-21 | 2001-05-21 | Pfizer Prod Inc | Compuesto anticanceroso y metodo de separacion de enantiomeros util para sintetizar dicho compuesto. |
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EP1170011A1 (en) * | 2000-07-06 | 2002-01-09 | Boehringer Ingelheim International GmbH | Novel use of inhibitors of the epidermal growth factor receptor |
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US7153958B2 (en) | 2000-11-21 | 2006-12-26 | Janssen Pharmaceutica N.V. | Farnesyl transferase inhibiting benzoheterocyclic derivatives |
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ID27562A (id) | 1998-08-27 | 2001-04-12 | Pfizer Prod Inc | Turunan-turunan kinolin-2-ona tersubstitusi alkunil yang berguna sebagai zat anti kanker |
ID29584A (id) * | 1999-02-11 | 2001-09-06 | Pfizer Prod Inc | Turunan-turunan kuinolin-2-on tersubstitusi heteroaril yang bermanfaat sebagai zat-zat anti kanker |
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