BRPI0811783A2 - Compostos de ((heteroarila bicíclica)imidazolil)metil-heteroarila como agonistas dos receptores adrenérgicos. - Google Patents

Compostos de ((heteroarila bicíclica)imidazolil)metil-heteroarila como agonistas dos receptores adrenérgicos.

Info

Publication number
BRPI0811783A2
BRPI0811783A2 BRPI0811783-7A2A BRPI0811783A BRPI0811783A2 BR PI0811783 A2 BRPI0811783 A2 BR PI0811783A2 BR PI0811783 A BRPI0811783 A BR PI0811783A BR PI0811783 A2 BRPI0811783 A2 BR PI0811783A2
Authority
BR
Brazil
Prior art keywords
heteroaryl
methyl
receptor agonists
adrenergic receptor
bicyclic heterocyclic
Prior art date
Application number
BRPI0811783-7A2A
Other languages
English (en)
Inventor
Santosh C Sinha
Todd M Heidelbaugh
Ken Chow
Smita S Bhat
Phong X Nguyen
Michael E Garst
Original Assignee
Allergan Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allergan Inc filed Critical Allergan Inc
Publication of BRPI0811783A2 publication Critical patent/BRPI0811783A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BRPI0811783-7A2A 2007-05-23 2008-05-21 Compostos de ((heteroarila bicíclica)imidazolil)metil-heteroarila como agonistas dos receptores adrenérgicos. BRPI0811783A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US93978107P 2007-05-23 2007-05-23
PCT/US2008/064284 WO2008147786A1 (en) 2007-05-23 2008-05-21 ((bicylicheteroaryl) imidazolyl) methylheteroaryl compounds as adrenergic receptor agonists

Publications (1)

Publication Number Publication Date
BRPI0811783A2 true BRPI0811783A2 (pt) 2014-11-11

Family

ID=39679306

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0811783-7A2A BRPI0811783A2 (pt) 2007-05-23 2008-05-21 Compostos de ((heteroarila bicíclica)imidazolil)metil-heteroarila como agonistas dos receptores adrenérgicos.

Country Status (8)

Country Link
EP (1) EP2162450B1 (pt)
JP (1) JP5492075B2 (pt)
CN (1) CN101711242B (pt)
AU (1) AU2008256926B2 (pt)
BR (1) BRPI0811783A2 (pt)
CA (1) CA2687973C (pt)
RU (1) RU2472788C9 (pt)
WO (1) WO2008147786A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2816088A1 (en) * 2010-10-28 2012-05-03 Viamet Pharmaceuticals, Inc. Metalloenzyme inhibitor compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ221729A (en) * 1986-09-15 1989-07-27 Janssen Pharmaceutica Nv Imidazolyl methyl-substituted benzimidazole derivatives and pharmaceutical compositions
SE9302332D0 (sv) * 1993-07-06 1993-07-06 Ab Astra New compounds
TR200201297T2 (tr) * 1999-02-11 2002-06-21 Pfizer Products Inc. Antikanser maddeleri olarak faydalı heteroaril-ikame edilmiş kinolin-2-on türevleri.
US6610723B2 (en) * 2001-01-29 2003-08-26 Hoffmann-La Roche Inc. Imidazole derivatives

Also Published As

Publication number Publication date
EP2162450B1 (en) 2015-02-25
EP2162450A1 (en) 2010-03-17
JP2010528033A (ja) 2010-08-19
JP5492075B2 (ja) 2014-05-14
WO2008147786A1 (en) 2008-12-04
AU2008256926B2 (en) 2013-09-19
CN101711242B (zh) 2013-09-25
AU2008256926A1 (en) 2008-12-04
RU2009147158A (ru) 2011-06-27
CN101711242A (zh) 2010-05-19
CA2687973A1 (en) 2008-12-04
RU2472788C9 (ru) 2013-04-20
CA2687973C (en) 2015-04-07
RU2472788C2 (ru) 2013-01-20

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2385 DE 20-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

B350 Update of information on the portal [chapter 15.35 patent gazette]