BR0308987A - Agentes antidiabéticos - Google Patents
Agentes antidiabéticosInfo
- Publication number
- BR0308987A BR0308987A BR0308987-8A BR0308987A BR0308987A BR 0308987 A BR0308987 A BR 0308987A BR 0308987 A BR0308987 A BR 0308987A BR 0308987 A BR0308987 A BR 0308987A
- Authority
- BR
- Brazil
- Prior art keywords
- formula
- antidiabetic agents
- compounds
- preparing compounds
- useful
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/18—Drugs for disorders of the endocrine system of the parathyroid hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Urology & Nephrology (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
"AGENTES ANTIDIABéTICOS". A presente invenção refere-se a compostos de fórmula I: em que X, Y, B, E, J, K, L, Z, e R~ 9~-R~ 12~ têm qualquer dos significados aqui descritos, os seus sais farmaceuticamente aceitáveis, baixam os níveis de glicose e são úteis para o tratamento de doenças em mamíferos tais como a Diabetes Mellitus Não-Dependente de Insulina. Também descritas estão composições farmacêuticas, processos para preparação de compostos de fórmula (I) e intermediários úteis para preparação de compostos de fórmula I.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US36978702P | 2002-04-03 | 2002-04-03 | |
PCT/IB2003/001131 WO2003082276A1 (en) | 2002-04-03 | 2003-03-25 | Antidiabetic agents |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0308987A true BR0308987A (pt) | 2005-01-04 |
Family
ID=28675585
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0308987-8A BR0308987A (pt) | 2002-04-03 | 2003-03-25 | Agentes antidiabéticos |
Country Status (8)
Country | Link |
---|---|
US (1) | US6696474B2 (pt) |
EP (1) | EP1490060A1 (pt) |
JP (1) | JP2005527554A (pt) |
AU (1) | AU2003215803A1 (pt) |
BR (1) | BR0308987A (pt) |
CA (1) | CA2481258A1 (pt) |
MX (1) | MXPA04009499A (pt) |
WO (1) | WO2003082276A1 (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1838968A (zh) | 2003-08-08 | 2006-09-27 | 艾伯吉尼斯公司 | 针对甲状旁腺激素(pth)之抗体和其用途 |
US7318925B2 (en) * | 2003-08-08 | 2008-01-15 | Amgen Fremont, Inc. | Methods of use for antibodies against parathyroid hormone |
US8288438B2 (en) * | 2005-03-21 | 2012-10-16 | Metabolex, Inc. | Methods for avoiding edema in the treatment or prevention of PPARγ-responsive diseases, including cancer |
BRPI0711416A2 (pt) * | 2006-05-11 | 2011-11-01 | Sanofi Aventis | ácidos carboxìlicos substituìdos com 4,5-difenil pirimidinila, processo para a produção e uso dos mesmos como medicamentos |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SK161499A3 (en) * | 1998-03-30 | 2000-06-12 | Japan Tobacco Inc | Process for producing isooxazolidinedione compound |
KR100613175B1 (ko) | 1998-08-27 | 2006-08-17 | 오노 야꾸힝 고교 가부시키가이샤 | 카르복실산 유도체 및 그 유도체를 유효 성분으로서함유하는 약제 |
-
2003
- 2003-03-17 US US10/390,466 patent/US6696474B2/en not_active Expired - Fee Related
- 2003-03-25 BR BR0308987-8A patent/BR0308987A/pt not_active IP Right Cessation
- 2003-03-25 CA CA002481258A patent/CA2481258A1/en not_active Abandoned
- 2003-03-25 WO PCT/IB2003/001131 patent/WO2003082276A1/en not_active Application Discontinuation
- 2003-03-25 MX MXPA04009499A patent/MXPA04009499A/es unknown
- 2003-03-25 EP EP03745204A patent/EP1490060A1/en not_active Withdrawn
- 2003-03-25 JP JP2003579814A patent/JP2005527554A/ja active Pending
- 2003-03-25 AU AU2003215803A patent/AU2003215803A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
JP2005527554A (ja) | 2005-09-15 |
CA2481258A1 (en) | 2003-10-09 |
US20030220381A1 (en) | 2003-11-27 |
AU2003215803A1 (en) | 2003-10-13 |
EP1490060A1 (en) | 2004-12-29 |
MXPA04009499A (es) | 2005-01-25 |
US6696474B2 (en) | 2004-02-24 |
WO2003082276A1 (en) | 2003-10-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 4A, 5A E 6A ANUIDADES |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2051 DE 27/04/2010. |